CN104884062B - N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物 - Google Patents

N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物 Download PDF

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Publication number
CN104884062B
CN104884062B CN201380068060.0A CN201380068060A CN104884062B CN 104884062 B CN104884062 B CN 104884062B CN 201380068060 A CN201380068060 A CN 201380068060A CN 104884062 B CN104884062 B CN 104884062B
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China
Prior art keywords
compound
methyl
acid
bacterium
plants
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Expired - Fee Related
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Chinese (zh)
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CN104884062A (zh
Inventor
B·洛尔斯巴赫
W·J·欧文
C·姚
L·施特尔策
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Adama Makhteshim Ltd
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Adama Makhteshim Ltd
Dow AgroSciences LLC
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/30—Derivatives containing the group >N—CO—N aryl or >N—CS—N—aryl
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Toxicology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CN201380068060.0A 2012-12-28 2013-12-23 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物 Expired - Fee Related CN104884062B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261746837P 2012-12-28 2012-12-28
US61/746,837 2012-12-28
PCT/US2013/077533 WO2014105841A1 (en) 2012-12-28 2013-12-23 N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxamides derivatives

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Publication Number Publication Date
CN104884062A CN104884062A (zh) 2015-09-02
CN104884062B true CN104884062B (zh) 2018-11-06

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US (2) US9321734B2 (enExample)
EP (1) EP2945634A4 (enExample)
JP (1) JP6258969B2 (enExample)
KR (1) KR20150100869A (enExample)
CN (1) CN104884062B (enExample)
AU (1) AU2013370490B2 (enExample)
BR (1) BR102013033716B1 (enExample)
CA (1) CA2894510A1 (enExample)
CL (1) CL2015001863A1 (enExample)
EC (1) ECSP15032846A (enExample)
GT (1) GT201500195A (enExample)
HK (1) HK1215376A1 (enExample)
IL (1) IL239563B (enExample)
MX (1) MX2015008444A (enExample)
RU (1) RU2015131149A (enExample)
UA (1) UA117743C2 (enExample)
WO (1) WO2014105841A1 (enExample)
ZA (1) ZA201504197B (enExample)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9271497B2 (en) * 2012-12-28 2016-03-01 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives
RU2015131149A (ru) 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные
RU2638556C2 (ru) 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
EP2938191B1 (en) 2012-12-28 2018-01-31 Dow AgroSciences LLC Synergistic fungicidal mixtures for fungal control in cereals
MX381341B (es) 2012-12-31 2025-03-12 Adama Makhteshim Ltd Derivados de 3-alquil-5-fluoro-4-sustituido-imino-3,4-dihidropirimidin-2(1h)-ona como fungicidas.
AU2014373853A1 (en) 2013-12-31 2016-08-11 Adama Makhteshim Ltd. Synergistic fungicidal mixtures and compositions for fungal control
EA036389B1 (ru) 2013-12-31 2020-11-03 Адама Мактешим Лтд. 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения
NZ732812A (en) 2014-12-30 2019-01-25 Dow Agrosciences Llc Use of picolinamides and other compounds as fungicides
WO2016109288A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Use of picolinamide compounds with fungicidal activity
EP3240773B9 (en) 2014-12-30 2021-01-13 Dow AgroSciences LLC Picolinamide compounds with fungicidal activity
NZ732657A (en) 2014-12-30 2019-01-25 Dow Agrosciences Llc Picolinamides with fungicidal activity and other related compounds
MX2017008418A (es) 2014-12-30 2017-09-28 Dow Agrosciences Llc Picolinamidas con actividad fungicida.
CN110573014B (zh) * 2017-04-27 2022-02-11 Upl有限公司 杀真菌组合
TWI774761B (zh) 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 用於穀物中的真菌防治之協同性混合物
CA3062074A1 (en) 2017-05-02 2018-11-08 Dow Agrosciences Llc Use of an acyclic picolinamide compound as a fungicide for fungal diseases on turfgrasses
TW201842851A (zh) 2017-05-02 2018-12-16 美商陶氏農業科學公司 用於穀類中的真菌防治之協同性混合物
US11632954B2 (en) 2017-07-17 2023-04-25 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1 -tosyl-3,4-dihydropyrimidin-2-one
BR102019004480B1 (pt) 2018-03-08 2023-03-28 Dow Agrosciences Llc Picolinamidas como fungicidas
KR102745084B1 (ko) * 2018-09-27 2024-12-23 에프엠씨 코포레이션 피리다지논 제초제 및 제초제 제조에 사용되는 피리다지논 중간체
EP3866597A4 (en) 2018-10-15 2022-06-29 Corteva Agriscience LLC Methods for sythesis of oxypicolinamides
BR112021008755A2 (pt) 2018-11-05 2021-08-10 Adama Makhteshim Ltd. misturas e composições contendo 5-fluoro-4-imino-3- metil-1-tosil-3,4-dihidropirimidina-2-ona, e métodos de uso.
EP4034529A1 (en) 2019-09-23 2022-08-03 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine -(1h)-one
EP4044811A4 (en) 2019-10-18 2023-09-27 Corteva Agriscience LLC METHOD FOR SYNTHESIS OF PICOLINAMIDS

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110034492A1 (en) * 2009-08-07 2011-02-10 Dow Agrosciences Llc N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
US20110263627A1 (en) * 2010-04-26 2011-10-27 Dow Agrosciences Llc N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives

Family Cites Families (63)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH421973A (de) 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
DE1214459B (de) 1964-03-19 1966-04-14 Koellisch Geb Zuendsteinauswechselvorrichtung
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3635977A (en) 1969-11-03 1972-01-18 American Cyanamid Co Certain 6-trifluoromethylcytosines and thiocytosines their synthesis and their use in the synthesis of uracisls and thiouracil
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
US4009272A (en) 1971-10-23 1977-02-22 Bayer Aktiengesellschaft Penicillins
CH579057A5 (enExample) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
JPS60123486A (ja) 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンｓおよびその製法
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
DE58908159D1 (de) 1988-03-09 1994-09-15 Ciba Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten.
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
DE69618959T2 (de) 1995-07-05 2002-08-29 E.I. Du Pont De Nemours And Co., Wilmington Pyrimidone und ihre verwendug als fungizide
US6072051A (en) 1995-11-02 2000-06-06 Chong Kun Dang Corp. Nucleoside derivatives and process for preparing the same
DK0888359T3 (da) 1996-03-11 2002-08-12 Syngenta Participations Ag Pyrimidin-4-on-derivat som pesticid
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
JP3495636B2 (ja) 1999-03-25 2004-02-09 株式会社マキタ 充電装置
US20020108099A1 (en) 2000-10-11 2002-08-08 Charles Paclat Method for developing business components
HUP0301363A2 (hu) 2000-10-13 2005-12-28 Shire Biochem Inc. Javított intercelluláris bejuttathatóságú dioxolán analógok
US7914799B2 (en) 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
AU2003274652A1 (en) 2002-10-23 2004-05-13 Obetherapy Biotechnology Compounds, compositions and methods for modulating fat metabolism
US20080269238A1 (en) 2004-04-01 2008-10-30 Takeda Pharmaceutical Company Limited Thiazolopyrimidine Derivative
JP4887500B2 (ja) 2004-09-16 2012-02-29 国立大学法人岐阜大学 ヌクレオシド類似体またはその塩
JP4548619B2 (ja) 2004-09-17 2010-09-22 株式会社安川電機 モータ制御装置
EP1871383B1 (en) 2005-04-04 2017-11-15 Intersect ENT, Inc. Device and methods for treating paranasal sinus conditions
TWI402034B (zh) 2005-07-28 2013-07-21 Dow Agrosciences Llc 具有被層狀液晶覆膜包覆之油球之水包油乳化劑之農用組成物
US20090163567A1 (en) 2005-11-22 2009-06-25 Ishihara Sangyo Kaisha, Ltd Germicide composition for agricultural and gardening applications and method for controlling plant disease
EP2044086A2 (en) 2006-06-30 2009-04-08 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
US20100029483A1 (en) 2006-10-16 2010-02-04 Rhodia Inc. Agricultural adjuvant compositions, pesticide compositions, and methods for using such compositions
US8093245B2 (en) 2006-12-14 2012-01-10 Lexicon Pharmaceuticals, Inc. 4-amino-1H-pyrimidin-2-one based compounds, compositions comprising them and methods of their use
WO2008083465A1 (en) 2007-01-08 2008-07-17 University Health Network Pyrimidine derivatives as anticancer agents
AU2008219166B2 (en) 2007-02-16 2013-05-16 Amgen Inc. Nitrogen-containing heterocyclyl ketones and their use as c-Met inhibitors
CA2683941C (en) 2007-04-27 2014-08-12 Asubio Pharma Co., Ltd. Nitrogen-containing six-membered aromatic ring derivatives and pharmaceutical products containing the same
US8373338B2 (en) 2008-10-22 2013-02-12 General Electric Company Enhanced color contrast light source at elevated color temperatures
PL2252594T3 (pl) 2008-01-22 2016-01-29 Dow Agrosciences Llc Pochodne 4-amino-5-fluoropirymidyny jako fungicydy
US20100284959A1 (en) 2008-01-23 2010-11-11 Gene Arrest Ltd. Sequence specific double-stranded dna/rna binding compounds and uses thereof
WO2010006697A2 (en) 2008-06-30 2010-01-21 Tibotec Pharmaceuticals Powders for reconstitution
CA2731332A1 (en) 2008-08-01 2010-04-29 Zoltan L. Benko Use of 5-fluorocytosine as a fungicide
WO2010033198A2 (en) 2008-09-17 2010-03-25 Sri International Analogs of indole-3-carbinol and their use as agents against infection
ME02254B (me) 2009-01-23 2015-12-31 Euro Celtique Sa Derivati hidroksamske kiseline
JP5784603B2 (ja) 2009-08-07 2015-09-24 ダウ アグロサイエンシィズ エルエルシー Ｎ１−スルホニル−５−フルオロピリミジノン誘導体
UA112284C2 (uk) 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні 5-фторпіримідинону
UA106889C2 (uk) 2009-08-07 2014-10-27 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-ацил-5-фторпіримідинону
JP5818791B2 (ja) 2009-08-07 2015-11-18 ダウ アグロサイエンシィズ エルエルシー ５−フルオロ−２−オキソピリミジン−１（２ｈ）−カルボキシレート誘導体
BR112012007975A2 (pt) 2009-10-07 2016-03-29 Dow Agrosciences Llc composição fungicida sinergística contendo 5-fluorocitosina para controle fúngico em cereais
US8522020B2 (en) 2009-12-03 2013-08-27 Osocad Remote Limited Liability Company System and method for validating a location of an untrusted device
US20120208700A1 (en) 2011-02-11 2012-08-16 Dow Agrosciences Llc Stable agrochemical oil dispersions
AU2011358608B2 (en) 2011-02-11 2016-04-14 Dow Agrosciences Llc Stable agrochemical oil dispersions
US8658660B2 (en) 2011-08-17 2014-02-25 Dow Agrosciences, Llc. 5-fluoro-4-imino-3,4-dihydropyrimidin-2-(1H)-ones derivatives
WO2013113781A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds i
JP6001793B2 (ja) 2012-11-07 2016-10-05 トヨタ自動車株式会社 燃料電池用触媒の製造方法
RU2638556C2 (ru) 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
US9271497B2 (en) 2012-12-28 2016-03-01 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives
RU2015131149A (ru) 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные
MX381341B (es) 2012-12-31 2025-03-12 Adama Makhteshim Ltd Derivados de 3-alquil-5-fluoro-4-sustituido-imino-3,4-dihidropirimidin-2(1h)-ona como fungicidas.
FR3008090B1 (fr) 2013-07-03 2015-07-31 Robertet Sa Nouveau procede de synthese de la khusimone
AU2014373853A1 (en) 2013-12-31 2016-08-11 Adama Makhteshim Ltd. Synergistic fungicidal mixtures and compositions for fungal control
EA036389B1 (ru) 2013-12-31 2020-11-03 Адама Мактешим Лтд. 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110034492A1 (en) * 2009-08-07 2011-02-10 Dow Agrosciences Llc N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
US20110263627A1 (en) * 2010-04-26 2011-10-27 Dow Agrosciences Llc N3-substituted-n1-sulfonyl-5-fluoropyrimidinone derivatives

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BR102013033716B1 (pt) 2019-05-14
US20150353506A1 (en) 2015-12-10
CA2894510A1 (en) 2014-07-03
MX2015008444A (es) 2015-09-23
AU2013370490A1 (en) 2015-07-02
BR102013033716A2 (pt) 2015-11-10
UA117743C2 (uk) 2018-09-25
US9840475B2 (en) 2017-12-12
CN104884062A (zh) 2015-09-02
WO2014105841A1 (en) 2014-07-03
IL239563B (en) 2018-02-28
IL239563A0 (en) 2015-08-31
ZA201504197B (en) 2017-04-26
RU2015131149A (ru) 2017-02-03
JP6258969B2 (ja) 2018-01-10
CL2015001863A1 (es) 2015-10-02
AU2013370490B2 (en) 2018-05-10
GT201500195A (es) 2016-02-14
US9321734B2 (en) 2016-04-26
EP2945634A4 (en) 2016-05-25
ECSP15032846A (es) 2016-01-29
US20160198711A1 (en) 2016-07-14
EP2945634A1 (en) 2015-11-25
JP2016505605A (ja) 2016-02-25
KR20150100869A (ko) 2015-09-02
HK1215376A1 (zh) 2016-08-26

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