KR101712339B1 - 신규하고 강력한 타펜타돌 용량형 - Google Patents

신규하고 강력한 타펜타돌 용량형 Download PDF

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Publication number
KR101712339B1
KR101712339B1 KR1020117012188A KR20117012188A KR101712339B1 KR 101712339 B1 KR101712339 B1 KR 101712339B1 KR 1020117012188 A KR1020117012188 A KR 1020117012188A KR 20117012188 A KR20117012188 A KR 20117012188A KR 101712339 B1 KR101712339 B1 KR 101712339B1
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South Korea
Prior art keywords
group
pentadol
opioid antagonist
hours
naltrexone
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Expired - Fee Related
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KR1020117012188A
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English (en)
Korean (ko)
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KR20110081880A (ko
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라메쉬 세샤
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그뤼넨탈 게엠베하
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Application filed by 그뤼넨탈 게엠베하 filed Critical 그뤼넨탈 게엠베하
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    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
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    • A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Otolaryngology (AREA)
  • Transplantation (AREA)
  • Toxicology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
KR1020117012188A 2008-10-30 2009-10-29 신규하고 강력한 타펜타돌 용량형 Expired - Fee Related KR101712339B1 (ko)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US19762508P 2008-10-30 2008-10-30
US61/197,625 2008-10-30
US20531209P 2009-01-21 2009-01-21
US61/205,312 2009-01-21
US26863009P 2009-06-15 2009-06-15
US61/268,630 2009-06-15
PCT/US2009/005866 WO2010096045A1 (en) 2008-10-30 2009-10-29 Novel and potent tapentadol dosage forms

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020177004316A Division KR101806796B1 (ko) 2008-10-30 2009-10-29 신규하고 강력한 타펜타돌 용량형

Publications (2)

Publication Number Publication Date
KR20110081880A KR20110081880A (ko) 2011-07-14
KR101712339B1 true KR101712339B1 (ko) 2017-03-06

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ID=42634123

Family Applications (2)

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KR1020117012188A Expired - Fee Related KR101712339B1 (ko) 2008-10-30 2009-10-29 신규하고 강력한 타펜타돌 용량형
KR1020177004316A Expired - Fee Related KR101806796B1 (ko) 2008-10-30 2009-10-29 신규하고 강력한 타펜타돌 용량형

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KR1020177004316A Expired - Fee Related KR101806796B1 (ko) 2008-10-30 2009-10-29 신규하고 강력한 타펜타돌 용량형

Country Status (26)

Country Link
US (1) US9642801B2 (enExample)
EP (1) EP2352494B1 (enExample)
JP (2) JP6216489B2 (enExample)
KR (2) KR101712339B1 (enExample)
CN (2) CN102281876A (enExample)
AU (2) AU2009340504A1 (enExample)
BR (1) BRPI0921725A2 (enExample)
CA (1) CA2741984C (enExample)
CL (1) CL2011000967A1 (enExample)
CO (1) CO6382115A2 (enExample)
CY (1) CY1122269T1 (enExample)
DK (1) DK2352494T3 (enExample)
EC (2) ECSP11011016A (enExample)
ES (1) ES2758831T3 (enExample)
HR (1) HRP20191909T1 (enExample)
HU (1) HUE047438T2 (enExample)
IL (2) IL212523A0 (enExample)
LT (1) LT2352494T (enExample)
MX (1) MX2011004455A (enExample)
NZ (1) NZ592437A (enExample)
PE (3) PE20190391A1 (enExample)
PL (1) PL2352494T3 (enExample)
PT (1) PT2352494T (enExample)
RU (2) RU2673882C1 (enExample)
SI (1) SI2352494T1 (enExample)
WO (1) WO2010096045A1 (enExample)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI2352494T1 (sl) 2008-10-30 2019-12-31 Gruenenthal Gmbh Nove in potentne dozirne oblike tapentadola
CA2757757C (en) * 2009-04-30 2017-10-24 Ulrich Jahnel Use of 1-phenyl-3-dimethylaminopropane compounds for treating rheumatoid pain
US10363251B2 (en) 2009-07-16 2019-07-30 Mallinckrodt Llc (+)-morphinans as antagonists of toll-like receptor 9 and therapeutic uses thereof
EP2566461A2 (de) * 2010-05-05 2013-03-13 Ratiopharm GmbH Festes tapentadol in nicht-kristalliner form
MX340188B (es) 2010-05-10 2016-06-30 Euro-Celtique S A * Elaboracion de granulos sin activos y tabletas que comprenden los mismos.
WO2011141490A1 (en) 2010-05-10 2011-11-17 Euro-Celtique S.A. Combination of active loaded granules with additional actives
SG184523A1 (en) 2010-05-10 2012-11-29 Euro Celtique Sa Pharmaceutical compositions comprising hydromorphone and naloxone
WO2012008984A1 (en) 2010-07-16 2012-01-19 Mallinckrodt Llc (+)-morphinans as antagonists of toll-like receptor 9 and therapeutic uses thereof
PT3650439T (pt) * 2010-07-23 2021-03-03 Gruenenthal Gmbh Sais ou cocristais de 3-(3-dimetilamino-1-etil-2-metilpropil)fenol
WO2012051246A1 (en) * 2010-10-12 2012-04-19 Ratiopharm Gmbh Tapentadol hydrobromide and crystalline forms thereof
EP3685827A1 (en) * 2011-03-04 2020-07-29 Grünenthal GmbH Aqueous pharmaceutical formulation of tapentadol for oral administration
PT3766489T (pt) 2011-05-03 2022-04-07 Gruenenthal Gmbh Composição farmacêutica aquosa semissólida contendo tapentadol
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