CN1234680C - 新的成像剂及其前体与制备方法 - Google Patents

新的成像剂及其前体与制备方法 Download PDF

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Publication number
CN1234680C
CN1234680C CNB02122255XA CN02122255A CN1234680C CN 1234680 C CN1234680 C CN 1234680C CN B02122255X A CNB02122255X A CN B02122255XA CN 02122255 A CN02122255 A CN 02122255A CN 1234680 C CN1234680 C CN 1234680C
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CN
China
Prior art keywords
compound
formula
group
compound according
exists
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CNB02122255XA
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English (en)
Chinese (zh)
Other versions
CN1401629A (zh
Inventor
田中�明
井上登美夫
富吉胜美
D·J·杨
E·E·金
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Heavy Industries Ltd
University of Texas System
Original Assignee
Sumitomo Heavy Industries Ltd
University of Texas System
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Application filed by Sumitomo Heavy Industries Ltd, University of Texas System filed Critical Sumitomo Heavy Industries Ltd
Publication of CN1401629A publication Critical patent/CN1401629A/zh
Application granted granted Critical
Publication of CN1234680C publication Critical patent/CN1234680C/zh
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/20—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals substituted additionally by nitrogen atoms, e.g. tryptophane
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
CNB02122255XA 2001-06-04 2002-06-04 新的成像剂及其前体与制备方法 Expired - Fee Related CN1234680C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/872156 2001-06-04
US09/872,156 US6824760B2 (en) 2001-06-04 2001-06-04 Imaging agents, precursors thereof and methods of manufacture

Publications (2)

Publication Number Publication Date
CN1401629A CN1401629A (zh) 2003-03-12
CN1234680C true CN1234680C (zh) 2006-01-04

Family

ID=25358962

Family Applications (1)

Application Number Title Priority Date Filing Date
CNB02122255XA Expired - Fee Related CN1234680C (zh) 2001-06-04 2002-06-04 新的成像剂及其前体与制备方法

Country Status (5)

Country Link
US (1) US6824760B2 (https=)
JP (1) JP2003064046A (https=)
KR (1) KR100483650B1 (https=)
CN (1) CN1234680C (https=)
TW (1) TWI244925B (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060115426A1 (en) * 2004-08-11 2006-06-01 Weichert Jamey P Methods of detecting breast cancer, brain cancer, and pancreatic cancer
US8845999B2 (en) * 2005-05-23 2014-09-30 The Regents Of The University Of California Tracers for monitoring the activity of sodium/glucose cotransporters in health and disease
WO2008015392A1 (en) 2006-08-03 2008-02-07 Hammersmith Imanet Limited Fluoride drying method
WO2012025464A1 (en) 2010-08-24 2012-03-01 Bayer Pharma Aktiengesellschaft Fluorodeuteriomethyl tyrosine derivatives
GB201021530D0 (en) * 2010-12-20 2011-02-02 Ge Healthcare Ltd Purification of precursor compound by crystallisation
EP2520557A1 (en) * 2011-05-03 2012-11-07 Bayer Pharma Aktiengesellschaft Novel precursors of glutamate derivatives
WO2015152128A1 (ja) * 2014-03-31 2015-10-08 長瀬産業株式会社 アミノ酸前駆体、アミノ酸およびその製造方法、ならびに該アミノ酸を用いたｐｅｔ診断用トレーサー

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3800302A1 (de) * 1988-01-08 1989-07-27 Kernforschungsanlage Juelich Radiohalogentyrosinderivate, deren herstellung und verwendung

Also Published As

Publication number Publication date
US6824760B2 (en) 2004-11-30
KR100483650B1 (ko) 2005-04-18
TWI244925B (en) 2005-12-11
CN1401629A (zh) 2003-03-12
KR20020092818A (ko) 2002-12-12
JP2003064046A (ja) 2003-03-05
US20030124059A1 (en) 2003-07-03

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Legal Events

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C06 Publication
PB01 Publication
C14 Grant of patent or utility model
GR01 Patent grant
CF01 Termination of patent right due to non-payment of annual fee

Granted publication date: 20060104

Termination date: 20160604

CF01 Termination of patent right due to non-payment of annual fee