CH436299A - Verfahren zur Herstellung von neuen Penicillinen - Google Patents
Verfahren zur Herstellung von neuen PenicillinenInfo
- Publication number
- CH436299A CH436299A CH524163A CH524163A CH436299A CH 436299 A CH436299 A CH 436299A CH 524163 A CH524163 A CH 524163A CH 524163 A CH524163 A CH 524163A CH 436299 A CH436299 A CH 436299A
- Authority
- CH
- Switzerland
- Prior art keywords
- acid
- solution
- mol
- salt
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
- C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
- C07D499/60—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
- C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
- C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
- C07D499/70—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with hetero rings as additional substituents on the carbon chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/76—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with hetero rings directly attached to the carboxamido radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Catalysts (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US19077462A | 1962-04-27 | 1962-04-27 | |
US19079562A | 1962-04-27 | 1962-04-27 | |
US19077662A | 1962-04-27 | 1962-04-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
CH436299A true CH436299A (de) | 1967-05-31 |
Family
ID=27392795
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CH524163A CH436299A (de) | 1962-04-27 | 1963-04-26 | Verfahren zur Herstellung von neuen Penicillinen |
Country Status (4)
Country | Link |
---|---|
CH (1) | CH436299A (el) |
DE (1) | DE1289053B (el) |
ES (1) | ES287497A1 (el) |
GB (1) | GB1051723A (el) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4918067A (en) * | 1986-07-24 | 1990-04-17 | Beecham Group P.L.C. | Heterocyclic substituted penicillin antibiotics |
ES2535516T3 (es) * | 2008-04-24 | 2015-05-12 | F2G Limited | Agentes antifúngicos de pirrol |
EP3415511A1 (en) | 2014-11-21 | 2018-12-19 | F2G Limited | Antifungal agents |
GB201609222D0 (en) | 2016-05-25 | 2016-07-06 | F2G Ltd | Pharmaceutical formulation |
US11819503B2 (en) | 2019-04-23 | 2023-11-21 | F2G Ltd | Method of treating coccidioides infection |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR61M (el) * | 1959-08-03 | 1961-01-09 | ||
US2996501A (en) * | 1960-03-31 | 1961-08-15 | Doyle Frank Peter | Synthetic penicillins |
-
0
- GB GB1051723D patent/GB1051723A/en active Active
-
1963
- 1963-04-23 DE DE1963B0071594 patent/DE1289053B/de active Pending
- 1963-04-26 CH CH524163A patent/CH436299A/de unknown
- 1963-04-27 ES ES287497A patent/ES287497A1/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
DE1289053B (de) | 1969-02-13 |
ES287497A1 (es) | 1963-12-01 |
GB1051723A (el) |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DE2448966A1 (de) | Penicillinderivate | |
DE1695602A1 (de) | Verfahren zur Herstellung von 1,2-disubstituierten Vinylverbindungen und deren Saeureanlagerungssalzen | |
DE2158855A1 (de) | Heterocyclisch substituierte Ureidocephalosporine | |
DE1963645C3 (de) | Verfahren zur Herstellung von Penicillinen | |
CH436299A (de) | Verfahren zur Herstellung von neuen Penicillinen | |
DE1670222C3 (de) | a-(Benzyloxycarbonyl)-thienyunethylpenicilline und deren Salze, Verfahren zu deren Herstellung und diese Verbindungen enthaltende antibakterielle Mittel | |
DE2225149C2 (de) | Oxofurylesterderivate der 6-(ą-Aminophenylacetamido)penicillansäure, Verfahren zu deren Herstellung und ihre Verwendung | |
DE2320040A1 (de) | Verfahren zur herstellung von 7acylamino-desacetoxy-cephalosporansaeureester | |
AT260420B (de) | Verfahren zur Herstellung neuer Penicillinderivate | |
CH521374A (de) | Verfahren zur Herstellung von 7-(a-(4-Pyridylthio)-acetamido)- 3-cephem-4-carbonsäuren | |
DE1929997C2 (de) | Acylureidopenicilline, Verfahren zu ihrer Herstellung und antibakterielle Mittel, die diese Verbindungen enthalten | |
DE2053886C3 (de) | Verfahren zur Herstellung von kristallinem Mononatrium- oder Monokaliumalpha- carboxybenzyl penicillin | |
DE2400489B2 (de) | Salze aus D- oder L-N-Methylephedrin und Enamin-Derivaten von a -Aminomonocarbonsäuren, Verfahren zu deren Herstellung und deren Verwendung | |
DE2325498A1 (de) | Penicillinverbindungen und verfahren zu ihrer herstellung | |
DE2265590C2 (de) | 7-Amino-3-[S-(1,2,3-triazol-5-yl)-thiomethyl]-3-cephem-4-carbonsäure und deren Verwendung | |
AT259132B (de) | Verfahren zur Herstellung von neuen Penicillinderivaten | |
CH625805A5 (el) | ||
DE2841706C2 (de) | N,N-Dimethylacetamid-Addukt der 7-[D(-)-α-(4-Äthyl-2,3-dioxo-1-piperazincarboxamido)-α-(4-hydroxyphenyl)-acetamido]-3-[5-(1-methyl-1,2,3,4-tetrazolyl)-thiomethyl]-Δ↑3↑-cephem--4-carbonsäure, Verfahren zu seiner Herstellung und seine Verwendung | |
DE2423048A1 (de) | Verfahren zur herstellung eines kristallinen solvats eines alkali- oder erdalkalimetallsalzes von 6-(d-alphaamino-p-hydroxyphenylacetamido) -penicillansaeure | |
DE1670115A1 (de) | Penicillansaeurederivate und Verfahren zu ihrer Herstellung | |
EP0241005B1 (de) | Verfahren zur Herstellung von 4-Halogenmethylbenzaldehyd | |
EP0031951B1 (de) | Formylderivate von Hydrazinomethylpenicillinen, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel | |
DE2065879A1 (de) | Verfahren zur herstellung von dl-6- aminoacylamidopenicillansaeuren | |
DE69227890T2 (de) | Verfahren zur herstellung von 5-amino-3-methylpyrazol | |
AT254857B (de) | Verfahren zur Herstellung von neuen Naphthalinverbindungen |