CN105228997B - Carm1抑制剂及其用途 - Google Patents

Carm1抑制剂及其用途 Download PDF

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Publication number
CN105228997B
CN105228997B CN201480020614.4A CN201480020614A CN105228997B CN 105228997 B CN105228997 B CN 105228997B CN 201480020614 A CN201480020614 A CN 201480020614A CN 105228997 B CN105228997 B CN 105228997B
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optionally substituted
certain embodiments
alkyl
compound
hydrogen
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CN105228997A (zh
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理查德·切兹沃思
奥斯卡·米格尔·莫拉代
吉迪恩·夏皮罗
雷·金
罗伯特·E·巴比尼
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Epizyme Inc
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CN201480020614.4A 2013-03-15 2014-03-14 Carm1抑制剂及其用途 Active CN105228997B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201361794442P 2013-03-15 2013-03-15
US61/794,442 2013-03-15
US201461937333P 2014-02-07 2014-02-07
US61/937,333 2014-02-07
PCT/US2014/028463 WO2014144169A1 (en) 2013-03-15 2014-03-14 Carm1 inhibitors and uses thereof

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CN105228997A CN105228997A (zh) 2016-01-06
CN105228997B true CN105228997B (zh) 2018-03-27

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US (6) US9738651B2 (enExample)
EP (1) EP2970219B1 (enExample)
JP (2) JP2016519078A (enExample)
KR (1) KR20160003647A (enExample)
CN (1) CN105228997B (enExample)
AU (2) AU2014227775B2 (enExample)
BR (1) BR112015022787A2 (enExample)
CA (1) CA2903813C (enExample)
EA (1) EA201591532A1 (enExample)
IL (1) IL241370A0 (enExample)
MX (1) MX2015012803A (enExample)
SG (1) SG11201507070XA (enExample)
WO (1) WO2014144169A1 (enExample)

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CN110382482A (zh) 2017-01-26 2019-10-25 亚瑞克西斯制药公司 稠合的杂-杂二环化合物及其使用方法
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