CO2019000672A2 - Procedimiento de tratamiento de dismenorrea y dolor menstrual - Google Patents

Procedimiento de tratamiento de dismenorrea y dolor menstrual

Info

Publication number
CO2019000672A2
CO2019000672A2 CONC2019/0000672A CO2019000672A CO2019000672A2 CO 2019000672 A2 CO2019000672 A2 CO 2019000672A2 CO 2019000672 A CO2019000672 A CO 2019000672A CO 2019000672 A2 CO2019000672 A2 CO 2019000672A2
Authority
CO
Colombia
Prior art keywords
dysmenorrhea
estetrol
treatment procedure
pain treatment
menstrual pain
Prior art date
Application number
CONC2019/0000672A
Other languages
English (en)
Inventor
Jost Maud
Glwadys Rausin
Original Assignee
Estetra Sprl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2016/076104 external-priority patent/WO2018065076A1/en
Application filed by Estetra Sprl filed Critical Estetra Sprl
Publication of CO2019000672A2 publication Critical patent/CO2019000672A2/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/566—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol having an oxo group in position 17, e.g. estrone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a un procedimiento para el tratamiento de la dismenorrea que implica la administración de un componente estrógeno que se selecciona preferentemente del grupo que consiste en estetrol y compuestos de tipo estetrol. Se ha descubierto sorprendentemente que los compuestos de tipo estetrol son capaces de mitigar la dismenorrea, bien cuando se usan solos o bien en combinación con componentes progestágenos, y esto en una medida que supera el efecto obtenido con otras composiciones y con un perfil de efectos secundarios favorable en comparación con procedimientos disponibles en la actualidad.
CONC2019/0000672A 2016-08-05 2019-01-24 Procedimiento de tratamiento de dismenorrea y dolor menstrual CO2019000672A2 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP16183025 2016-08-05
PCT/EP2016/076104 WO2018065076A1 (en) 2016-10-28 2016-10-28 Method for the management of dysmenorrhea and menstrual pain
PCT/EP2017/069908 WO2018024912A1 (en) 2016-08-05 2017-08-07 Method for the management of dysmenorrhea and menstrual pain

Publications (1)

Publication Number Publication Date
CO2019000672A2 true CO2019000672A2 (es) 2019-04-30

Family

ID=56609757

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2019/0000672A CO2019000672A2 (es) 2016-08-05 2019-01-24 Procedimiento de tratamiento de dismenorrea y dolor menstrual

Country Status (12)

Country Link
US (2) US20190167700A1 (es)
JP (2) JP6557298B2 (es)
KR (1) KR20220144885A (es)
AU (1) AU2022231672B2 (es)
BR (1) BR112019002203A2 (es)
CA (1) CA3178291A1 (es)
CO (1) CO2019000672A2 (es)
CR (1) CR20190112A (es)
MX (1) MX2022011436A (es)
PE (1) PE20190739A1 (es)
PH (1) PH12019500172A1 (es)
WO (1) WO2018024912A1 (es)

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JP2018533542A (ja) 2016-10-28 2018-11-15 エステトラ ソシエテ プリーヴ ア レスポンサビリテ リミテ 月経困難症および月経痛の管理のための方法
KR20220144885A (ko) 2016-08-05 2022-10-27 에스테트라, 소시에떼 아 레스폰서빌리떼 리미떼 월경통 및 생리통의 관리방법
GEP20227407B (en) 2018-02-07 2022-08-25 Estetra Sprl Contraceptive composition with reduced cardiovascular effects
JOP20200260A1 (ar) 2018-04-19 2019-10-19 Estetra Sprl مركبات واستخداماتها للتخفيف من الأعراض المصاحبة لانقطاع الطمث
TWI801561B (zh) 2018-04-19 2023-05-11 比利時商依思特拉私人有限責任公司 化合物及其用於緩解絕經相關症狀的用途
TW202203935A (zh) 2020-04-16 2022-02-01 比利時商埃斯特拉有限責任公司 具有降低之副作用之避孕組成物

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