CH618972A5 - - Google Patents

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Publication number
CH618972A5
CH618972A5 CH691676A CH691676A CH618972A5 CH 618972 A5 CH618972 A5 CH 618972A5 CH 691676 A CH691676 A CH 691676A CH 691676 A CH691676 A CH 691676A CH 618972 A5 CH618972 A5 CH 618972A5
Authority
CH
Switzerland
Prior art keywords
alkyl
phenyl
benzyl
methyl
cycloalkyl
Prior art date
Application number
CH691676A
Other languages
English (en)
French (fr)
Inventor
Roger Garrick Harrison
William Boffey Jamieson
William James Ross
John Christopher Saunders
Original Assignee
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd
Publication of CH618972A5 publication Critical patent/CH618972A5/fr

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38Nitrogen atoms
    • C07D231/40Acylated on said nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88Nitrogen atoms, e.g. allantoin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/041,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • C07D249/061,2,3-Triazoles; Hydrogenated 1,2,3-triazoles with aryl radicals directly attached to ring atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/101,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/14Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D257/00Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04Five-membered rings
    • C07D257/06Five-membered rings with nitrogen atoms directly attached to the ring carbon atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH691676A 1975-06-05 1976-06-02 CH618972A5 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB24225/75A GB1547564A (en) 1975-06-05 1975-06-05 Acylated amino-heteroaryl compounds

Publications (1)

Publication Number Publication Date
CH618972A5 true CH618972A5 (pl) 1980-08-29

Family

ID=10208295

Family Applications (2)

Application Number Title Priority Date Filing Date
CH691676A CH618972A5 (pl) 1975-06-05 1976-06-02
CH49980A CH622254A5 (pl) 1975-06-05 1980-01-22

Family Applications After (1)

Application Number Title Priority Date Filing Date
CH49980A CH622254A5 (pl) 1975-06-05 1980-01-22

Country Status (31)

Country Link
US (2) US4166123A (pl)
JP (1) JPS51146465A (pl)
AR (2) AR219280A1 (pl)
AT (1) AT355562B (pl)
AU (1) AU506564B2 (pl)
BE (1) BE842578A (pl)
BG (2) BG26515A3 (pl)
CA (1) CA1081219A (pl)
CH (2) CH618972A5 (pl)
CS (1) CS219320B2 (pl)
DD (1) DD125206A5 (pl)
DE (1) DE2625227A1 (pl)
DK (1) DK243576A (pl)
ES (2) ES448477A1 (pl)
FR (1) FR2313046A1 (pl)
GB (1) GB1547564A (pl)
GR (1) GR60336B (pl)
HU (1) HU174190B (pl)
IE (1) IE43579B1 (pl)
IL (1) IL49691A (pl)
MX (1) MX3638E (pl)
NL (1) NL7606179A (pl)
NZ (1) NZ181010A (pl)
PH (1) PH14627A (pl)
PL (2) PL101468B1 (pl)
PT (1) PT65180B (pl)
RO (1) RO70771A (pl)
SE (1) SE431646B (pl)
SU (2) SU648094A3 (pl)
YU (2) YU137276A (pl)
ZA (1) ZA763210B (pl)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7810634A (nl) * 1977-10-28 1979-05-02 May & Baker Ltd Tetrazool-derivaten.
NO800583L (no) * 1979-03-02 1980-09-03 Glaxo Group Ltd Fremgangsmaate for fremstilling av farmakologisk aktive triazolderivater
US4801718A (en) * 1980-09-16 1989-01-31 Eli Lilly And Company Thiaiazolyl benzamides
US4943634A (en) * 1980-09-16 1990-07-24 Eli Lilly And Company N-heterocyclic benzamides
US5086184A (en) * 1980-09-16 1992-02-04 Dowelanco N-heterocyclic benzamides
MA19269A1 (fr) * 1980-09-16 1982-04-01 Lilly Co Eli Perfectionnement relatif a des derives de n-arylbenzamides .
DE3100516A1 (de) * 1981-01-10 1982-08-12 C.H. Boehringer Sohn, 6507 Ingelheim Pyridylaminobenzoesaeuren, ihre herstellung und verwendung
US5464860A (en) * 1988-11-30 1995-11-07 Novapharme N(pyrazol-3-yl) benzamides and pharmaceutical compositions
FR2662692B1 (fr) * 1990-05-30 1995-04-28 Novapharme Derives heterocycliques doues d'activite anticonvulsivante, procede de preparation et composition pharmaceutique.
US5258397A (en) * 1988-11-30 1993-11-02 Novapharme 3-Isoxazoyl derivatives endowed with anticonvulsant activity, procedure for their preparation and their pharmaceutical compositions
US5073566A (en) * 1989-11-30 1991-12-17 Eli Lilly And Company Angiotensin ii antagonist 1,3-imidazoles and use thereas
US5612360A (en) * 1992-06-03 1997-03-18 Eli Lilly And Company Angiotensin II antagonists
US5401851A (en) * 1992-06-03 1995-03-28 Eli Lilly And Company Angiotensin II antagonists
WO1998024768A1 (fr) * 1996-12-03 1998-06-11 Banyu Pharmaceutical Co., Ltd. Nouveaux derives d'uree
DE69719544T2 (de) * 1996-12-12 2003-11-06 Banyu Pharma Co Ltd Pyrazolderivate
EP0945439B1 (en) * 1996-12-13 2003-03-19 Banyu Pharmaceutical Co., Ltd. Aminopyrazole derivatives
DE69729315T2 (de) 1996-12-16 2005-06-23 Banyu Pharmaceutical Co., Ltd. Aminopyrazolderivate
US6906069B1 (en) 1999-01-08 2005-06-14 Amgen Inc. LXR modulators
WO2001060818A1 (en) * 2000-02-14 2001-08-23 Tularik Inc. Lxr modulators
US6673543B2 (en) 2000-04-05 2004-01-06 Tularik, Inc. Solid phase synthesis of LXR ligands
WO2002023986A1 (fr) * 2000-08-25 2002-03-28 Sankyo Company, Limited Derives de 4-acylaminopyrazole
WO2003063796A2 (en) * 2002-01-30 2003-08-07 Tularik Inc. Heterocyclic arylsulfonamidobenzylic compounds
US7335779B2 (en) * 2002-03-08 2008-02-26 Quonova, Llc Modulation of pathogenicity
KR100849021B1 (ko) 2007-06-19 2008-07-29 (주)더페이스샵코리아 카페익산 유도체 및 이를 함유하는 조성물
BR102020008433A2 (pt) 2020-04-28 2021-11-03 Universidade Federal Do Parana Repelentes de artrópodes obtidos a partir da transformação química de ácido lático, lactatos ou outros derivados do ácido lático

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA698428A (en) 1964-11-24 W. Lynn John Substituted triazole compounds and polymerization products thereof
US2467895A (en) * 1946-04-12 1949-04-19 American Cyanamid Co Piperazine derivatives and method of preparing the same
US2953491A (en) * 1957-11-21 1960-09-20 American Cyanamid Co Fungicide
US2914536A (en) * 1957-11-21 1959-11-24 American Cyanamid Co Novel 3-acylamino triazoles
GB1111680A (en) 1965-12-01 1968-05-01 Shell Int Research Improvements in or relating to ester-base compositions
US3457350A (en) * 1966-10-26 1969-07-22 American Cyanamid Co Method of treating asthma
GB1497536A (en) 1973-12-17 1978-01-12 Lilly Industries Ltd 2-acylaminooxazoles methods for their preparation and their use

Also Published As

Publication number Publication date
GR60336B (en) 1978-05-09
GB1547564A (en) 1979-06-20
SE7606225L (sv) 1976-12-06
CS219320B2 (en) 1983-03-25
AR219280A1 (es) 1980-08-15
US4089962A (en) 1978-05-16
RO70771A (ro) 1983-08-03
US4166123A (en) 1979-08-28
CA1081219A (en) 1980-07-08
AR217662A1 (es) 1980-04-15
ATA412376A (de) 1979-08-15
NZ181010A (en) 1978-04-28
BG25211A3 (en) 1978-08-10
IE43579L (en) 1976-12-05
BE842578A (fr) 1976-12-03
PT65180B (en) 1978-11-06
JPS51146465A (en) 1976-12-16
IE43579B1 (en) 1981-04-08
SE431646B (sv) 1984-02-20
IL49691A0 (en) 1976-07-30
IL49691A (en) 1980-09-16
PL101468B1 (pl) 1978-12-30
SU648094A3 (ru) 1979-02-15
AU506564B2 (en) 1980-01-10
BG26515A3 (pl) 1979-04-12
HU174190B (hu) 1979-11-28
YU123376A (en) 1982-10-31
DD125206A5 (pl) 1977-04-06
YU137276A (en) 1982-10-31
ES460711A1 (es) 1978-04-16
ES448477A1 (es) 1977-11-01
AU1461876A (en) 1977-12-08
PL101455B1 (pl) 1978-12-30
ZA763210B (en) 1978-01-25
NL7606179A (nl) 1976-12-07
CH622254A5 (pl) 1981-03-31
RO70771B (ro) 1983-07-30
PH14627A (en) 1981-10-12
PT65180A (en) 1976-07-01
DE2625227A1 (de) 1976-12-23
AT355562B (de) 1980-03-10
MX3638E (es) 1981-04-13
DK243576A (da) 1976-12-06
FR2313046A1 (fr) 1976-12-31
SU654168A3 (ru) 1979-03-25
FR2313046B1 (pl) 1982-09-24

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PL Patent ceased