CN101312733A - 戊酸雌二醇或雌二醇与地诺孕素组合以口服避孕药形式口服治疗功能失调性子宫出血的用途 - Google Patents

戊酸雌二醇或雌二醇与地诺孕素组合以口服避孕药形式口服治疗功能失调性子宫出血的用途 Download PDF

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Publication number
CN101312733A
CN101312733A CNA2006800381810A CN200680038181A CN101312733A CN 101312733 A CN101312733 A CN 101312733A CN A2006800381810 A CNA2006800381810 A CN A2006800381810A CN 200680038181 A CN200680038181 A CN 200680038181A CN 101312733 A CN101312733 A CN 101312733A
Authority
CN
China
Prior art keywords
estradiol
dienogest
combination
daily dosage
dosage units
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CNA2006800381810A
Other languages
English (en)
Chinese (zh)
Inventor
S·宙恩
P·布德
J·昂德里卡
A·塞西
H·齐默尔曼
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Pharma AG
Original Assignee
Schering AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35811580&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN101312733(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering AG filed Critical Schering AG
Publication of CN101312733A publication Critical patent/CN101312733A/zh
Pending legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30Oestrogens

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
CNA2006800381810A 2005-10-13 2006-10-12 戊酸雌二醇或雌二醇与地诺孕素组合以口服避孕药形式口服治疗功能失调性子宫出血的用途 Pending CN101312733A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05022324A EP1787649B1 (de) 2005-10-13 2005-10-13 Verwendung von Estradiolvalerat in Kombination mit Dienogest zur oralen Therapie der dysfunktionellen uterinen Blutung in Einheit mit einer oralen Kontrazeption
EP05022324.7 2005-10-13

Publications (1)

Publication Number Publication Date
CN101312733A true CN101312733A (zh) 2008-11-26

Family

ID=35811580

Family Applications (1)

Application Number Title Priority Date Filing Date
CNA2006800381810A Pending CN101312733A (zh) 2005-10-13 2006-10-12 戊酸雌二醇或雌二醇与地诺孕素组合以口服避孕药形式口服治疗功能失调性子宫出血的用途

Country Status (22)

Country Link
EP (2) EP1787649B1 (https=)
JP (2) JP5735200B2 (https=)
KR (2) KR101218872B1 (https=)
CN (1) CN101312733A (https=)
AR (1) AR056694A1 (https=)
AT (2) ATE424828T1 (https=)
CA (1) CA2623024C (https=)
CL (1) CL2011000283A1 (https=)
CY (2) CY1110321T1 (https=)
DE (2) DE502005006837D1 (https=)
DK (2) DK1787649T3 (https=)
DO (1) DOP2006000221A (https=)
ES (2) ES2322479T3 (https=)
HR (1) HRP20090256T1 (https=)
ME (1) ME01056B (https=)
PE (2) PE20100090A1 (https=)
PL (2) PL1787649T3 (https=)
PT (2) PT1787649E (https=)
SI (2) SI1787649T1 (https=)
TW (2) TWI328453B (https=)
UY (1) UY29861A1 (https=)
WO (1) WO2007042296A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004019743B4 (de) 2004-04-20 2008-11-27 Bayer Schering Pharma Aktiengesellschaft Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens
SI1787649T1 (sl) * 2005-10-13 2009-08-31 Bayer Schering Pharma Ag Uporaba estradiolvalerata v kombinaciji z dienogestom za oralno terapijo disfunkcionalne maternične krvavitve skupaj z oralno kontracepcijo
US8153616B2 (en) 2005-10-17 2012-04-10 Bayer Pharma Aktiengesellschaft Combination preparation for oral contraception and oral therapy of dysfunctional uterine bleeding containing estradiol valerate and dienogest and method of using same
EP1930010A1 (de) 2006-10-20 2008-06-11 Bayer Schering Pharma Aktiengesellschaft Verwendung von Estradiolvalerat oder 17ß-Estradiol in Kombination mit Dienogest zur oralen Therapie für den Erhalt und/oder die Steigerung der weiblichen Libido

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4429374C1 (de) * 1994-08-12 1996-02-01 Jenapharm Gmbh Pharmazeutische Präparate zur Kontrazeption/Hormonsubstitution mit biogener Estrogenkomponente
DE19540253C2 (de) * 1995-10-28 1998-06-04 Jenapharm Gmbh Mehrphasenpräparat zur Kontrazeption auf der Basis natürlicher Estrogene
ATE249222T1 (de) * 1996-07-26 2003-09-15 Wyeth Corp Biphasische orale verhuetungsmethode und kit die eine kombination von progestin und eines oestrogens enthalten
US6251956B1 (en) 1998-08-20 2001-06-26 Ortho Pharmaceutical Corporation Combination progestin oral contraceptive regimen
EP1462106A1 (en) * 2003-03-28 2004-09-29 Pantarhei Bioscience B.V. Pharmaceutical compositions and kits comprising 17-beta-estradiol and a progesteron for the treatment of gynecological disorders
DE102004019743B4 (de) * 2004-04-20 2008-11-27 Bayer Schering Pharma Aktiengesellschaft Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens
SI1787649T1 (sl) * 2005-10-13 2009-08-31 Bayer Schering Pharma Ag Uporaba estradiolvalerata v kombinaciji z dienogestom za oralno terapijo disfunkcionalne maternične krvavitve skupaj z oralno kontracepcijo

Also Published As

Publication number Publication date
CA2623024A1 (en) 2007-04-19
EP1933843A1 (de) 2008-06-25
ES2322479T3 (es) 2009-06-22
WO2007042296A1 (de) 2007-04-19
ATE424828T1 (de) 2009-03-15
JP5735200B2 (ja) 2015-06-17
JP2009511526A (ja) 2009-03-19
SI1933843T1 (sl) 2011-06-30
PT1787649E (pt) 2009-05-08
EP1787649A1 (de) 2007-05-23
ES2360302T3 (es) 2011-06-02
CL2011000283A1 (es) 2011-07-08
PT1933843E (pt) 2011-04-29
KR20080065651A (ko) 2008-07-14
HRP20090256T1 (en) 2009-06-30
AR056694A1 (es) 2007-10-17
DE502005006837D1 (de) 2009-04-23
PL1933843T3 (pl) 2011-06-30
SI1787649T1 (sl) 2009-08-31
CA2623024C (en) 2012-03-06
TW200731977A (en) 2007-09-01
DOP2006000221A (es) 2007-08-31
PE20100090A1 (es) 2010-03-12
DK1787649T3 (da) 2009-06-02
TWI328453B (en) 2010-08-11
UY29861A1 (es) 2007-05-31
DE502006008853D1 (de) 2011-03-17
EP1787649B1 (de) 2009-03-11
TW200829255A (en) 2008-07-16
ATE497387T1 (de) 2011-02-15
CY1111406T1 (el) 2015-08-05
KR20100082389A (ko) 2010-07-16
PL1787649T3 (pl) 2009-08-31
KR101218872B1 (ko) 2013-01-07
CY1110321T1 (el) 2015-01-14
DK1933843T3 (da) 2011-04-18
PE20070555A1 (es) 2007-07-12
JP2013047269A (ja) 2013-03-07
ME01056B (me) 2012-10-20
EP1933843B1 (de) 2011-02-02

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