CN102281876A - 新型有效的他喷他多剂型 - Google Patents

新型有效的他喷他多剂型 Download PDF

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Publication number
CN102281876A
CN102281876A CN2009801538254A CN200980153825A CN102281876A CN 102281876 A CN102281876 A CN 102281876A CN 2009801538254 A CN2009801538254 A CN 2009801538254A CN 200980153825 A CN200980153825 A CN 200980153825A CN 102281876 A CN102281876 A CN 102281876A
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China
Prior art keywords
tapentadol
dosage form
antagonist
hours
pain
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN2009801538254A
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English (en)
Chinese (zh)
Inventor
R·塞沙
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gruenenthal GmbH
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Gruenenthal GmbH
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42634123&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN102281876(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gruenenthal GmbH filed Critical Gruenenthal GmbH
Publication of CN102281876A publication Critical patent/CN102281876A/zh
Pending legal-status Critical Current

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    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Otolaryngology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Transplantation (AREA)
  • Toxicology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
CN2009801538254A 2008-10-30 2009-10-29 新型有效的他喷他多剂型 Pending CN102281876A (zh)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US19762508P 2008-10-30 2008-10-30
US61/197625 2008-10-30
US20531209P 2009-01-21 2009-01-21
US61/205312 2009-01-21
US26863009P 2009-06-15 2009-06-15
US61/268630 2009-06-15
PCT/US2009/005866 WO2010096045A1 (en) 2008-10-30 2009-10-29 Novel and potent tapentadol dosage forms

Related Child Applications (1)

Application Number Title Priority Date Filing Date
CN201410398429.0A Division CN104257600A (zh) 2008-10-30 2009-10-29 新型有效的他喷他多剂型

Publications (1)

Publication Number Publication Date
CN102281876A true CN102281876A (zh) 2011-12-14

Family

ID=42634123

Family Applications (2)

Application Number Title Priority Date Filing Date
CN2009801538254A Pending CN102281876A (zh) 2008-10-30 2009-10-29 新型有效的他喷他多剂型
CN201410398429.0A Pending CN104257600A (zh) 2008-10-30 2009-10-29 新型有效的他喷他多剂型

Family Applications After (1)

Application Number Title Priority Date Filing Date
CN201410398429.0A Pending CN104257600A (zh) 2008-10-30 2009-10-29 新型有效的他喷他多剂型

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US (1) US9642801B2 (enExample)
EP (1) EP2352494B1 (enExample)
JP (2) JP6216489B2 (enExample)
KR (2) KR101806796B1 (enExample)
CN (2) CN102281876A (enExample)
AU (2) AU2009340504A1 (enExample)
BR (1) BRPI0921725A2 (enExample)
CA (1) CA2741984C (enExample)
CL (1) CL2011000967A1 (enExample)
CO (1) CO6382115A2 (enExample)
CY (1) CY1122269T1 (enExample)
DK (1) DK2352494T3 (enExample)
EC (2) ECSP11011016A (enExample)
ES (1) ES2758831T3 (enExample)
HR (1) HRP20191909T1 (enExample)
HU (1) HUE047438T2 (enExample)
IL (2) IL212523A0 (enExample)
LT (1) LT2352494T (enExample)
MX (1) MX2011004455A (enExample)
NZ (1) NZ592437A (enExample)
PE (3) PE20142368A1 (enExample)
PL (1) PL2352494T3 (enExample)
PT (1) PT2352494T (enExample)
RU (2) RU2599846C2 (enExample)
SI (1) SI2352494T1 (enExample)
WO (1) WO2010096045A1 (enExample)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103432107A (zh) * 2013-08-20 2013-12-11 安徽省先锋制药有限公司 一种盐酸他喷他多对乙酰氨基酚口腔崩解片及其制备方法
CN103655523A (zh) * 2013-12-24 2014-03-26 南京艾德凯腾生物医药有限责任公司 他喷他多组合物
CN105218386A (zh) * 2010-07-23 2016-01-06 格吕伦塔尔有限公司 3-(3-二甲基氨基-1-乙基-2-甲基-丙基)-苯酚的盐或共晶体
US9642801B2 (en) 2008-10-30 2017-05-09 Gruenenthal Gmbh And potent tapentadol dosage forms

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG175184A1 (en) * 2009-04-30 2011-12-29 Gruenenthal Gmbh Use of 1-phenyl-3-dimethylaminopropane compounds for treating rheumatoid pain
US10363251B2 (en) 2009-07-16 2019-07-30 Mallinckrodt Llc (+)-morphinans as antagonists of toll-like receptor 9 and therapeutic uses thereof
WO2011138037A2 (de) * 2010-05-05 2011-11-10 Ratiopharm Gmbh Festes tapentadol in nicht-kristalliner form
US9901540B2 (en) 2010-05-10 2018-02-27 Euro-Celtique S.A. Combination of active loaded granules with additional actives
EP2568968B1 (en) 2010-05-10 2017-07-12 Euro-Celtique S.A. Manufacturing of active-free granules and tablets comprising the same
SE1251371A1 (sv) 2010-05-10 2012-12-27 Euro Celtique Sa Farmaceutiska kompositioner innefattande hydromorfon och naloxon
WO2012008984A1 (en) * 2010-07-16 2012-01-19 Mallinckrodt Llc (+)-morphinans as antagonists of toll-like receptor 9 and therapeutic uses thereof
WO2012051246A1 (en) * 2010-10-12 2012-04-19 Ratiopharm Gmbh Tapentadol hydrobromide and crystalline forms thereof
KR102051800B1 (ko) * 2011-03-04 2019-12-04 그뤼넨탈 게엠베하 경구 투여를 위한 타펜타돌의 수성 약제학적 제형
CA2828637C (en) * 2011-03-04 2019-06-11 Grunenthal Gmbh Semisolid aqueous pharmaceutical composition containing tapentadol
PL2736501T3 (pl) * 2011-07-29 2018-06-29 Grünenthal GmbH Dooponowe lub nadtwardówkowe podawanie 3-[(1S,2S)-3-(dimetyloamino)-1-etylo-2-metylopropylo]fenolu
EP2606879A1 (en) * 2011-12-21 2013-06-26 Hexal AG Multiple unit pellet tablet formulation comprising an opioid
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