KR101806796B1 - 신규하고 강력한 타펜타돌 용량형 - Google Patents
신규하고 강력한 타펜타돌 용량형 Download PDFInfo
- Publication number
- KR101806796B1 KR101806796B1 KR1020177004316A KR20177004316A KR101806796B1 KR 101806796 B1 KR101806796 B1 KR 101806796B1 KR 1020177004316 A KR1020177004316 A KR 1020177004316A KR 20177004316 A KR20177004316 A KR 20177004316A KR 101806796 B1 KR101806796 B1 KR 101806796B1
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- South Korea
- Prior art keywords
- hours
- medicament
- antagonist
- administered
- dosage form
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
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- QVRBGKYLLCLCHL-UHFFFAOYSA-N CC1C=CC=C1 Chemical compound CC1C=CC=C1 QVRBGKYLLCLCHL-UHFFFAOYSA-N 0.000 description 1
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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- A—HUMAN NECESSITIES
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- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Dispersion Chemistry (AREA)
- Inorganic Chemistry (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Toxicology (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US19762508P | 2008-10-30 | 2008-10-30 | |
| US61/197,625 | 2008-10-30 | ||
| US20531209P | 2009-01-21 | 2009-01-21 | |
| US61/205,312 | 2009-01-21 | ||
| US26863009P | 2009-06-15 | 2009-06-15 | |
| US61/268,630 | 2009-06-15 | ||
| PCT/US2009/005866 WO2010096045A1 (en) | 2008-10-30 | 2009-10-29 | Novel and potent tapentadol dosage forms |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020117012188A Division KR101712339B1 (ko) | 2008-10-30 | 2009-10-29 | 신규하고 강력한 타펜타돌 용량형 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| KR20170020940A KR20170020940A (ko) | 2017-02-24 |
| KR101806796B1 true KR101806796B1 (ko) | 2017-12-08 |
Family
ID=42634123
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020117012188A Expired - Fee Related KR101712339B1 (ko) | 2008-10-30 | 2009-10-29 | 신규하고 강력한 타펜타돌 용량형 |
| KR1020177004316A Expired - Fee Related KR101806796B1 (ko) | 2008-10-30 | 2009-10-29 | 신규하고 강력한 타펜타돌 용량형 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020117012188A Expired - Fee Related KR101712339B1 (ko) | 2008-10-30 | 2009-10-29 | 신규하고 강력한 타펜타돌 용량형 |
Country Status (26)
| Country | Link |
|---|---|
| US (1) | US9642801B2 (enExample) |
| EP (1) | EP2352494B1 (enExample) |
| JP (2) | JP6216489B2 (enExample) |
| KR (2) | KR101712339B1 (enExample) |
| CN (2) | CN104257600A (enExample) |
| AU (2) | AU2009340504A1 (enExample) |
| BR (1) | BRPI0921725A2 (enExample) |
| CA (1) | CA2741984C (enExample) |
| CL (1) | CL2011000967A1 (enExample) |
| CO (1) | CO6382115A2 (enExample) |
| CY (1) | CY1122269T1 (enExample) |
| DK (1) | DK2352494T3 (enExample) |
| EC (2) | ECSP11011016A (enExample) |
| ES (1) | ES2758831T3 (enExample) |
| HR (1) | HRP20191909T1 (enExample) |
| HU (1) | HUE047438T2 (enExample) |
| IL (2) | IL212523A0 (enExample) |
| LT (1) | LT2352494T (enExample) |
| MX (1) | MX2011004455A (enExample) |
| NZ (1) | NZ592437A (enExample) |
| PE (3) | PE20190391A1 (enExample) |
| PL (1) | PL2352494T3 (enExample) |
| PT (1) | PT2352494T (enExample) |
| RU (2) | RU2599846C2 (enExample) |
| SI (1) | SI2352494T1 (enExample) |
| WO (1) | WO2010096045A1 (enExample) |
Families Citing this family (34)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6216489B2 (ja) | 2008-10-30 | 2017-10-18 | グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング | 新規の、効力のあるタペンタドール剤形 |
| PL2424514T3 (pl) * | 2009-04-30 | 2017-08-31 | Grünenthal GmbH | Tapentadol do leczenia bólu w reumatoidalnym zapaleniu stawów |
| US10363251B2 (en) | 2009-07-16 | 2019-07-30 | Mallinckrodt Llc | (+)-morphinans as antagonists of toll-like receptor 9 and therapeutic uses thereof |
| US20130116333A1 (en) * | 2010-05-05 | 2013-05-09 | Ratiopharm Gmbh | Solid tapentadol in non-crystalline form |
| WO2011141489A1 (en) | 2010-05-10 | 2011-11-17 | Euro-Celtique S.A. | Manufacturing of active-free granules and tablets comprising the same |
| KR101858797B1 (ko) | 2010-05-10 | 2018-05-16 | 유로-셀티큐 에스.에이. | 히드로모르폰 및 날록손을 포함하는 제약 조성물 |
| NZ603170A (en) | 2010-05-10 | 2015-04-24 | Euro Celtique Sa | Combination of active loaded granules with additional actives |
| EP2593095B1 (en) | 2010-07-16 | 2019-03-27 | Mallinckrodt LLC | (+)-morphinans as antagonists of toll-like receptor 9 and therapeutic uses thereof |
| EP3650439B1 (en) * | 2010-07-23 | 2021-02-24 | Grünenthal GmbH | Salts or co-crystals of 3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol |
| WO2012051246A1 (en) * | 2010-10-12 | 2012-04-19 | Ratiopharm Gmbh | Tapentadol hydrobromide and crystalline forms thereof |
| SI3287123T1 (sl) * | 2011-03-04 | 2020-07-31 | Gruenenthal Gmbh | Vodna farmacevtska formulacija tapentadola za peroralno uporabo |
| KR101911362B1 (ko) | 2011-03-04 | 2018-10-25 | 그뤼넨탈 게엠베하 | 타펜타돌을 함유하는 반고체 수성 약제학적 조성물 |
| HUE036567T2 (hu) * | 2011-07-29 | 2018-07-30 | Gruenenthal Gmbh | 3-[(1S,2S)-3-(dimetilamino)-1-etil-2-metilpropil]fenol intratekális vagy epidurális adagolásra |
| EP2606879A1 (en) * | 2011-12-21 | 2013-06-26 | Hexal AG | Multiple unit pellet tablet formulation comprising an opioid |
| WO2014012653A1 (en) | 2012-07-16 | 2014-01-23 | Grünenthal GmbH | Pharmaceutical patch for transdermal administration of tapentadol |
| WO2015023675A2 (en) | 2013-08-12 | 2015-02-19 | Pharmaceutical Manufacturing Research Services, Inc. | Extruded immediate release abuse deterrent pill |
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