CN106008583A - 含硼的小分子 - Google Patents
含硼的小分子 Download PDFInfo
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- CN106008583A CN106008583A CN201610328000.3A CN201610328000A CN106008583A CN 106008583 A CN106008583 A CN 106008583A CN 201610328000 A CN201610328000 A CN 201610328000A CN 106008583 A CN106008583 A CN 106008583A
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Classifications
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- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
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- C—CHEMISTRY; METALLURGY
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- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
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- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H23/00—Compounds containing boron, silicon or a metal, e.g. chelates or vitamin B12
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Enzymes And Modification Thereof (AREA)
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| US75522705P | 2005-12-30 | 2005-12-30 | |
| US60/755,227 | 2005-12-30 | ||
| PCT/US2006/005542 WO2006089067A2 (en) | 2005-02-16 | 2006-02-16 | Boron-containing small molecules |
| USPCT/US2006/05542 | 2006-02-16 | ||
| US11/357,687 US7582621B2 (en) | 2005-02-16 | 2006-02-16 | Boron-containing small molecules |
| US11/357,687 | 2006-02-16 | ||
| US74636106P | 2006-05-03 | 2006-05-03 | |
| US60/746,361 | 2006-05-03 | ||
| CNA2006800536192A CN101505603A (zh) | 2005-12-30 | 2006-08-16 | 含硼的小分子 |
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| CN201610328016.4A Pending CN106008571A (zh) | 2005-12-30 | 2006-08-16 | 含硼的小分子 |
| CN201610327999.XA Pending CN105949230A (zh) | 2005-12-30 | 2006-08-16 | 含硼的小分子 |
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| CN201610327999.XA Pending CN105949230A (zh) | 2005-12-30 | 2006-08-16 | 含硼的小分子 |
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| CN106008583A (zh) | 2005-12-30 | 2016-10-12 | 安纳考尔医药公司 | 含硼的小分子 |
| BRPI0708051A2 (pt) * | 2006-02-16 | 2011-05-17 | Anacor Pharmaceuticals Inc | moléculas pequenas contendo boro como agentes antiflamatórios |
| JP2009536660A (ja) * | 2006-05-02 | 2009-10-15 | アナコール ファーマシューティカルズ，インコーポレイテッド | 加水分解耐性ホウ素含有治療剤及びその使用方法 |
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| JO3396B1 (ar) | 2007-06-20 | 2019-10-20 | Anacor Pharmaceuticals Inc | جزيئات صغيرة تحتوي على البورون |
| US20090175810A1 (en) | 2008-01-03 | 2009-07-09 | Gareth Winckle | Compositions and methods for treating diseases of the nail |
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2016
- 2016-02-17 US US15/046,322 patent/US9566289B2/en not_active Expired - Fee Related
- 2016-03-11 US US15/068,352 patent/US9549938B2/en not_active Expired - Fee Related
- 2016-04-05 US US15/091,394 patent/US9572823B2/en not_active Expired - Fee Related
- 2016-04-20 US US15/134,286 patent/US9566290B2/en not_active Expired - Fee Related
- 2016-11-18 US US15/355,393 patent/US20170066787A1/en not_active Abandoned
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040259842A1 (en) * | 2001-10-11 | 2004-12-23 | Katsuhiko Mikoshiba | Intracellular calcuim concentration increase inhibitors |
Non-Patent Citations (3)
| Title |
|---|
| HAYNES, R. R ET AL.,: "Arylboronic acids. VIII. Reactions of boronophthalide", 《 JOURNAL OF ORGANIC CHEMISTRY》 * |
| KENJI OSHIMA ET AL.,: "Regiospecific Glycosidation of Unprotected Sugars via Arylboronic Activation", 《J. AM. CHEM. SOC.》 * |
| MORTON, R. K.: ""Substrate specificity and inhibition of alkaline phosphatases of cow milk and calf intestinal mucosa"", 《BIOCHEMICAL JOURNAL》 * |
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