CA2379875A1 - New effectors of dipeptidyl peptidase iv for topical use - Google Patents
New effectors of dipeptidyl peptidase iv for topical use Download PDFInfo
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- CA2379875A1 CA2379875A1 CA002379875A CA2379875A CA2379875A1 CA 2379875 A1 CA2379875 A1 CA 2379875A1 CA 002379875 A CA002379875 A CA 002379875A CA 2379875 A CA2379875 A CA 2379875A CA 2379875 A1 CA2379875 A1 CA 2379875A1
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- A—HUMAN NECESSITIES
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- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06104—Dipeptides with the first amino acid being acidic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
- C07K5/0806—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
-
- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08G—MACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
- C08G65/00—Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule
- C08G65/02—Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule from cyclic ethers by opening of the heterocyclic ring
- C08G65/32—Polymers modified by chemical after-treatment
- C08G65/329—Polymers modified by chemical after-treatment with organic compounds
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- A—HUMAN NECESSITIES
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| Application Number | Priority Date | Filing Date | Title |
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| DE19940130.6 | 1999-08-24 | ||
| DE19940130A DE19940130A1 (de) | 1999-08-24 | 1999-08-24 | Neue Effektoren der Dipeptidyl Peptidase IV zur topischen Anwendung |
| PCT/EP2000/008118 WO2001014318A2 (de) | 1999-08-24 | 2000-08-20 | Neue effektoren der dipeptidyl peptidase iv zur topischen anwendung |
Publications (1)
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| CA2379875A1 true CA2379875A1 (en) | 2001-03-01 |
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| CA002379875A Abandoned CA2379875A1 (en) | 1999-08-24 | 2000-08-20 | New effectors of dipeptidyl peptidase iv for topical use |
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| EP1228061A4 (en) | 1999-11-12 | 2004-12-15 | Guilford Pharm Inc | DIPEPTIDYL PEPTIDASE IV INHIBITORS; METHODS OF MANUFACTURE AND USE OF SAID INHIBITORS |
| WO2001062266A2 (en) | 2000-02-25 | 2001-08-30 | Novo Nordisk A/S | Use of dpp-iv inhibitors for the treatment of diabetes |
| US7064145B2 (en) * | 2000-02-25 | 2006-06-20 | Novo Nordisk A/S | Inhibition of beta cell degeneration |
| DE60042585D1 (de) | 2000-02-29 | 2009-09-03 | Univ Firenze | 3-Aza-6,8-dioxabicycloÄ3.2.1Üoctane und Analoga sowie diese enthaltende kombinatorische Bibliotheken |
| JP2003528135A (ja) * | 2000-03-31 | 2003-09-24 | プロバイオドラッグ アーゲー | 糖尿病のランゲルハンス島シグナリングの改善方法及びその防止方法 |
| US6605589B1 (en) | 2000-03-31 | 2003-08-12 | Parker Hughes Institute | Cathepsin inhibitors in cancer treatment |
| US6573096B1 (en) | 2000-04-01 | 2003-06-03 | The Research Foundation At State University Of New York | Compositions and methods for inhibition of cancer invasion and angiogenesis |
| DE10025464A1 (de) | 2000-05-23 | 2001-12-06 | Inst Medizintechnologie Magdeb | Kombinierte Verwendung von Enzyminhibitoren zur Therapie von Autoimmunerkrankungen, bei Transplantationen und Tumorerkrankungen sowie Kombinationen von Enzyminhibitoren umfassende pharmazeutische Zubereitungen |
| US6841685B2 (en) | 2000-06-07 | 2005-01-11 | State Of Oregon Acting By And Through The State Board Of Higher Education On Behalf Of Oregon State University | Methods for making bis-heterocyclic alkaloids |
| GB0014969D0 (en) | 2000-06-19 | 2000-08-09 | Smithkline Beecham Plc | Novel method of treatment |
| EP1313470A4 (en) | 2000-08-17 | 2005-02-16 | Gliatech Inc | NEW ALICYCLIC IMIDAZOLE AS H 3 ACTIVE SUBSTANCES |
| US7785810B2 (en) | 2000-09-09 | 2010-08-31 | The Research Foundation Of State University Of New York | Method and compositions for isolating metastatic cancer cells, and use in measuring metastatic potential of a cancer thereof |
| AU2002328946A1 (en) | 2001-08-13 | 2003-03-03 | Probiodrug Ag | Irreversible cysteine protease inhibitors of legumain |
| JP2005523288A (ja) | 2002-02-19 | 2005-08-04 | ファルマシア・アンド・アップジョン・カンパニー・エルエルシー | 疾病治療用の縮合した二環式−ｎ−架橋−複素環式芳香族カルボキサミド |
| CA2521907A1 (en) | 2003-04-10 | 2004-10-21 | Pfizer Inc. | Bicyclic compounds as nr2b receptor antagonists |
-
1999
- 1999-08-24 DE DE19940130A patent/DE19940130A1/de not_active Withdrawn
-
2000
- 2000-08-20 BR BR0013577-1A patent/BR0013577A/pt not_active Application Discontinuation
- 2000-08-20 CN CN00811936A patent/CN1370181A/zh active Pending
- 2000-08-20 DE DE50014187T patent/DE50014187D1/de not_active Expired - Fee Related
- 2000-08-20 AT AT00953186T patent/ATE357455T1/de not_active IP Right Cessation
- 2000-08-20 AU AU65721/00A patent/AU769404B2/en not_active Ceased
- 2000-08-20 NZ NZ528770A patent/NZ528770A/en unknown
- 2000-08-20 JP JP2001518409A patent/JP2003519099A/ja not_active Withdrawn
- 2000-08-20 PT PT00953186T patent/PT1206485E/pt unknown
- 2000-08-20 MX MXPA02001800A patent/MXPA02001800A/es unknown
- 2000-08-20 ES ES00953186T patent/ES2282130T3/es not_active Expired - Lifetime
- 2000-08-20 CA CA002379875A patent/CA2379875A1/en not_active Abandoned
- 2000-08-20 EP EP00953186A patent/EP1206485B1/de not_active Expired - Lifetime
- 2000-08-20 WO PCT/EP2000/008118 patent/WO2001014318A2/de not_active Ceased
- 2000-08-20 EP EP07104464A patent/EP1792910A2/de not_active Withdrawn
- 2000-08-20 IL IL14817000A patent/IL148170A0/xx unknown
- 2000-08-20 KR KR1020027002338A patent/KR20020040787A/ko not_active Withdrawn
-
2002
- 2002-01-29 ZA ZA200200794A patent/ZA200200794B/en unknown
- 2002-02-22 NO NO20020858A patent/NO20020858L/no not_active Application Discontinuation
- 2002-02-22 US US10/082,001 patent/US6949515B2/en not_active Expired - Fee Related
-
2005
- 2005-03-01 US US11/069,926 patent/US7335645B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200200794B (en) | 2003-03-26 |
| US20030092630A2 (en) | 2003-05-15 |
| PT1206485E (pt) | 2007-05-31 |
| EP1206485A2 (de) | 2002-05-22 |
| WO2001014318A3 (de) | 2001-11-01 |
| JP2003519099A (ja) | 2003-06-17 |
| ATE357455T1 (de) | 2007-04-15 |
| NO20020858D0 (no) | 2002-02-22 |
| US7335645B2 (en) | 2008-02-26 |
| BR0013577A (pt) | 2002-04-30 |
| KR20020040787A (ko) | 2002-05-30 |
| US6949515B2 (en) | 2005-09-27 |
| WO2001014318A2 (de) | 2001-03-01 |
| EP1206485B1 (de) | 2007-03-21 |
| EP1792910A2 (de) | 2007-06-06 |
| IL148170A0 (en) | 2002-09-12 |
| ES2282130T3 (es) | 2007-10-16 |
| US20020165164A1 (en) | 2002-11-07 |
| NZ528770A (en) | 2005-02-25 |
| MXPA02001800A (es) | 2003-09-25 |
| DE50014187D1 (de) | 2007-05-03 |
| CN1370181A (zh) | 2002-09-18 |
| DE19940130A1 (de) | 2001-03-01 |
| AU769404B2 (en) | 2004-01-29 |
| AU6572100A (en) | 2001-03-19 |
| NO20020858L (no) | 2002-02-22 |
| US20050209159A1 (en) | 2005-09-22 |
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| Date | Code | Title | Description |
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| FZDE | Discontinued |