CN106573939B - 用于治疗呼吸道合胞病毒感染的噻吩并[3,2-d]嘧啶、呋喃并[3,2-d]嘧啶和吡咯并[3,2-d]嘧啶 - Google Patents

用于治疗呼吸道合胞病毒感染的噻吩并[3,2-d]嘧啶、呋喃并[3,2-d]嘧啶和吡咯并[3,2-d]嘧啶 Download PDF

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CN106573939B
CN106573939B CN201580041342.0A CN201580041342A CN106573939B CN 106573939 B CN106573939 B CN 106573939B CN 201580041342 A CN201580041342 A CN 201580041342A CN 106573939 B CN106573939 B CN 106573939B
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CN106573939A (zh
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M.O.H.克拉克
R.L.马克曼
D.西格尔
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Gilead Sciences Inc
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    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
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    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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CN201580041342.0A 2014-07-28 2015-07-22 用于治疗呼吸道合胞病毒感染的噻吩并[3,2-d]嘧啶、呋喃并[3,2-d]嘧啶和吡咯并[3,2-d]嘧啶 Active CN106573939B (zh)

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US201462029896P 2014-07-28 2014-07-28
US62/029,896 2014-07-28
PCT/US2015/041574 WO2016018697A1 (en) 2014-07-28 2015-07-22 Thieno [3,2-d] pyrimidine, furo [3,2,d] pyrimidine, and pyrrolo [3,2-d] pyrimidines useful for treating respiratory syncitial virus infections

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JP6991188B2 (ja) 2022-01-12
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