CN101084224B - 具有杀真菌活性的噻吩并-嘧啶化合物 - Google Patents

具有杀真菌活性的噻吩并-嘧啶化合物 Download PDF

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Publication number
CN101084224B
CN101084224B CN2005800440617A CN200580044061A CN101084224B CN 101084224 B CN101084224 B CN 101084224B CN 2005800440617 A CN2005800440617 A CN 2005800440617A CN 200580044061 A CN200580044061 A CN 200580044061A CN 101084224 B CN101084224 B CN 101084224B
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CN
China
Prior art keywords
compound
mmol
compounds
plants
mixture
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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CN2005800440617A
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English (en)
Chinese (zh)
Other versions
CN101084224A (zh
Inventor
W·K·布鲁斯特
C·J·R·克利奇
T·W·巴尔科
N·T·布罗
W·R·埃里克森
J·E·亨特
C·T·洛
M·J·克里斯
T·L·西多尔
C·N·耶里斯
Y·朱
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Corteva Agriscience LLC
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Dow AgroSciences LLC
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Publication of CN101084224A publication Critical patent/CN101084224A/zh
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Publication of CN101084224B publication Critical patent/CN101084224B/zh
Anticipated expiration legal-status Critical
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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
CN2005800440617A 2004-10-21 2005-10-21 具有杀真菌活性的噻吩并-嘧啶化合物 Expired - Fee Related CN101084224B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62157704P 2004-10-21 2004-10-21
US60/621,577 2004-10-21
PCT/US2005/038145 WO2006047397A1 (en) 2004-10-21 2005-10-21 Thieno-pyrimidine compounds having fungicidal activity

Publications (2)

Publication Number Publication Date
CN101084224A CN101084224A (zh) 2007-12-05
CN101084224B true CN101084224B (zh) 2013-12-04

Family

ID=35722379

Family Applications (1)

Application Number Title Priority Date Filing Date
CN2005800440617A Expired - Fee Related CN101084224B (zh) 2004-10-21 2005-10-21 具有杀真菌活性的噻吩并-嘧啶化合物

Country Status (8)

Country Link
US (1) US8008487B2 (https=)
EP (1) EP1802632B1 (https=)
JP (2) JP5122293B2 (https=)
KR (3) KR20140008471A (https=)
CN (1) CN101084224B (https=)
AT (1) ATE516291T1 (https=)
BR (1) BRPI0516242B1 (https=)
WO (1) WO2006047397A1 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8008487B2 (en) * 2004-10-21 2011-08-30 Dow Agrosciences Llc Substituted thieno[2,3-D]pyrimidines as fungicides
EP1937691A1 (en) * 2005-10-21 2008-07-02 Dow Agrosciences LLC Thieno-pyrimidine compounds having fungicidal activity
AP2008004687A0 (en) * 2006-05-22 2008-12-31 Basf Se Insecticidal methods using 4-amino-5-chloro-thieno(2,3-d)-pyrimidine compounds
US8318384B2 (en) 2007-04-30 2012-11-27 The Governors Of The University Of Alberta Anode catalyst and methods of making and using the same
CN102186479A (zh) * 2008-09-10 2011-09-14 凯利普西斯公司 用于治疗疾病的组胺受体的氨基嘧啶抑制剂
PL2455371T3 (pl) 2009-07-16 2014-05-30 Sds Biotech Corp Pochodne 4-(3-butynylo)aminopirymidyny jako środki do zwalczania szkodników do stosowania w rolnictwie i ogrodnictwie
BR112012002164B1 (pt) 2009-07-30 2021-04-20 Merial, Inc compostos inseticidas de 4-amino-tieno[2,3-d]-pirimidina e métodos para seu uso
AU2011354895B2 (en) 2011-01-14 2016-05-05 Sds Biotech K. K. Agri-horticultural pest control compositions comprising 4- (3-butynyl)aminopyrimidine derivatives
ES2618813T3 (es) * 2011-06-27 2017-06-22 Merial, Inc. Compuestos y composiciones de éter amido-piridílico y uso contra los parásitos
AR088218A1 (es) 2011-07-19 2014-05-21 Infinity Pharmaceuticals Inc Compuestos heterociclicos utiles como inhibidores de pi3k
AR090037A1 (es) 2011-11-15 2014-10-15 Xention Ltd Derivados de tieno y/o furo-pirimidinas y piridinas inhibidores de los canales de potasio
CN105315296B (zh) * 2014-07-04 2018-04-03 沈阳中化农药化工研发有限公司 取代芳氧吡啶类化合物及其用途
CN104725398B (zh) * 2015-01-29 2017-01-18 杨威 一种jak/stat3磷酸化抑制剂及其制备方法与用途
CN109776427B (zh) * 2017-11-13 2022-08-23 沈阳中化农药化工研发有限公司 嘧啶双胺类化合物及其用途
MX2021010319A (es) * 2019-03-01 2021-12-10 Revolution Medicines Inc Compuestos biciclicos de heteroarilo y usos de estos.
CN115626893B (zh) * 2022-10-10 2024-04-02 山西永津集团有限公司 一种2-羟基-5-羟甲基吡啶的合成方法

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4146716A (en) * 1975-11-28 1979-03-27 Imperial Chemical Industries Limited Thienopyrimidines
US5124333A (en) * 1989-08-02 1992-06-23 Ube Industries, Ltd. Aminopyrimidine derivatives and harmful organisms preventive agent
US5141941A (en) * 1988-11-21 1992-08-25 Ube Industries, Ltd. Aralkylamine derivatives, and fungicides containing the same
CN1168671A (zh) * 1994-12-07 1997-12-24 诺瓦蒂斯有限公司 新的嘧啶基氧基-和嘧啶基氨基-乙基苯基二氧戊环衍生物

Family Cites Families (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4196207A (en) * 1977-05-23 1980-04-01 Ici Australia Limited Process for controlling eradicating or preventing infestations of animals by Ixodid ticks
GB2043061B (en) * 1979-03-05 1983-05-11 Ici Ltd Thienopyrimidine and quinazoline derivatives
JPS5942387A (ja) * 1982-07-21 1984-03-08 Sankyo Co Ltd チエノピリミジン誘導体および殺虫、殺ダニ剤
EP0193885B1 (de) 1985-03-02 1989-06-14 BASF Aktiengesellschaft Thiophenderivate
JPS6267A (ja) * 1985-03-14 1987-01-06 Sankyo Co Ltd フエノキシアルキルアミン誘導体、その製法および殺虫殺ダニ剤
JPH0363265A (ja) * 1989-08-02 1991-03-19 Ube Ind Ltd アルキルアミノピリミジン誘導体、その製造法及び殺虫・殺ダニ・殺線虫剤
JPH075569B2 (ja) * 1989-08-02 1995-01-25 宇部興産株式会社 アラルキルアミン誘導体、その製法及び殺菌、殺虫剤
EP0424125A3 (en) 1989-10-18 1991-10-09 Ube Industries, Ltd. Aralkylamine derivatives, preparation method thereof and fungicides containing the same
DE4008726A1 (de) * 1990-03-19 1991-09-26 Basf Ag Thieno(2,3-d)pyrimidinderivate
US5137879A (en) * 1990-03-30 1992-08-11 Dowelanco Furopyrimidin-4-imine derivatives
AU651337B2 (en) * 1990-03-30 1994-07-21 Dowelanco Thienopyrimidine derivatives
JP2730019B2 (ja) * 1990-04-06 1998-03-25 宇部興産株式会社 アラルキルアミン誘導体，その製造法及び殺菌剤
JP2762430B2 (ja) 1991-01-18 1998-06-04 宇部興産株式会社 アラルキルアミノピリミジン類の製法
EP0519211A1 (de) * 1991-05-17 1992-12-23 Hoechst Schering AgrEvo GmbH Substituierte 4-Aminopyrimidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel
JP3063266B2 (ja) 1991-08-30 2000-07-12 セイコーエプソン株式会社 液晶パネル及びその製造方法
JPH0710712A (ja) * 1993-06-25 1995-01-13 Ube Ind Ltd 花卉園芸用殺菌剤
US5654307A (en) * 1994-01-25 1997-08-05 Warner-Lambert Company Bicyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family
US6232320B1 (en) * 1998-06-04 2001-05-15 Abbott Laboratories Cell adhesion-inhibiting antiinflammatory compounds
AU4231299A (en) * 1998-06-04 1999-12-20 Abbott Laboratories Cell adhesion-inhibiting antinflammatory compounds
CA2390948A1 (en) * 1999-06-03 2000-12-14 Abbott Laboratories Cell adhesion-inhibiting antiinflammatory compounds
WO2003022214A2 (en) * 2001-09-06 2003-03-20 Millennium Pharmaceuticals, Inc. Piperazine and homopiperazine compounds
AU2002357193A1 (en) 2001-12-19 2003-07-09 Smithkline Beecham Corporation Thienopyrimidine compounds as protein tyrosine kinase inhibitors
WO2004092123A2 (en) * 2003-04-10 2004-10-28 Microbia, Inc. Inhibitors of fungal invasion
ES2324536T7 (es) * 2003-06-11 2012-03-16 Xention Limited Derivados de tenopirimidina como inhibidores de los canales de potasio.
GB0315950D0 (en) * 2003-06-11 2003-08-13 Xention Discovery Ltd Compounds
US8008487B2 (en) * 2004-10-21 2011-08-30 Dow Agrosciences Llc Substituted thieno[2,3-D]pyrimidines as fungicides

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4146716A (en) * 1975-11-28 1979-03-27 Imperial Chemical Industries Limited Thienopyrimidines
US5141941A (en) * 1988-11-21 1992-08-25 Ube Industries, Ltd. Aralkylamine derivatives, and fungicides containing the same
US5124333A (en) * 1989-08-02 1992-06-23 Ube Industries, Ltd. Aminopyrimidine derivatives and harmful organisms preventive agent
CN1168671A (zh) * 1994-12-07 1997-12-24 诺瓦蒂斯有限公司 新的嘧啶基氧基-和嘧啶基氨基-乙基苯基二氧戊环衍生物

Also Published As

Publication number Publication date
KR20140008471A (ko) 2014-01-21
WO2006047397A1 (en) 2006-05-04
JP2012180362A (ja) 2012-09-20
US8008487B2 (en) 2011-08-30
BRPI0516242A (pt) 2008-08-26
BRPI0516242B1 (pt) 2014-10-07
HK1118534A1 (en) 2009-02-13
ATE516291T1 (de) 2011-07-15
KR101386797B1 (ko) 2014-04-21
JP5122293B2 (ja) 2013-01-16
JP2008517936A (ja) 2008-05-29
JP5572664B2 (ja) 2014-08-13
US20060089370A1 (en) 2006-04-27
EP1802632B1 (en) 2011-07-13
CN101084224A (zh) 2007-12-05
KR20140094626A (ko) 2014-07-30
EP1802632A1 (en) 2007-07-04
KR20070063602A (ko) 2007-06-19

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