CH619468A5 - - Google Patents

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Publication number
CH619468A5
CH619468A5 CH26976A CH26976A CH619468A5 CH 619468 A5 CH619468 A5 CH 619468A5 CH 26976 A CH26976 A CH 26976A CH 26976 A CH26976 A CH 26976A CH 619468 A5 CH619468 A5 CH 619468A5
Authority
CH
Switzerland
Prior art keywords
methylene chloride
formula
acid
compounds
solution
Prior art date
Application number
CH26976A
Other languages
German (de)
English (en)
Inventor
Paul Dr Stadler
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Priority to CH26976A priority Critical patent/CH619468A5/de
Priority to DK000577A priority patent/DK150490C/da
Priority to FI770008A priority patent/FI62094C/fi
Priority to DE19772700234 priority patent/DE2700234A1/de
Priority to SE7700084A priority patent/SE434401B/xx
Priority to US05/757,616 priority patent/US4145549A/en
Priority to NL7700124A priority patent/NL7700124A/xx
Priority to HU77SA3003A priority patent/HU176871B/hu
Priority to IE43/77A priority patent/IE44560B1/en
Priority to ES454917A priority patent/ES454917A1/es
Priority to CA269,389A priority patent/CA1108128A/en
Priority to NZ183045A priority patent/NZ183045A/xx
Priority to CS77170A priority patent/CS200205B2/cs
Priority to JP123977A priority patent/JPS5287197A/ja
Priority to GB916/77A priority patent/GB1571835A/en
Priority to AU21228/77A priority patent/AU512003B2/en
Priority to AT0008777A priority patent/AT364817B/de
Priority to SU772439829A priority patent/SU725565A3/ru
Priority to ZA00770151A priority patent/ZA77151B/xx
Priority to BE174010A priority patent/BE850304A/xx
Priority to YU62/77A priority patent/YU39377B/xx
Priority to FR7700760A priority patent/FR2337727A1/fr
Publication of CH619468A5 publication Critical patent/CH619468A5/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/081—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing O or S as heteroatoms, e.g. Cys, Ser
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CH26976A 1976-01-12 1976-01-12 CH619468A5 (fi)

Priority Applications (22)

Application Number Priority Date Filing Date Title
CH26976A CH619468A5 (fi) 1976-01-12 1976-01-12
DK000577A DK150490C (da) 1976-01-12 1977-01-03 Fremgangsmaade til fremstilling af 2-aminooctahydro-oxazolo-(3,2-a)pyrrolo(2,1-c)pyrazinderivater
FI770008A FI62094C (fi) 1976-01-12 1977-01-03 Foerfarande foer framstaellning av 2-amino-oktahydro-oxazolo(3,2-a)pyrrolo(2,1-c)pyratzinderivat
DE19772700234 DE2700234A1 (de) 1976-01-12 1977-01-05 Organische verbindungen und verfahren zu deren herstellung
SE7700084A SE434401B (sv) 1976-01-12 1977-01-05 Forfarande for framstellning av 2-karbobensoxiamino-oktahydro-oxazolo(3,2-a)pyrrolo(2,1-c)pyrazinderivat
US05/757,616 US4145549A (en) 1976-01-12 1977-01-07 Process for preparing oxazolo 3,2-a!pyrrolo 2,1-c!pyrazine derivatives
NL7700124A NL7700124A (nl) 1976-01-12 1977-01-07 Werkwijzen voor het bereiden en toepassen van heterocyclische verbindingen.
HU77SA3003A HU176871B (en) 1976-01-12 1977-01-10 Process for producing 2-amino-oktahydro-oxasolo-square bracket-3,2-a-square bracket closed-pyrrolo-square bracket-2,1-c-square bracket closed-pyrasine derivatives
IE43/77A IE44560B1 (en) 1976-01-12 1977-01-10 Aminicyclols
ES454917A ES454917A1 (es) 1976-01-12 1977-01-10 Procedimiento para la produccion de aminocicloles.
CA269,389A CA1108128A (en) 1976-01-12 1977-01-10 Cyclization process for an ergot alkaloid
NZ183045A NZ183045A (en) 1976-01-12 1977-01-10 Aminocylol production
CS77170A CS200205B2 (en) 1976-01-12 1977-01-11 Method of producing aminocyclols
JP123977A JPS5287197A (en) 1976-01-12 1977-01-11 Improvement in organic compound
GB916/77A GB1571835A (en) 1976-01-12 1977-01-11 Aminocyclols
AU21228/77A AU512003B2 (en) 1976-01-12 1977-01-11 Oxazolo(3, 2-a) pyrolo-2-(2, 1-c) pyrazine derivatives
AT0008777A AT364817B (de) 1976-01-12 1977-01-11 Verfahren zur herstellung von aminocyclolen
SU772439829A SU725565A3 (ru) 1976-01-12 1977-01-12 Способ получени производных октагидрооксазоло/3,2-а/пирроло /2,1-с/пиразина
ZA00770151A ZA77151B (en) 1976-01-12 1977-01-12 Improvements in or relating to organic compounds
BE174010A BE850304A (fr) 1976-01-12 1977-01-12 Procede de preparation de composes peptidiques
YU62/77A YU39377B (en) 1976-01-12 1977-01-12 Process for the manufacture of aminocyclols
FR7700760A FR2337727A1 (fr) 1976-01-12 1977-01-12 Procede de preparation de composes peptidiques

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH26976A CH619468A5 (fi) 1976-01-12 1976-01-12

Publications (1)

Publication Number Publication Date
CH619468A5 true CH619468A5 (fi) 1980-09-30

Family

ID=4183149

Family Applications (1)

Application Number Title Priority Date Filing Date
CH26976A CH619468A5 (fi) 1976-01-12 1976-01-12

Country Status (22)

Country Link
US (1) US4145549A (fi)
JP (1) JPS5287197A (fi)
AT (1) AT364817B (fi)
AU (1) AU512003B2 (fi)
BE (1) BE850304A (fi)
CA (1) CA1108128A (fi)
CH (1) CH619468A5 (fi)
CS (1) CS200205B2 (fi)
DE (1) DE2700234A1 (fi)
DK (1) DK150490C (fi)
ES (1) ES454917A1 (fi)
FI (1) FI62094C (fi)
FR (1) FR2337727A1 (fi)
GB (1) GB1571835A (fi)
HU (1) HU176871B (fi)
IE (1) IE44560B1 (fi)
NL (1) NL7700124A (fi)
NZ (1) NZ183045A (fi)
SE (1) SE434401B (fi)
SU (1) SU725565A3 (fi)
YU (1) YU39377B (fi)
ZA (1) ZA77151B (fi)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1584464A (en) * 1977-04-19 1981-02-11 Farmaceutici Italia Ergot alkaloids
JPS5423487U (fi) * 1977-07-19 1979-02-15
EP0003286B1 (de) * 1978-01-20 1982-03-24 Sandoz Ag Ergopeptidalkaloid-Derivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zusammensetzungen
YU41110B (en) * 1978-07-19 1986-12-31 Lek Tovarna Farmacevtskih Process for preparing dextrorotatory ergot alcaloids acid addition salts
DE3303616A1 (de) * 1982-02-12 1983-08-25 Sandoz-Patent-GmbH, 7850 Lörrach Mutterkornalkaloide, verfahren zu deren herstellung sowie diese verbindungen enthaltende pharmazeutische zubereitungen
RU2266906C1 (ru) * 2004-04-29 2005-12-27 Общество с ограниченной ответственностью "Исследовательский Институт Химического Разнообразия" (ООО "Исследовательский Институт Химического Разнообразия") Анелированные карбамоилазагетероциклы, способы их получения (варианты), фармацевтическая композиция, фокусированная библиотека
US20080161324A1 (en) * 2006-09-14 2008-07-03 Johansen Lisa M Compositions and methods for treatment of viral diseases

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2533698A (en) * 1950-12-12 Urethanes containing the lysergic
CH507249A (de) * 1968-05-31 1971-05-15 Sandoz Ag Verfahren zur Herstellung von 2-Brom-a-ergokryptin
GB1298277A (en) * 1969-04-18 1972-11-29 Sandoz Ltd Preparation of ergot peptide alkaloids
JPS4735440A (fi) * 1971-03-29 1972-11-25
CH581136A5 (fi) * 1972-09-26 1976-10-29 Sandoz Ag
SE397093B (sv) * 1973-07-09 1977-10-17 Sandoz Ag Forfarande for framstellning av oktahydro-oxazolo(3,2-a)pyrrolo(2,1-c)pyrazinderivat
CH587858A5 (fi) * 1973-11-28 1977-05-13 Sandoz Ag
DE2525962A1 (de) * 1974-06-21 1976-01-08 Sandoz Ag Neue heterocyclische verbindungen, ihre herstellung und verwendung
CH601321A5 (fi) * 1975-01-06 1978-07-14 Sandoz Ag

Also Published As

Publication number Publication date
SU725565A3 (ru) 1980-03-30
FI62094C (fi) 1982-11-10
FR2337727B1 (fi) 1980-04-30
SE434401B (sv) 1984-07-23
FR2337727A1 (fr) 1977-08-05
IE44560B1 (en) 1982-01-13
HU176871B (en) 1981-05-28
BE850304A (fr) 1977-07-12
IE44560L (en) 1977-07-12
GB1571835A (en) 1980-07-23
CS200205B2 (en) 1980-08-29
FI62094B (fi) 1982-07-30
YU6277A (en) 1982-10-31
ES454917A1 (es) 1978-04-01
AU2122877A (en) 1978-07-20
ZA77151B (en) 1978-08-30
NL7700124A (nl) 1977-07-14
DK577A (da) 1977-07-13
AU512003B2 (en) 1980-09-18
CA1108128A (en) 1981-09-01
DE2700234A1 (de) 1977-07-14
DK150490C (da) 1987-10-19
US4145549A (en) 1979-03-20
NZ183045A (en) 1979-03-16
FI770008A (fi) 1977-07-13
DK150490B (da) 1987-03-09
JPS5287197A (en) 1977-07-20
ATA8777A (de) 1981-04-15
AT364817B (de) 1981-11-25
YU39377B (en) 1984-12-31

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PL Patent ceased