CN101084224B - 具有杀真菌活性的噻吩并-嘧啶化合物 - Google Patents

具有杀真菌活性的噻吩并-嘧啶化合物 Download PDF

Info

Publication number
CN101084224B
CN101084224B CN2005800440617A CN200580044061A CN101084224B CN 101084224 B CN101084224 B CN 101084224B CN 2005800440617 A CN2005800440617 A CN 2005800440617A CN 200580044061 A CN200580044061 A CN 200580044061A CN 101084224 B CN101084224 B CN 101084224B
Authority
CN
China
Prior art keywords
compound
mmol
compounds
plants
mixture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CN2005800440617A
Other languages
English (en)
Chinese (zh)
Other versions
CN101084224A (zh
Inventor
W·K·布鲁斯特
C·J·R·克利奇
T·W·巴尔科
N·T·布罗
W·R·埃里克森
J·E·亨特
C·T·洛
M·J·克里斯
T·L·西多尔
C·N·耶里斯
Y·朱
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Corteva Agriscience LLC
Original Assignee
Dow AgroSciences LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow AgroSciences LLC filed Critical Dow AgroSciences LLC
Publication of CN101084224A publication Critical patent/CN101084224A/zh
Application granted granted Critical
Publication of CN101084224B publication Critical patent/CN101084224B/zh
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
CN2005800440617A 2004-10-21 2005-10-21 具有杀真菌活性的噻吩并-嘧啶化合物 Expired - Fee Related CN101084224B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62157704P 2004-10-21 2004-10-21
US60/621,577 2004-10-21
PCT/US2005/038145 WO2006047397A1 (en) 2004-10-21 2005-10-21 Thieno-pyrimidine compounds having fungicidal activity

Publications (2)

Publication Number Publication Date
CN101084224A CN101084224A (zh) 2007-12-05
CN101084224B true CN101084224B (zh) 2013-12-04

Family

ID=35722379

Family Applications (1)

Application Number Title Priority Date Filing Date
CN2005800440617A Expired - Fee Related CN101084224B (zh) 2004-10-21 2005-10-21 具有杀真菌活性的噻吩并-嘧啶化合物

Country Status (8)

Country Link
US (1) US8008487B2 (https=)
EP (1) EP1802632B1 (https=)
JP (2) JP5122293B2 (https=)
KR (3) KR101386797B1 (https=)
CN (1) CN101084224B (https=)
AT (1) ATE516291T1 (https=)
BR (1) BRPI0516242B1 (https=)
WO (1) WO2006047397A1 (https=)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101084224B (zh) * 2004-10-21 2013-12-04 美国陶氏益农公司 具有杀真菌活性的噻吩并-嘧啶化合物
WO2007046809A1 (en) * 2005-10-21 2007-04-26 Dow Agrosciences Llc Thieno-pyrimidine compounds having fungicidal activity
MX2008013965A (es) 2006-05-22 2008-11-12 Basf Se Metodos insecticidas usando compuestos de 4-amino-5-cloro-tieno[2, 3-d]-pirimidina.
US8318384B2 (en) 2007-04-30 2012-11-27 The Governors Of The University Of Alberta Anode catalyst and methods of making and using the same
AU2009291783A1 (en) * 2008-09-10 2010-03-18 Alcon Research, Ltd Aminopyrimidine inhibitors of histamine receptors for the treatment of disease
US8586505B2 (en) 2009-07-16 2013-11-19 Sds Biotech K. K. 4-(3-butynyl)aminopyrimidine derivatives as pest control agents for agricultural and horticultural use
CN102596968B (zh) * 2009-07-30 2015-05-06 梅里亚有限公司 杀虫的4-氨基-噻吩并[2,3-d]-嘧啶化合物及其使用方法
NZ613449A (en) * 2011-01-14 2015-08-28 Sds Biotech Corp Agri-horticultural pest control compositions comprising 4-(3-butynyl)aminopyrimidine derivatives
ES2618813T3 (es) * 2011-06-27 2017-06-22 Merial, Inc. Compuestos y composiciones de éter amido-piridílico y uso contra los parásitos
MX2014000648A (es) 2011-07-19 2014-09-25 Infinity Pharmaceuticals Inc Compuestos heterociclicos y sus usos.
AR090037A1 (es) 2011-11-15 2014-10-15 Xention Ltd Derivados de tieno y/o furo-pirimidinas y piridinas inhibidores de los canales de potasio
CN105315296B (zh) * 2014-07-04 2018-04-03 沈阳中化农药化工研发有限公司 取代芳氧吡啶类化合物及其用途
CN104725398B (zh) * 2015-01-29 2017-01-18 杨威 一种jak/stat3磷酸化抑制剂及其制备方法与用途
CN109776427B (zh) * 2017-11-13 2022-08-23 沈阳中化农药化工研发有限公司 嘧啶双胺类化合物及其用途
WO2020180768A1 (en) * 2019-03-01 2020-09-10 Revolution Medicines, Inc. Bicyclic heteroaryl compounds and uses thereof
CN115626893B (zh) * 2022-10-10 2024-04-02 山西永津集团有限公司 一种2-羟基-5-羟甲基吡啶的合成方法

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4146716A (en) * 1975-11-28 1979-03-27 Imperial Chemical Industries Limited Thienopyrimidines
US5124333A (en) * 1989-08-02 1992-06-23 Ube Industries, Ltd. Aminopyrimidine derivatives and harmful organisms preventive agent
US5141941A (en) * 1988-11-21 1992-08-25 Ube Industries, Ltd. Aralkylamine derivatives, and fungicides containing the same
CN1168671A (zh) * 1994-12-07 1997-12-24 诺瓦蒂斯有限公司 新的嘧啶基氧基-和嘧啶基氨基-乙基苯基二氧戊环衍生物

Family Cites Families (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA782648B (en) * 1977-05-23 1979-06-27 Ici Australia Ltd The prevention,control or eradication of infestations of ixodid ticks
GB2043061B (en) 1979-03-05 1983-05-11 Ici Ltd Thienopyrimidine and quinazoline derivatives
JPS5942387A (ja) * 1982-07-21 1984-03-08 Sankyo Co Ltd チエノピリミジン誘導体および殺虫、殺ダニ剤
DE3663945D1 (en) 1985-03-02 1989-07-20 Basf Ag Thiophene derivatives
JPS6267A (ja) * 1985-03-14 1987-01-06 Sankyo Co Ltd フエノキシアルキルアミン誘導体、その製法および殺虫殺ダニ剤
JPH075569B2 (ja) * 1989-08-02 1995-01-25 宇部興産株式会社 アラルキルアミン誘導体、その製法及び殺菌、殺虫剤
JPH0363265A (ja) * 1989-08-02 1991-03-19 Ube Ind Ltd アルキルアミノピリミジン誘導体、その製造法及び殺虫・殺ダニ・殺線虫剤
EP0424125A3 (en) 1989-10-18 1991-10-09 Ube Industries, Ltd. Aralkylamine derivatives, preparation method thereof and fungicides containing the same
DE4008726A1 (de) 1990-03-19 1991-09-26 Basf Ag Thieno(2,3-d)pyrimidinderivate
BR9101256A (pt) * 1990-03-30 1991-11-05 Dowelanco Composto,composicao fungicida,processo fungicida,composicao inseticida ou acaricida e processo inseticida ou acaricida
US5137879A (en) * 1990-03-30 1992-08-11 Dowelanco Furopyrimidin-4-imine derivatives
JP2730019B2 (ja) * 1990-04-06 1998-03-25 宇部興産株式会社 アラルキルアミン誘導体，その製造法及び殺菌剤
JP2762430B2 (ja) 1991-01-18 1998-06-04 宇部興産株式会社 アラルキルアミノピリミジン類の製法
EP0519211A1 (de) * 1991-05-17 1992-12-23 Hoechst Schering AgrEvo GmbH Substituierte 4-Aminopyrimidine, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel
JP3063266B2 (ja) 1991-08-30 2000-07-12 セイコーエプソン株式会社 液晶パネル及びその製造方法
JPH0710712A (ja) * 1993-06-25 1995-01-13 Ube Ind Ltd 花卉園芸用殺菌剤
US5679683A (en) * 1994-01-25 1997-10-21 Warner-Lambert Company Tricyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family
CA2333770A1 (en) * 1998-06-04 1999-12-09 Abbott Laboratories Cell adhesion-inhibiting antinflammatory compounds
US6232320B1 (en) * 1998-06-04 2001-05-15 Abbott Laboratories Cell adhesion-inhibiting antiinflammatory compounds
JP2004509059A (ja) * 1999-06-03 2004-03-25 アボット・ラボラトリーズ 細胞接着抑制性抗炎症化合物
AU2002336462A1 (en) * 2001-09-06 2003-03-24 Millennium Pharmaceuticals, Inc. Piperazine and homopiperazine compounds
EP1463507A1 (en) 2001-12-19 2004-10-06 SmithKline Beecham Corporation Thienopyrimidine compounds as protein tyrosine kinase inhibitors
WO2004092123A2 (en) * 2003-04-10 2004-10-28 Microbia, Inc. Inhibitors of fungal invasion
GB0315950D0 (en) * 2003-06-11 2003-08-13 Xention Discovery Ltd Compounds
PL1641803T6 (pl) * 2003-06-11 2011-04-29 Xention Ltd Pochodne tienopirymidyny jako inhibitory kanału potasowego
CN101084224B (zh) * 2004-10-21 2013-12-04 美国陶氏益农公司 具有杀真菌活性的噻吩并-嘧啶化合物

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4146716A (en) * 1975-11-28 1979-03-27 Imperial Chemical Industries Limited Thienopyrimidines
US5141941A (en) * 1988-11-21 1992-08-25 Ube Industries, Ltd. Aralkylamine derivatives, and fungicides containing the same
US5124333A (en) * 1989-08-02 1992-06-23 Ube Industries, Ltd. Aminopyrimidine derivatives and harmful organisms preventive agent
CN1168671A (zh) * 1994-12-07 1997-12-24 诺瓦蒂斯有限公司 新的嘧啶基氧基-和嘧啶基氨基-乙基苯基二氧戊环衍生物

Also Published As

Publication number Publication date
ATE516291T1 (de) 2011-07-15
JP2012180362A (ja) 2012-09-20
KR20140094626A (ko) 2014-07-30
HK1118534A1 (en) 2009-02-13
JP5122293B2 (ja) 2013-01-16
JP2008517936A (ja) 2008-05-29
KR101386797B1 (ko) 2014-04-21
WO2006047397A1 (en) 2006-05-04
CN101084224A (zh) 2007-12-05
BRPI0516242A (pt) 2008-08-26
US8008487B2 (en) 2011-08-30
BRPI0516242B1 (pt) 2014-10-07
KR20070063602A (ko) 2007-06-19
KR20140008471A (ko) 2014-01-21
JP5572664B2 (ja) 2014-08-13
US20060089370A1 (en) 2006-04-27
EP1802632B1 (en) 2011-07-13
EP1802632A1 (en) 2007-07-04

Similar Documents

Publication Publication Date Title
JP5572664B2 (ja) 殺真菌活性を有するチエノ−ピリミジン化合物
US10231453B2 (en) 5-substituted imidazole derivatives
EP1434776A1 (en) Thiazolyl substituted aminopyrimidines as plant protection agents
EP1455579A1 (en) Pyrazoles-pyrimidine fungicides
EP3625215B1 (en) Formimidamidine compounds useful against phytopathogenic microorganisms
CN115052875B (zh) 作为作物保护用杀真菌剂的4-(4-(4,5-二氢异恶唑-3-基)噻唑-2-基)哌啶硫亚胺或亚砜亚胺衍生物及相关化合物
CN114761403B (zh) 用作作物保护杀菌剂的1-(4-(4-(5-苯基-4,5-二氢异噁唑-3-基)噻唑-2-基)哌啶-1-基)-乙烷-1-酮衍生物及相关化合物
AU2020210116B2 (en) 3-substituted phenylamidine compounds, preparation and use thereof
TW201641493A (zh) 新穎三唑衍生物
CN109476606B (zh) 苯并磺内酰胺和类似物及其作为杀真菌剂的用途
CN114514228A (zh) 用作农业杀真菌剂的吡啶酰胺衍生物
CN111542517A (zh) 作为农用化学品的苯并咪唑化合物
JPH09176170A (ja) 殺微生物剤
TW202104222A (zh) 噁二唑化合物、該噁二唑化合物的應用及該噁二唑化合物的製備方法
HK1118534B (en) Thieno-pyrimidine compounds having fungicidal activity
AU2017333782A1 (en) Novel 5-substituted imidazolylmethyl derivatives
WO2020157710A1 (en) 4-substituted isoxazole/isoxazoline (hetero) arylamidine compounds, preparation and use thereof
WO2020035825A1 (en) N'-(4-(benzylamino)-phenyl)-n-ethyl-n-methylformimidamide derivatives and related compounds for protecting agricultural crops against phytopathogenic microorganisms
JP2008524292A (ja) 新規のトリアゾロピリミジン誘導体

Legal Events

Date Code Title Description
C06 Publication
PB01 Publication
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
REG Reference to a national code

Ref country code: HK

Ref legal event code: DE

Ref document number: 1118534

Country of ref document: HK

C14 Grant of patent or utility model
GR01 Patent grant
REG Reference to a national code

Ref country code: HK

Ref legal event code: GR

Ref document number: 1118534

Country of ref document: HK

CF01 Termination of patent right due to non-payment of annual fee

Granted publication date: 20131204

Termination date: 20151021

EXPY Termination of patent right or utility model