CN102552162A - 制备含有可压性差的治疗性化合物的组合物的挤压方法 - Google Patents
制备含有可压性差的治疗性化合物的组合物的挤压方法 Download PDFInfo
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- CN102552162A CN102552162A CN2011103445944A CN201110344594A CN102552162A CN 102552162 A CN102552162 A CN 102552162A CN 2011103445944 A CN2011103445944 A CN 2011103445944A CN 201110344594 A CN201110344594 A CN 201110344594A CN 102552162 A CN102552162 A CN 102552162A
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- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (4)
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| US67958705P | 2005-05-10 | 2005-05-10 | |
| US60/679,587 | 2005-05-10 | ||
| US69315505P | 2005-06-23 | 2005-06-23 | |
| US60/693,155 | 2005-06-23 |
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| CN200680014443XA Division CN101166517B (zh) | 2005-05-10 | 2006-05-08 | 制备含有可压性差的治疗性化合物的组合物的挤压方法 |
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| CN102552162A true CN102552162A (zh) | 2012-07-11 |
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| EP (1) | EP1881819A1 (https=) |
| JP (1) | JP5400377B2 (https=) |
| KR (2) | KR20080007357A (https=) |
| CN (1) | CN102552162A (https=) |
| AU (2) | AU2006244213B2 (https=) |
| BR (1) | BRPI0608609A2 (https=) |
| CA (1) | CA2607624A1 (https=) |
| IL (1) | IL186456A0 (https=) |
| MA (1) | MA29465B1 (https=) |
| MX (1) | MX2007014041A (https=) |
| NO (1) | NO20076298L (https=) |
| NZ (2) | NZ562304A (https=) |
| RU (1) | RU2405539C2 (https=) |
| TN (1) | TNSN07415A1 (https=) |
| WO (1) | WO2006122021A1 (https=) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2024047555A1 (en) * | 2022-08-31 | 2024-03-07 | Sacmi Cooperativa Meccanici Imola Societa' Cooperativa | Method and apparatus for making solid medicines |
| CN118234387A (zh) * | 2021-11-16 | 2024-06-21 | 帝斯曼知识产权资产管理有限公司 | 包含封装的活性成分的颗粒 |
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| DE102005005449A1 (de) | 2005-02-04 | 2006-08-10 | Grünenthal GmbH | Verfahren zur Herstellung einer gegen Missbrauch gesicherten Darreichungsform |
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| MX2010011962A (es) * | 2008-04-30 | 2010-11-30 | Novartis Ag | Proceso continuo para hacer composiciones farmaceuticas. |
| BRPI0913843A2 (pt) * | 2008-07-03 | 2015-10-20 | Novartis Ag | processo de granulação por fusão |
| WO2011009602A1 (en) | 2009-07-22 | 2011-01-27 | Grünenthal GmbH | Hot-melt extruded controlled release dosage form |
| TWI473628B (zh) | 2009-07-22 | 2015-02-21 | 用於對氧化敏感之類鴉片藥劑之抗破壞劑型 | |
| WO2012028318A1 (en) | 2010-09-02 | 2012-03-08 | Grünenthal GmbH | Tamper resistant dosage form comprising an anionic polymer |
| CA2808219C (en) | 2010-09-02 | 2019-05-14 | Gruenenthal Gmbh | Tamper resistant dosage form comprising inorganic salt |
| AU2012289764B2 (en) | 2011-07-29 | 2017-03-02 | Grünenthal GmbH | Tamper-resistant tablet providing immediate drug release |
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| US20130225697A1 (en) | 2012-02-28 | 2013-08-29 | Grunenthal Gmbh | Tamper-resistant dosage form comprising pharmacologically active compound and anionic polymer |
| PL2838512T3 (pl) | 2012-04-18 | 2018-12-31 | Grünenthal GmbH | Farmaceutyczna postać dawkowania odporna na niewłaściwe użycie i odporna na uderzeniowe uwalnianie dawki |
| US10064945B2 (en) | 2012-05-11 | 2018-09-04 | Gruenenthal Gmbh | Thermoformed, tamper-resistant pharmaceutical dosage form containing zinc |
| GB201218012D0 (en) * | 2012-10-08 | 2012-11-21 | Jagotec Ag | Dosage forms |
| AU2014273227B2 (en) | 2013-05-29 | 2019-08-15 | Grunenthal Gmbh | Tamper-resistant dosage form containing one or more particles |
| JP6466417B2 (ja) | 2013-05-29 | 2019-02-06 | グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング | 二峰性放出プロファイルを有する改変防止（ｔａｍｐｅｒ−ｒｅｓｉｓｔａｎｔ）剤形 |
| JP6449871B2 (ja) | 2013-07-12 | 2019-01-09 | グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング | エチレン−酢酸ビニルポリマーを含有する改変防止剤形 |
| CA3042642A1 (en) | 2013-08-12 | 2015-02-19 | Pharmaceutical Manufacturing Research Services, Inc. | Extruded immediate release abuse deterrent pill |
| EP3073994A1 (en) | 2013-11-26 | 2016-10-05 | Grünenthal GmbH | Preparation of a powdery pharmaceutical composition by means of cryo-milling |
| US10172797B2 (en) | 2013-12-17 | 2019-01-08 | Pharmaceutical Manufacturing Research Services, Inc. | Extruded extended release abuse deterrent pill |
| US9492444B2 (en) | 2013-12-17 | 2016-11-15 | Pharmaceutical Manufacturing Research Services, Inc. | Extruded extended release abuse deterrent pill |
| EP3142646A1 (en) | 2014-05-12 | 2017-03-22 | Grünenthal GmbH | Tamper resistant immediate release capsule formulation comprising tapentadol |
| EA201692388A1 (ru) | 2014-05-26 | 2017-05-31 | Грюненталь Гмбх | Лекарственная форма в виде множества частиц, защищенная от вызываемого этанолом сброса дозы |
| CA2955229C (en) | 2014-07-17 | 2020-03-10 | Pharmaceutical Manufacturing Research Services, Inc. | Immediate release abuse deterrent liquid fill dosage form |
| WO2016064873A1 (en) | 2014-10-20 | 2016-04-28 | Pharmaceutical Manufacturing Research Services, Inc. | Extended release abuse deterrent liquid fill dosage form |
| CA2983640A1 (en) | 2015-04-24 | 2016-10-27 | Grunenthal Gmbh | Tamper-resistant fixed dose combination providing fast release of two drugs from different particles |
| US20160310437A1 (en) | 2015-04-24 | 2016-10-27 | Grünenthal GmbH | Tamper-resistant fixed dose combination providing fast release of two drugs from particles |
| BR112017021475A2 (pt) | 2015-04-24 | 2018-07-10 | Gruenenthal Gmbh | forma de dosagem resistente à adulteração (tamper) com liberação imediata e resistência contra extração de solvente |
| MX2017013643A (es) | 2015-04-24 | 2018-03-08 | Gruenenthal Gmbh | Combinacion de dosis fija resistente a la manipulacion que proporciona una liberacion rapida de dos farmacos desde particulas y una matriz. |
| WO2017042325A1 (en) | 2015-09-10 | 2017-03-16 | Grünenthal GmbH | Protecting oral overdose with abuse deterrent immediate release formulations |
| DE102018010063A1 (de) | 2018-03-16 | 2019-09-19 | Ludwig-Maximilians-Universität München | Herstellung vesikulärer Phospholipid-Gele durch Schnecken-Extrusion |
| CN108888599B (zh) * | 2018-07-26 | 2021-06-08 | 国药集团致君（深圳）制药有限公司 | 双氯芬酸钠缓释组合物及其制备方法 |
| CN116887866A (zh) | 2020-12-03 | 2023-10-13 | 巴特尔纪念研究院 | 聚合物纳米颗粒和dna纳米结构组合物及用于非病毒递送的方法 |
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| US12441996B2 (en) | 2023-12-08 | 2025-10-14 | Battelle Memorial Institute | Use of DNA origami nanostructures for molecular information based data storage systems |
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| WO2007106182A2 (en) * | 2005-11-09 | 2007-09-20 | Novartis Ag | Process for making pharmaceutical compositions with a transient plasticizer |
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2006
- 2006-05-08 EP EP06759308A patent/EP1881819A1/en not_active Withdrawn
- 2006-05-08 CA CA002607624A patent/CA2607624A1/en not_active Abandoned
- 2006-05-08 KR KR1020077026095A patent/KR20080007357A/ko not_active Ceased
- 2006-05-08 KR KR1020137031633A patent/KR20130135403A/ko not_active Ceased
- 2006-05-08 NZ NZ562304A patent/NZ562304A/en not_active IP Right Cessation
- 2006-05-08 WO PCT/US2006/017708 patent/WO2006122021A1/en not_active Ceased
- 2006-05-08 CN CN2011103445944A patent/CN102552162A/zh active Pending
- 2006-05-08 RU RU2007145522/15A patent/RU2405539C2/ru not_active IP Right Cessation
- 2006-05-08 US US11/909,509 patent/US20100152299A1/en not_active Abandoned
- 2006-05-08 BR BRPI0608609-8A patent/BRPI0608609A2/pt not_active IP Right Cessation
- 2006-05-08 AU AU2006244213A patent/AU2006244213B2/en not_active Ceased
- 2006-05-08 MX MX2007014041A patent/MX2007014041A/es active IP Right Grant
- 2006-05-08 JP JP2008511233A patent/JP5400377B2/ja not_active Expired - Fee Related
- 2006-05-08 NZ NZ585116A patent/NZ585116A/en not_active IP Right Cessation
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- 2007-10-07 IL IL186456A patent/IL186456A0/en unknown
- 2007-11-09 TN TNP2007000415A patent/TNSN07415A1/en unknown
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- 2007-12-06 NO NO20076298A patent/NO20076298L/no not_active Application Discontinuation
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2010
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- 2011-11-30 US US13/307,864 patent/US20120077879A1/en not_active Abandoned
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN118234387A (zh) * | 2021-11-16 | 2024-06-21 | 帝斯曼知识产权资产管理有限公司 | 包含封装的活性成分的颗粒 |
| WO2024047555A1 (en) * | 2022-08-31 | 2024-03-07 | Sacmi Cooperativa Meccanici Imola Societa' Cooperativa | Method and apparatus for making solid medicines |
Also Published As
| Publication number | Publication date |
|---|---|
| EP1881819A1 (en) | 2008-01-30 |
| MA29465B1 (fr) | 2008-05-02 |
| AU2006244213A1 (en) | 2006-11-16 |
| RU2405539C2 (ru) | 2010-12-10 |
| JP2008540540A (ja) | 2008-11-20 |
| WO2006122021A1 (en) | 2006-11-16 |
| TNSN07415A1 (en) | 2009-03-17 |
| IL186456A0 (en) | 2008-01-20 |
| KR20080007357A (ko) | 2008-01-18 |
| KR20130135403A (ko) | 2013-12-10 |
| US20120077879A1 (en) | 2012-03-29 |
| US20100152299A1 (en) | 2010-06-17 |
| AU2010212296B2 (en) | 2011-06-16 |
| AU2006244213B2 (en) | 2010-05-13 |
| CA2607624A1 (en) | 2006-11-16 |
| MX2007014041A (es) | 2008-02-11 |
| NO20076298L (no) | 2007-12-06 |
| NZ585116A (en) | 2011-12-22 |
| BRPI0608609A2 (pt) | 2010-01-19 |
| NZ562304A (en) | 2010-06-25 |
| RU2007145522A (ru) | 2009-06-20 |
| JP5400377B2 (ja) | 2014-01-29 |
| AU2010212296A1 (en) | 2010-09-02 |
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