CA3178291A1 - Method for the management of dysmenorrhea and menstrual pain - Google Patents
Method for the management of dysmenorrhea and menstrual painInfo
- Publication number
- CA3178291A1 CA3178291A1 CA3178291A CA3178291A CA3178291A1 CA 3178291 A1 CA3178291 A1 CA 3178291A1 CA 3178291 A CA3178291 A CA 3178291A CA 3178291 A CA3178291 A CA 3178291A CA 3178291 A1 CA3178291 A1 CA 3178291A1
- Authority
- CA
- Canada
- Prior art keywords
- composition
- estetrol
- dysmenorrhea
- hemostatic
- treatment
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/566—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol having an oxo group in position 17, e.g. estrone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
- A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
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- Animal Behavior & Ethology (AREA)
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- Reproductive Health (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Bioinformatics & Cheminformatics (AREA)
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- Gynecology & Obstetrics (AREA)
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| CA3178291A CA3178291A1 (en) | 2016-08-05 | 2016-10-28 | Method for the management of dysmenorrhea and menstrual pain |
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| EP16183025 | 2016-08-05 | ||
| CA3178291A CA3178291A1 (en) | 2016-08-05 | 2016-10-28 | Method for the management of dysmenorrhea and menstrual pain |
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| CA3041016A CA3041016C (en) | 2016-10-28 | 2016-10-28 | Method for the management of dysmenorrhea and menstrual pain |
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| CN116077454A (zh) | 2015-06-18 | 2023-05-09 | 埃斯特拉有限责任公司 | 含雌四醇组分的口腔分散剂量单位 |
| ES2877186T3 (es) | 2015-06-18 | 2021-11-16 | Estetra Sprl | Comprimido orodispersable que contiene estetrol |
| JP6813150B2 (ja) | 2015-06-18 | 2021-01-13 | エステトラ ソシエテ プリーヴ ア レスポンサビリテ リミテ | エステトロールを含有する口腔内崩壊錠 |
| CA3178291A1 (en) * | 2016-08-05 | 2018-04-12 | Estetra Srl | Method for the management of dysmenorrhea and menstrual pain |
| MY205032A (en) * | 2016-10-28 | 2024-09-28 | Estetra Sprl | Method for the management of dysmenorrhea and menstrual pain |
| CA3178181A1 (en) * | 2018-02-07 | 2019-08-15 | Estetra Srl | Contraceptive composition with reduced cardiovascular effects |
| TWI801561B (zh) | 2018-04-19 | 2023-05-11 | 比利時商依思特拉私人有限責任公司 | 化合物及其用於緩解絕經相關症狀的用途 |
| JOP20200260A1 (ar) * | 2018-04-19 | 2019-10-19 | Estetra Sprl | مركبات واستخداماتها للتخفيف من الأعراض المصاحبة لانقطاع الطمث |
| DE102019115343A1 (de) * | 2019-06-06 | 2020-12-10 | EVESTRA GmbH | Vaginalring für die hormonelle Kontrazeption |
| HU231240B1 (hu) | 2019-09-03 | 2022-04-28 | Richter Gedeon Nyrt. | Ipari eljárás nagytisztaságú ösztetrol hatóanyag előállítására |
| TWI893101B (zh) | 2020-04-16 | 2025-08-11 | 比利時商埃斯特拉有限責任公司 | 具有降低之副作用之避孕組成物 |
| CL2021001762A1 (es) * | 2021-07-01 | 2022-01-21 | Univ Pontificia Catolica Chile | Uso del estetrol como tratamiento para la endometriosis |
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| US12233074B2 (en) | 2022-02-10 | 2025-02-25 | Estetra Srl | Contraceptive methods with improved pearl index |
| KR20250151374A (ko) * | 2023-02-23 | 2025-10-21 | 에스테트라, 소시에떼 아 레스폰서빌리떼 리미떼 | 통증의 완화 및 치료에 사용되는 에스테트롤 및 드로스피레논을 포함하는 조성물 |
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2016
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2017
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- 2017-08-07 PH PH1/2019/500172A patent/PH12019500172B1/en unknown
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| US20190167700A1 (en) | 2019-06-06 |
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| US11896602B2 (en) | 2024-02-13 |
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| BR112019002203A2 (pt) | 2019-05-14 |
| CO2019000672A2 (es) | 2019-04-30 |
| US20230041304A1 (en) | 2023-02-09 |
| MX2022011436A (es) | 2022-11-14 |
| AU2022231672A1 (en) | 2022-10-06 |
| PH12019500172B1 (en) | 2024-02-28 |
| JP6557298B2 (ja) | 2019-08-07 |
| JP2018165263A (ja) | 2018-10-25 |
| PE20190739A1 (es) | 2019-05-23 |
| PH12019500172A1 (en) | 2019-07-29 |
| WO2018024912A1 (en) | 2018-02-08 |
| JP7177313B2 (ja) | 2022-11-24 |
| KR20220144885A (ko) | 2022-10-27 |
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