CN101583369B - 局部制剂及其用途 - Google Patents

局部制剂及其用途 Download PDF

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Publication number
CN101583369B
CN101583369B CN200780049827.XA CN200780049827A CN101583369B CN 101583369 B CN101583369 B CN 101583369B CN 200780049827 A CN200780049827 A CN 200780049827A CN 101583369 B CN101583369 B CN 101583369B
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China
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derivant
formula
analog
another
derivative
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Expired - Fee Related
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English (en)
Chinese (zh)
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CN101583369A (zh
Inventor
拉里·麦凯
卡奴·帕泰尔
罗伯特·约翰·卡彭
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Arthritis Relief Plus Ltd
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Arthritis Relief Plus Ltd
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Publication of CN101583369A publication Critical patent/CN101583369A/zh
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Expired - Fee Related legal-status Critical Current
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00—Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18—Magnoliophyta (angiosperms)
    • A61K36/185—Magnoliopsida (dicotyledons)
    • A61K36/30—Boraginaceae (Borage family), e.g. comfrey, lungwort or forget-me-not
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/14—Quaternary ammonium compounds, e.g. edrophonium, choline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00—Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Botany (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Medical Informatics (AREA)
  • Biotechnology (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
CN200780049827.XA 2006-11-15 2007-11-15 局部制剂及其用途 Expired - Fee Related CN101583369B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US86600106P 2006-11-15 2006-11-15
US60/866,001 2006-11-15
US98107707P 2007-10-18 2007-10-18
US60/981,077 2007-10-18
PCT/AU2007/001753 WO2008058333A1 (en) 2006-11-15 2007-11-15 Topical formulation and uses thereof

Publications (2)

Publication Number Publication Date
CN101583369A CN101583369A (zh) 2009-11-18
CN101583369B true CN101583369B (zh) 2015-03-11

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Application Number Title Priority Date Filing Date
CN200780049827.XA Expired - Fee Related CN101583369B (zh) 2006-11-15 2007-11-15 局部制剂及其用途

Country Status (11)

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US (2) US10322155B2 (enExample)
EP (2) EP2086561A4 (enExample)
JP (1) JP5694665B2 (enExample)
CN (1) CN101583369B (enExample)
AU (1) AU2007321711B2 (enExample)
CA (1) CA2669918C (enExample)
HK (1) HK1251167A1 (enExample)
MY (1) MY151457A (enExample)
NZ (1) NZ577604A (enExample)
RU (1) RU2467759C2 (enExample)
WO (1) WO2008058333A1 (enExample)

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ES2958410T3 (es) 2009-08-21 2024-02-08 Novan Inc Geles tópicos
US8932398B2 (en) 2009-10-29 2015-01-13 Mylan Group Gallotannic compounds for lithographic printing plate coating compositions
US8591876B2 (en) 2010-12-15 2013-11-26 Novan, Inc. Methods of decreasing sebum production in the skin
WO2013006613A1 (en) * 2011-07-05 2013-01-10 Novan, Inc. Methods of manufacturing topical compositions and apparatus for same
US20150141389A1 (en) * 2012-04-27 2015-05-21 Dow Corning Corporation Topical Formulation Compositions Containing Silicone Based Excipients To Deliver Actives To A Substrate
DE202012013584U1 (de) * 2012-10-22 2018-01-15 Briu Gmbh Pharmazeutische Formulierung enthaltend Curcumin
US9775789B2 (en) * 2012-12-06 2017-10-03 D & J Rosée Inc. Topical liposome compositions containing phenolic anti-inflammatory agents and their methods of preparation
US20150005391A1 (en) 2013-06-26 2015-01-01 COLE Research & Design, Inc. Method of reducing scarring
PE20161173A1 (es) * 2014-02-10 2016-10-27 Troikaa Pharmaceuticals Ltd Formulaciones topicas de la heparina
AU2015372438B9 (en) * 2014-12-24 2021-07-08 Sanofi-Aventis Healthcare Pty Ltd Formulation and method of use
WO2017020125A1 (en) * 2015-07-31 2017-02-09 Delivra Inc. Transdermal formulations for delivery of capsaicinoids
US9867827B1 (en) * 2015-08-27 2018-01-16 Florida A&M University Methods and formulations for topical treatment of psoriasis
US10099995B2 (en) 2015-12-24 2018-10-16 Cole Research and Design, LLC Resveratrol esters
CN113413375A (zh) * 2016-05-30 2021-09-21 傅远桥 皮肤多种损伤创面治疗的外用药物组合物及其制备方法
WO2018164662A1 (en) 2017-03-06 2018-09-13 Elsohly Mahmoud A Resveratrol esters
CN108175765A (zh) * 2017-12-01 2018-06-19 东南大学 一种酸敏控释抗炎凝胶及其制备方法与应用
DE202017107326U1 (de) * 2017-12-01 2018-11-21 Kerstin Kräft Hautpflegeemulsion
GR1009658B (el) * 2018-06-18 2019-11-28 Δημητριος Ιωαννη Πουλακας Γελη για την ανακουφιση του πονου αρθρωσεων και ρευματικων παθησεων
CN110526746A (zh) * 2019-08-05 2019-12-03 深圳市芭田生态工程股份有限公司 一种聚氨酯包膜尿素的表面处理方法及聚氨酯包膜尿素
JP7163261B2 (ja) * 2019-09-27 2022-10-31 富士フイルム株式会社 水中油型乳化組成物、及び皮膚外用剤
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WO2021260712A1 (en) * 2020-06-26 2021-12-30 Rohan Sharadanand Phatak A liposomal composition of pterocarpus santalinus and the process thereof
US12109283B2 (en) * 2021-01-20 2024-10-08 Galaxy Surfactants Ltd. Safe and ecofriendly persistent sanitizing gel for topical application
US20240009262A1 (en) * 2022-07-09 2024-01-11 Uab Orbio World Cleansing pad and composition for reducing toxins
CN116392470B (zh) * 2022-10-11 2025-08-01 上海市皮肤病医院 紫草酸在制备治疗糖尿病溃疡药物中的应用
CN116036024B (zh) * 2022-11-15 2024-03-08 国科温州研究院(温州生物材料与工程研究所) 一种植物多酚微球及其制备方法和应用

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Also Published As

Publication number Publication date
MY151457A (en) 2014-05-30
JP5694665B2 (ja) 2015-04-01
NZ577604A (en) 2012-06-29
US10322155B2 (en) 2019-06-18
JP2010509374A (ja) 2010-03-25
US20110038965A1 (en) 2011-02-17
AU2007321711A1 (en) 2008-05-22
HK1251167A1 (en) 2019-01-25
EP3284470A1 (en) 2018-02-21
US20190255133A1 (en) 2019-08-22
WO2008058333A1 (en) 2008-05-22
RU2467759C2 (ru) 2012-11-27
RU2009122520A (ru) 2010-12-20
EP2086561A1 (en) 2009-08-12
EP2086561A4 (en) 2010-05-12
US11844820B2 (en) 2023-12-19
CN101583369A (zh) 2009-11-18
AU2007321711B2 (en) 2013-01-17
CA2669918C (en) 2020-03-10
CA2669918A1 (en) 2008-05-22

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Granted publication date: 20150311