JP2003064046A - 新造影剤、その前駆体、及び、製造方法 - Google Patents

新造影剤、その前駆体、及び、製造方法

Info

Publication number
JP2003064046A
JP2003064046A JP2002161471A JP2002161471A JP2003064046A JP 2003064046 A JP2003064046 A JP 2003064046A JP 2002161471 A JP2002161471 A JP 2002161471A JP 2002161471 A JP2002161471 A JP 2002161471A JP 2003064046 A JP2003064046 A JP 2003064046A
Authority
JP
Japan
Prior art keywords
group
compound
compound according
formula
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002161471A
Other languages
English (en)
Japanese (ja)
Other versions
JP2003064046A5 (https=
Inventor
Akira Tanaka
明 田中
Tomio Inoue
登美夫 井上
Katsumi Tomiyoshi
勝美 冨吉
David J Yang
ジェイ．ヤン デイビッド
E Edmund Kim
キム イー．エドモンド
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sumitomo Heavy Industries Ltd
MD Anderson Cancer Center
Original Assignee
Sumitomo Heavy Industries Ltd
MD Anderson Cancer Center
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Heavy Industries Ltd, MD Anderson Cancer Center filed Critical Sumitomo Heavy Industries Ltd
Publication of JP2003064046A publication Critical patent/JP2003064046A/ja
Publication of JP2003064046A5 publication Critical patent/JP2003064046A5/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/20—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals substituted additionally by nitrogen atoms, e.g. tryptophane
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
JP2002161471A 2001-06-04 2002-06-03 新造影剤、その前駆体、及び、製造方法 Pending JP2003064046A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/872156 2001-06-04
US09/872,156 US6824760B2 (en) 2001-06-04 2001-06-04 Imaging agents, precursors thereof and methods of manufacture

Publications (2)

Publication Number Publication Date
JP2003064046A true JP2003064046A (ja) 2003-03-05
JP2003064046A5 JP2003064046A5 (https=) 2008-02-14

Family

ID=25358962

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002161471A Pending JP2003064046A (ja) 2001-06-04 2002-06-03 新造影剤、その前駆体、及び、製造方法

Country Status (5)

Country Link
US (1) US6824760B2 (https=)
JP (1) JP2003064046A (https=)
KR (1) KR100483650B1 (https=)
CN (1) CN1234680C (https=)
TW (1) TWI244925B (https=)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015152128A1 (ja) * 2014-03-31 2015-10-08 長瀬産業株式会社 アミノ酸前駆体、アミノ酸およびその製造方法、ならびに該アミノ酸を用いたｐｅｔ診断用トレーサー
JP2017078066A (ja) * 2011-05-03 2017-04-27 ピラマル イメージング ソシエテ アノニム グルタミン酸誘導体の新規前駆体

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060115426A1 (en) * 2004-08-11 2006-06-01 Weichert Jamey P Methods of detecting breast cancer, brain cancer, and pancreatic cancer
US8845999B2 (en) * 2005-05-23 2014-09-30 The Regents Of The University Of California Tracers for monitoring the activity of sodium/glucose cotransporters in health and disease
WO2008015392A1 (en) 2006-08-03 2008-02-07 Hammersmith Imanet Limited Fluoride drying method
WO2012025464A1 (en) 2010-08-24 2012-03-01 Bayer Pharma Aktiengesellschaft Fluorodeuteriomethyl tyrosine derivatives
GB201021530D0 (en) * 2010-12-20 2011-02-02 Ge Healthcare Ltd Purification of precursor compound by crystallisation

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3800302A1 (de) * 1988-01-08 1989-07-27 Kernforschungsanlage Juelich Radiohalogentyrosinderivate, deren herstellung und verwendung

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2017078066A (ja) * 2011-05-03 2017-04-27 ピラマル イメージング ソシエテ アノニム グルタミン酸誘導体の新規前駆体
WO2015152128A1 (ja) * 2014-03-31 2015-10-08 長瀬産業株式会社 アミノ酸前駆体、アミノ酸およびその製造方法、ならびに該アミノ酸を用いたｐｅｔ診断用トレーサー

Also Published As

Publication number Publication date
US6824760B2 (en) 2004-11-30
KR100483650B1 (ko) 2005-04-18
TWI244925B (en) 2005-12-11
CN1401629A (zh) 2003-03-12
KR20020092818A (ko) 2002-12-12
US20030124059A1 (en) 2003-07-03
CN1234680C (zh) 2006-01-04

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