CH569012A5 - 4-piperidylidene benzocycloheptathiophenes - - antihistamines and serotonin and acetyl choline inhibitors - Google Patents

4-piperidylidene benzocycloheptathiophenes - - antihistamines and serotonin and acetyl choline inhibitors

Info

Publication number
CH569012A5
CH569012A5 CH98672A CH98672A CH569012A5 CH 569012 A5 CH569012 A5 CH 569012A5 CH 98672 A CH98672 A CH 98672A CH 98672 A CH98672 A CH 98672A CH 569012 A5 CH569012 A5 CH 569012A5
Authority
CH
Switzerland
Prior art keywords
piperidylidene
benzo
thiophen
halogen
formula
Prior art date
Application number
CH98672A
Other languages
German (de)
English (en)
Inventor
J P Bourquin
G Schwarb
E Waldvogel
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to BE794377D priority Critical patent/BE794377A/xx
Application filed by Sandoz Ag filed Critical Sandoz Ag
Priority to CH98672A priority patent/CH569012A5/de
Priority to US286281A priority patent/US3862156A/en
Priority to JP47117590A priority patent/JPS5760351B2/ja
Priority to DD167577A priority patent/DD102701A5/xx
Priority to SE7300501A priority patent/SE383347B/sv
Priority to FI110/73A priority patent/FI55843C/fi
Priority to NL7300796A priority patent/NL7300796A/xx
Priority to GB311873A priority patent/GB1415591A/en
Priority to HUSA2447A priority patent/HU165130B/hu
Priority to CY992A priority patent/CY992A/xx
Priority to DE2302944A priority patent/DE2302944C2/de
Priority to CS7300000504A priority patent/CS179977B2/cs
Priority to AU51377/73A priority patent/AU482530B2/en
Priority to FR7302444A priority patent/FR2183663B2/fr
Priority to SU2017993A priority patent/SU520914A3/ru
Priority to ES438598A priority patent/ES438598A1/es
Priority to AT685675A priority patent/AT337181B/de
Publication of CH569012A5 publication Critical patent/CH569012A5/de
Priority to SE7600275A priority patent/SE423712B/sv
Priority to DK16376A priority patent/DK16376A/da
Priority to FI790145A priority patent/FI59591C/fi
Priority to HK112/79A priority patent/HK11279A/xx
Priority to MY114/79A priority patent/MY7900114A/xx
Priority to JP55175690A priority patent/JPS5817756B2/ja

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/08—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing alicyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CH98672A 1972-01-24 1972-01-24 4-piperidylidene benzocycloheptathiophenes - - antihistamines and serotonin and acetyl choline inhibitors CH569012A5 (en)

Priority Applications (24)

Application Number Priority Date Filing Date Title
BE794377D BE794377A (fr) 1972-01-24 Nouveaux derives du benzo-cyclohepta-thiophene
CH98672A CH569012A5 (en) 1972-01-24 1972-01-24 4-piperidylidene benzocycloheptathiophenes - - antihistamines and serotonin and acetyl choline inhibitors
US286281A US3862156A (en) 1972-01-24 1972-09-05 4h-benzo{8 4,5{9 cyclohepta{8 1,2-6{9 thiophenes
JP47117590A JPS5760351B2 (sv) 1972-01-24 1972-11-22
DD167577A DD102701A5 (sv) 1972-01-24 1972-12-15
SE7300501A SE383347B (sv) 1972-01-24 1973-01-15 Forfarande for framstellning av nya 4 h-benso (4,5)cyklohepta (1,2-b)tiofenderivat
FI110/73A FI55843C (fi) 1972-01-24 1973-01-16 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 9,10-dihydro-9- eller -10-hydroxi-imino-4-(1-alkyl-4-piperidyliden)-4h-benso(4,5)cyklohepta(1,2-b)tiofenderivat och deras syraadditionssalter
NL7300796A NL7300796A (sv) 1972-01-24 1973-01-19
DE2302944A DE2302944C2 (de) 1972-01-24 1973-01-22 9,10-Dihydro-4-(1-subst.-4-piperidyliden)-4H-benzol [4,5] cyclohepta [1,2-b] thiophene, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
HUSA2447A HU165130B (sv) 1972-01-24 1973-01-22
CY992A CY992A (en) 1972-01-24 1973-01-22 Benzocycloheptathiophene derivatives
GB311873A GB1415591A (en) 1972-01-24 1973-01-22 Benzocycloheptathiophene derivatives
CS7300000504A CS179977B2 (en) 1972-01-24 1973-01-23 Method for producing novel derivatives of benzocycloheptathiophenone
AU51377/73A AU482530B2 (en) 1973-01-23 Benzocycloheptathiophenes
FR7302444A FR2183663B2 (sv) 1972-01-24 1973-01-24
SU2017993A SU520914A3 (ru) 1972-01-24 1974-04-23 Способ получени производных бензоциклогептатиофенонов или их солей
ES438598A ES438598A1 (es) 1972-01-24 1975-06-16 Procedimiento para la obtencion de derivados de benzocilo- heptatiofeno.
AT685675A AT337181B (de) 1972-01-24 1975-09-05 Verfahren zur herstellung neuer 4-(4-piperidyliden)-4h-benzo(4,5)cyclohepta(1,2-b)thiophen-derivate und ihrer saureadditionssalze
SE7600275A SE423712B (sv) 1972-01-24 1976-01-13 Forfarande for framstellning av 4-(1-bensyl-4-piperidyliden)-4h-benso-/4.5/cyklohepta/1,2-b/-tiofen-10(9h) /eller 9 (10h) /-on-derivat
DK16376A DK16376A (da) 1972-01-24 1976-01-15 Fremgangsmade til fremstilling af terapeutisk aktive 4h-benzo(4,5)cyclohepta(1,2-b)thiophenderivater
FI790145A FI59591C (fi) 1972-01-24 1979-01-17 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara 4h-benso(4,5)syklohepta(1,2-b)tiofen-derivat
HK112/79A HK11279A (en) 1972-01-24 1979-03-08 Benzocycloheptathiophene derivatives
MY114/79A MY7900114A (en) 1972-01-24 1979-12-30 Benzocycloheptathiophene derivatives
JP55175690A JPS5817756B2 (ja) 1972-01-24 1980-12-11 ４Ｈ−ベンゾ〔４，５〕シクロヘプタ〔１，２−ｂ〕チオフエン誘導体の製法

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH98672A CH569012A5 (en) 1972-01-24 1972-01-24 4-piperidylidene benzocycloheptathiophenes - - antihistamines and serotonin and acetyl choline inhibitors

Publications (1)

Publication Number Publication Date
CH569012A5 true CH569012A5 (en) 1975-11-14

Family

ID=4199812

Family Applications (1)

Application Number Title Priority Date Filing Date
CH98672A CH569012A5 (en) 1972-01-24 1972-01-24 4-piperidylidene benzocycloheptathiophenes - - antihistamines and serotonin and acetyl choline inhibitors

Country Status (6)

Country Link
JP (1) JPS5817756B2 (sv)
CH (1) CH569012A5 (sv)
CS (1) CS179977B2 (sv)
ES (1) ES438598A1 (sv)
SE (1) SE423712B (sv)
SU (1) SU520914A3 (sv)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS649343U (sv) * 1987-07-07 1989-01-19

Also Published As

Publication number Publication date
ES438598A1 (es) 1977-05-16
CS179977B2 (en) 1977-12-30
AU5137773A (en) 1974-07-25
JPS57112390A (en) 1982-07-13
SE7600275L (sv) 1976-01-13
JPS5817756B2 (ja) 1983-04-09
SE423712B (sv) 1982-05-24
SU520914A3 (ru) 1976-07-05

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