CH667087A5 - In der seitenkette ungesaettigte 1-hydroxyvitamin d-verbindungen. - Google Patents

In der seitenkette ungesaettigte 1-hydroxyvitamin d-verbindungen. Download PDF

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Publication number
CH667087A5
CH667087A5 CH4259/85A CH425985A CH667087A5 CH 667087 A5 CH667087 A5 CH 667087A5 CH 4259/85 A CH4259/85 A CH 4259/85A CH 425985 A CH425985 A CH 425985A CH 667087 A5 CH667087 A5 CH 667087A5
Authority
CH
Switzerland
Prior art keywords
compounds
compound
hydroxy
vitamin
side chain
Prior art date
Application number
CH4259/85A
Other languages
German (de)
English (en)
Inventor
Hector F Deluca
Heinrich K Schnoes
Rafal R Sicinski
Yoko Tanaka
Original Assignee
Wisconsin Alumni Res Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wisconsin Alumni Res Found filed Critical Wisconsin Alumni Res Found
Publication of CH667087A5 publication Critical patent/CH667087A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0042—Nitrogen only

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Nutrition Science (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
CH4259/85A 1984-01-30 1985-01-07 In der seitenkette ungesaettigte 1-hydroxyvitamin d-verbindungen. CH667087A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57511684A 1984-01-30 1984-01-30

Publications (1)

Publication Number Publication Date
CH667087A5 true CH667087A5 (de) 1988-09-15

Family

ID=24299022

Family Applications (1)

Application Number Title Priority Date Filing Date
CH4259/85A CH667087A5 (de) 1984-01-30 1985-01-07 In der seitenkette ungesaettigte 1-hydroxyvitamin d-verbindungen.

Country Status (11)

Country Link
JP (1) JPS61501146A (ja)
AU (1) AU589113B2 (ja)
BE (1) BE901602A (ja)
CH (1) CH667087A5 (ja)
DE (2) DE3590020C2 (ja)
DK (1) DK437585D0 (ja)
FR (1) FR2558830B1 (ja)
GB (1) GB2153359B (ja)
IE (1) IE57947B1 (ja)
NL (1) NL8520003A (ja)
WO (1) WO1985003299A1 (ja)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6421A (en) * 1987-02-27 1989-01-05 Teijin Ltd Preventive for osteoporosis
CA2166898C (en) * 1993-07-09 2004-09-07 Roger Bouillon Novel structural analogues of vitamin d

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3697559A (en) * 1971-02-25 1972-10-10 Wisconsin Alumni Res Found 1,25-dihydroxycholecalciferol
US3741996A (en) * 1971-12-02 1973-06-26 Wisconsin Alumni Res Found 1{60 -hydroxycholecalciferol
US3907843A (en) * 1974-06-14 1975-09-23 Wisconsin Alumni Res Found 1{60 -Hydroxyergocalciferol and processes for preparing same
US4225596A (en) * 1978-10-13 1980-09-30 Wisconsin Alumni Research Foundation Method for treating calcium imbalance and improving calcium absorption in mammals
US4264513A (en) * 1979-05-21 1981-04-28 Wisconsin Alumni Research Foundation 1α-hydroxy-25-keto-27-nor-cholecalciferol and processes for preparing same
NL8320218A (nl) * 1982-07-26 1984-06-01 Wisconsin Alumni Res Found Nieuwe vitamine d analogen.
US4508651A (en) * 1983-03-21 1985-04-02 Hoffmann-La Roche Inc. Synthesis of 1α,25-dihydroxyergocalciferol
DE3590021C2 (de) * 1984-01-30 1992-09-10 Wisconsin Alumni Res Found 1alpha-Hydroxyvitamin D-Derivat und dieses enthaltendes Arzneimittel

Also Published As

Publication number Publication date
GB2153359B (en) 1987-08-12
JPS61501146A (ja) 1986-06-12
FR2558830B1 (fr) 1987-11-20
AU3831785A (en) 1985-08-09
JPH0455424B2 (ja) 1992-09-03
IE57947B1 (en) 1993-05-19
NL8520003A (nl) 1985-12-02
IE850212L (en) 1985-07-30
DK437585A (da) 1985-09-27
AU589113B2 (en) 1989-10-05
WO1985003299A1 (en) 1985-08-01
GB8502163D0 (en) 1985-02-27
BE901602A (fr) 1985-05-17
FR2558830A1 (fr) 1985-08-02
DE3590020T1 (de) 1986-01-23
GB2153359A (en) 1985-08-21
DK437585D0 (da) 1985-09-27
DE3590020C2 (de) 1995-03-09

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Date Code Title Description
PL Patent ceased