CA2651596C - Percutaneous absorption preparations of antidementia drugs - Google Patents

Percutaneous absorption preparations of antidementia drugs Download PDF

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Publication number
CA2651596C
CA2651596C CA2651596A CA2651596A CA2651596C CA 2651596 C CA2651596 C CA 2651596C CA 2651596 A CA2651596 A CA 2651596A CA 2651596 A CA2651596 A CA 2651596A CA 2651596 C CA2651596 C CA 2651596C
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CA
Canada
Prior art keywords
drug
meth
acrylate
percutaneous absorption
absorption preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CA2651596A
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English (en)
French (fr)
Other versions
CA2651596A1 (en
Inventor
Takeshi Ito
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Teikoku Seiyaku Co Ltd
Original Assignee
Teikoku Seiyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teikoku Seiyaku Co Ltd filed Critical Teikoku Seiyaku Co Ltd
Publication of CA2651596A1 publication Critical patent/CA2651596A1/en
Application granted granted Critical
Publication of CA2651596C publication Critical patent/CA2651596C/en
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7084—Transdermal patches having a drug layer or reservoir, and one or more separate drug-free skin-adhesive layers, e.g. between drug reservoir and skin, or surrounding the drug reservoir; Liquid-filled reservoir patches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CA2651596A 2006-05-08 2006-12-25 Percutaneous absorption preparations of antidementia drugs Active CA2651596C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US79829606P 2006-05-08 2006-05-08
US60/798,296 2006-05-08
PCT/JP2006/325813 WO2007129427A1 (ja) 2006-05-08 2006-12-25 抗認知症薬物の経皮吸収製剤

Publications (2)

Publication Number Publication Date
CA2651596A1 CA2651596A1 (en) 2007-11-15
CA2651596C true CA2651596C (en) 2014-03-25

Family

ID=38667540

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2651596A Active CA2651596C (en) 2006-05-08 2006-12-25 Percutaneous absorption preparations of antidementia drugs

Country Status (16)

Country Link
US (2) US7858114B2 (https=)
EP (1) EP2016939B1 (https=)
JP (1) JP5122445B2 (https=)
KR (1) KR20090009951A (https=)
CN (1) CN101460156B (https=)
AU (1) AU2006343077B2 (https=)
BR (1) BRPI0621655A2 (https=)
CA (1) CA2651596C (https=)
ES (1) ES2466647T3 (https=)
IL (1) IL195174A0 (https=)
IN (1) IN266817B (https=)
MY (1) MY149152A (https=)
NO (1) NO20084614L (https=)
NZ (1) NZ572809A (https=)
RU (1) RU2428179C2 (https=)
WO (1) WO2007129427A1 (https=)

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EP2514414A4 (en) * 2009-12-16 2013-05-29 Goto Takeshi TRANSDERMAL ABSORBED PREPARATION OF ANTI-DENSITY ACTIVE SUBSTANCE
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WO2017002865A1 (ja) 2015-06-29 2017-01-05 積水化学工業株式会社 コアシェル構造体及び外用剤
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Also Published As

Publication number Publication date
IL195174A0 (en) 2009-08-03
US20110059141A1 (en) 2011-03-10
US7858114B2 (en) 2010-12-28
EP2016939A1 (en) 2009-01-21
JP5122445B2 (ja) 2013-01-16
EP2016939A4 (en) 2013-01-09
US20070259028A1 (en) 2007-11-08
CA2651596A1 (en) 2007-11-15
AU2006343077B2 (en) 2012-11-08
BRPI0621655A2 (pt) 2011-12-20
CN101460156B (zh) 2011-06-08
IN266817B (https=) 2015-06-03
MY149152A (en) 2013-07-15
RU2428179C2 (ru) 2011-09-10
KR20090009951A (ko) 2009-01-23
RU2008148131A (ru) 2010-06-20
WO2007129427A1 (ja) 2007-11-15
EP2016939B1 (en) 2014-03-19
AU2006343077A1 (en) 2007-11-15
ES2466647T3 (es) 2014-06-10
NO20084614L (no) 2009-02-06
CN101460156A (zh) 2009-06-17
JPWO2007129427A1 (ja) 2009-09-17
HK1130175A1 (en) 2009-12-24
NZ572809A (en) 2011-02-25

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