CA2763768A1 - Methods of administration of thrombopoietin agonist compounds - Google Patents

Methods of administration of thrombopoietin agonist compounds Download PDF

Info

Publication number
CA2763768A1
CA2763768A1 CA2763768A CA2763768A CA2763768A1 CA 2763768 A1 CA2763768 A1 CA 2763768A1 CA 2763768 A CA2763768 A CA 2763768A CA 2763768 A CA2763768 A CA 2763768A CA 2763768 A1 CA2763768 A1 CA 2763768A1
Authority
CA
Canada
Prior art keywords
compound
dose
amount
pharmaceutically acceptable
days
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2763768A
Other languages
English (en)
French (fr)
Inventor
Connie L. Erickson-Miller
Julian Jenkins
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
GlaxoSmithKline LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43223061&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CA2763768(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by GlaxoSmithKline LLC filed Critical GlaxoSmithKline LLC
Publication of CA2763768A1 publication Critical patent/CA2763768A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • A61K31/41521,2-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. antipyrine, phenylbutazone, sulfinpyrazone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/04Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00Preparations for use in therapy

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA2763768A 2009-05-29 2010-05-27 Methods of administration of thrombopoietin agonist compounds Abandoned CA2763768A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18214809P 2009-05-29 2009-05-29
US61/182,148 2009-05-29
PCT/US2010/036294 WO2010138656A1 (en) 2009-05-29 2010-05-27 Methods of administration of thrombopoietin agonist compounds

Publications (1)

Publication Number Publication Date
CA2763768A1 true CA2763768A1 (en) 2010-12-02

Family

ID=43223061

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2763768A Abandoned CA2763768A1 (en) 2009-05-29 2010-05-27 Methods of administration of thrombopoietin agonist compounds

Country Status (20)

Country Link
US (1) US8609693B2 (enExample)
EP (2) EP3127427B1 (enExample)
JP (3) JP2012528184A (enExample)
KR (1) KR20120015355A (enExample)
CN (2) CN102458120A (enExample)
AU (1) AU2010254046C1 (enExample)
BR (1) BRPI1014548A2 (enExample)
CA (1) CA2763768A1 (enExample)
DK (1) DK3127427T3 (enExample)
EA (2) EA201690401A1 (enExample)
ES (2) ES2782898T3 (enExample)
HU (1) HUE049075T2 (enExample)
IL (1) IL216365A (enExample)
MX (1) MX2011012668A (enExample)
PL (2) PL2434894T3 (enExample)
PT (2) PT3127427T (enExample)
SG (1) SG176088A1 (enExample)
SI (1) SI3127427T1 (enExample)
WO (1) WO2010138656A1 (enExample)
ZA (1) ZA201108374B (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20120149749A1 (en) * 2008-10-16 2012-06-14 Michael Arning Method of treating thrombocytopenia
JP2012528184A (ja) 2009-05-29 2012-11-12 グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー トロンボポエチンアゴニスト化合物の投与の方法

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Also Published As

Publication number Publication date
ES2605593T3 (es) 2017-03-15
PT3127427T (pt) 2020-04-17
US8609693B2 (en) 2013-12-17
PT2434894T (pt) 2016-11-29
AU2010254046B2 (en) 2013-10-10
HUE049075T2 (hu) 2020-08-28
EA201690401A1 (ru) 2016-06-30
ES2782898T3 (es) 2020-09-16
EP2434894A1 (en) 2012-04-04
KR20120015355A (ko) 2012-02-21
JP2012528184A (ja) 2012-11-12
JP2017226668A (ja) 2017-12-28
EP3127427A1 (en) 2017-02-08
AU2010254046C1 (en) 2014-03-06
CN102458120A (zh) 2012-05-16
BRPI1014548A2 (pt) 2015-08-25
PL3127427T3 (pl) 2020-06-15
AU2010254046A1 (en) 2011-12-08
EP2434894B1 (en) 2016-08-31
US20120064036A1 (en) 2012-03-15
WO2010138656A1 (en) 2010-12-02
SI3127427T1 (sl) 2020-07-31
EP2434894A4 (en) 2013-02-20
EP3127427B1 (en) 2020-01-08
IL216365A (en) 2015-09-24
CN104173337A (zh) 2014-12-03
SG176088A1 (en) 2011-12-29
EA024557B1 (ru) 2016-09-30
DK3127427T3 (da) 2020-04-06
ZA201108374B (en) 2012-07-25
PL2434894T3 (pl) 2017-04-28
MX2011012668A (es) 2011-12-16
IL216365A0 (en) 2012-01-31
JP2016020360A (ja) 2016-02-04
EA201171462A1 (ru) 2012-05-30

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Legal Events

Date Code Title Description
EEER Examination request

Effective date: 20130606

FZDE Discontinued

Effective date: 20190528