CH623317A5 - Process for the preparation of benzamides - Google Patents

Process for the preparation of benzamides Download PDF

Info

Publication number
CH623317A5
CH623317A5 CH1581976A CH1581976A CH623317A5 CH 623317 A5 CH623317 A5 CH 623317A5 CH 1581976 A CH1581976 A CH 1581976A CH 1581976 A CH1581976 A CH 1581976A CH 623317 A5 CH623317 A5 CH 623317A5
Authority
CH
Switzerland
Prior art keywords
formula
compound
hydrogen
starting material
halogen
Prior art date
Application number
CH1581976A
Other languages
German (de)
English (en)
Inventor
Willy Dr Burkard
Pierre-Charles Dr Wyss
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH623317A5 publication Critical patent/CH623317A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CH1581976A 1976-02-16 1976-12-16 Process for the preparation of benzamides CH623317A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
AT107076A AT345842B (de) 1976-02-16 1976-02-16 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxyden und salzen

Publications (1)

Publication Number Publication Date
CH623317A5 true CH623317A5 (en) 1981-05-29

Family

ID=3505951

Family Applications (5)

Application Number Title Priority Date Filing Date
CH1581976A CH623317A5 (en) 1976-02-16 1976-12-16 Process for the preparation of benzamides
CH554480A CH622787A5 (en) 1976-02-16 1980-07-18 Process for the preparation of benzamides
CH554680A CH623577A5 (en) 1976-02-16 1980-07-18 Process for the preparation of benzamides
CH554380A CH622786A5 (en) 1976-02-16 1980-07-18 Process for the preparation of benzamides
CH554580A CH623576A5 (en) 1976-02-16 1980-07-18 Process for the preparation of benzamides

Family Applications After (4)

Application Number Title Priority Date Filing Date
CH554480A CH622787A5 (en) 1976-02-16 1980-07-18 Process for the preparation of benzamides
CH554680A CH623577A5 (en) 1976-02-16 1980-07-18 Process for the preparation of benzamides
CH554380A CH622786A5 (en) 1976-02-16 1980-07-18 Process for the preparation of benzamides
CH554580A CH623576A5 (en) 1976-02-16 1980-07-18 Process for the preparation of benzamides

Country Status (28)

Country Link
JP (1) JPS52100476A (es)
AR (2) AR214307A1 (es)
AT (5) AT345842B (es)
AU (1) AU506427B2 (es)
BE (1) BE851422A (es)
CA (1) CA1076112A (es)
CH (5) CH623317A5 (es)
DE (1) DE2706179C2 (es)
DK (1) DK148824C (es)
ES (4) ES455907A1 (es)
FI (1) FI65426C (es)
FR (1) FR2340940A1 (es)
GB (1) GB1512194A (es)
GR (1) GR62413B (es)
HR (1) HRP930495B1 (es)
IE (1) IE44482B1 (es)
IL (1) IL51406A (es)
LU (2) LU76771A1 (es)
MC (1) MC1136A1 (es)
NL (2) NL179382C (es)
NO (2) NO148417C (es)
NZ (1) NZ183316A (es)
PH (1) PH12847A (es)
PT (1) PT66195B (es)
SE (1) SE426822B (es)
SI (1) SI7710060A8 (es)
YU (1) YU39983B (es)
ZA (1) ZA77746B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4829506B2 (ja) * 2004-02-17 2011-12-07 石原産業株式会社 チオアミド系化合物又はその塩、並びにそれらを含有するサイトカイン産生抑制剤
ATE414694T1 (de) * 2005-05-03 2008-12-15 Bayer Cropscience Sa Neue heterocyclylethylbenzamid-derivate
RU2570898C2 (ru) * 2014-03-27 2015-12-20 Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Российский химико-технологический университет имени Д.И. Менделеева (РХТУ им. Д.И. Менделеева)" Способ получения n-[2-(морфолин-4-ил)этил]-4-хлорбензамида (варианты)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH451142A (de) * 1965-01-19 1968-05-15 Sandoz Ag Verfahren zur Herstellung neuer basisch substituierter Benzoesäureamide
FR1501846A (fr) * 1966-09-26 1967-11-18 Bellon Labor Sa Roger Procédé amélioré pour la préparation des thioamides
US3787419A (en) * 1971-07-01 1974-01-22 American Home Prod N-substituted-alpha,alpha,alpha-trifluoro-m-toluamides

Also Published As

Publication number Publication date
IL51406A0 (en) 1977-04-29
CA1076112A (en) 1980-04-22
DK51677A (da) 1977-08-17
ES467449A1 (es) 1978-10-16
HRP930495B1 (en) 1996-10-31
ES455907A1 (es) 1978-05-01
NL179382B (nl) 1986-04-01
ATA107076A (de) 1978-02-15
IE44482B1 (en) 1981-12-16
AT345842B (de) 1978-10-10
AT349481B (de) 1979-04-10
SE7701669L (sv) 1977-08-17
NL930082I2 (nl) 1994-08-16
LU88300I2 (de) 1994-09-09
YU6077A (en) 1983-01-21
MC1136A1 (fr) 1977-11-18
NL930082I1 (nl) 1993-09-16
AT349479B (de) 1979-04-10
NZ183316A (en) 1979-04-26
BE851422A (fr) 1977-08-16
SE426822B (sv) 1983-02-14
FI65426C (fi) 1984-05-10
ZA77746B (en) 1977-12-28
JPS6215547B2 (es) 1987-04-08
FR2340940B1 (es) 1981-01-09
LU76771A1 (es) 1978-04-13
GR62413B (en) 1979-04-11
ATA25778A (de) 1978-09-15
AR212554A1 (es) 1978-07-31
NO1994008I1 (no) 1994-08-03
IL51406A (en) 1979-12-30
DK148824B (da) 1985-10-14
AU506427B2 (en) 1980-01-03
AR214307A1 (es) 1979-05-31
PH12847A (en) 1979-09-12
DK148824C (da) 1986-04-21
GB1512194A (en) 1978-05-24
ATA25878A (de) 1978-09-15
NO148417C (no) 1983-10-12
DE2706179C2 (de) 1984-02-02
CH623576A5 (en) 1981-06-15
PT66195B (fr) 1979-01-17
IE44482L (en) 1977-08-16
NL7701144A (nl) 1977-08-18
NO148417B (no) 1983-06-27
AT349480B (de) 1979-04-10
ATA25678A (de) 1978-09-15
CH623577A5 (en) 1981-06-15
FR2340940A1 (fr) 1977-09-09
NL179382C (nl) 1986-09-01
PT66195A (fr) 1977-03-01
FI65426B (fi) 1984-01-31
YU39983B (en) 1985-06-30
DE2706179A1 (de) 1977-08-18
FI770356A (es) 1977-08-17
CH622787A5 (en) 1981-04-30
AU2109977A (en) 1978-07-13
ES467455A1 (es) 1978-10-16
AT349482B (de) 1979-04-10
SI7710060A8 (en) 1996-12-31
ATA25578A (de) 1978-09-15
CH622786A5 (en) 1981-04-30
JPS52100476A (en) 1977-08-23
NO770488L (no) 1977-08-17
ES467448A1 (es) 1978-10-16

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Legal Events

Date Code Title Description
PUE Assignment

Owner name: F. HOFFMANN-LA ROCHE AG

SPCF Supplementary protection certificate filed

Free format text: IKS 50085/900308, 951106

SPCF Supplementary protection certificate filed

Free format text: IKS 50085/900308, 951106

SPCG Supplementary protection certificate granted

Free format text: IKS 50085/900308, 951106, EXPIRES:20011215

PL Patent ceased
SPCL Supplementary protection certificate deletion