CA2632286C - Use of (r)-3-[1-(2,6-dichloro-3-fluror-phenyl)-ethoxyl]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)-pyridin-2-ylamine for treatment of cancer - Google Patents
Use of (r)-3-[1-(2,6-dichloro-3-fluror-phenyl)-ethoxyl]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)-pyridin-2-ylamine for treatment of cancer Download PDFInfo
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
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| US74276605P | 2005-12-05 | 2005-12-05 | |
| US60/742,766 | 2005-12-05 | ||
| US86463706P | 2006-11-07 | 2006-11-07 | |
| US60/864,637 | 2006-11-07 | ||
| PCT/IB2006/003397 WO2007066187A2 (en) | 2005-12-05 | 2006-11-23 | Method of treating abnormal cell growth |
Publications (2)
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| CA2632286A1 CA2632286A1 (en) | 2007-06-14 |
| CA2632286C true CA2632286C (en) | 2011-11-15 |
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| JP (1) | JP4619346B2 (enExample) |
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| CY (1) | CY1110931T1 (enExample) |
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| PT (1) | PT1959955E (enExample) |
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| SI (1) | SI1959955T1 (enExample) |
| TW (1) | TWI321050B (enExample) |
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| PL2450437T3 (pl) | 2006-04-14 | 2017-12-29 | Cell Signaling Technology Inc | Defekty genu i zmutowana kinaza ALK w ludzkich guzach litych |
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| SI1959955T1 (sl) | 2011-02-28 |
| NZ568654A (en) | 2012-02-24 |
| CY1110931T1 (el) | 2015-06-10 |
| US7825137B2 (en) | 2010-11-02 |
| CA2632286A1 (en) | 2007-06-14 |
| AR056832A1 (es) | 2007-10-24 |
| IL191471A (en) | 2013-03-24 |
| PL1959955T3 (pl) | 2011-04-29 |
| AU2006323027A1 (en) | 2007-06-14 |
| US20080300273A1 (en) | 2008-12-04 |
| AU2006323027B2 (en) | 2012-08-02 |
| TW200727899A (en) | 2007-08-01 |
| HK1126121A1 (en) | 2009-08-28 |
| ATE488237T1 (de) | 2010-12-15 |
| DE602006018354D1 (de) | 2010-12-30 |
| BRPI0619424B1 (pt) | 2022-02-08 |
| WO2007066187A2 (en) | 2007-06-14 |
| RU2008122471A (ru) | 2009-12-10 |
| KR20080072965A (ko) | 2008-08-07 |
| EP1959955A2 (en) | 2008-08-27 |
| WO2007066187A3 (en) | 2008-01-17 |
| DK1959955T3 (da) | 2011-02-07 |
| JP2007153894A (ja) | 2007-06-21 |
| IL191471A0 (en) | 2009-08-03 |
| KR101026676B1 (ko) | 2011-04-04 |
| BRPI0619424A2 (pt) | 2011-10-04 |
| JP4619346B2 (ja) | 2011-01-26 |
| PT1959955E (pt) | 2011-01-04 |
| EP1959955B1 (en) | 2010-11-17 |
| TWI321050B (en) | 2010-03-01 |
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