CA2181351C - Process and intermediates for preparing naphthyridonecarboxylic acid salts - Google Patents

Process and intermediates for preparing naphthyridonecarboxylic acid salts

Info

Publication number
CA2181351C
CA2181351C CA002181351A CA2181351A CA2181351C CA 2181351 C CA2181351 C CA 2181351C CA 002181351 A CA002181351 A CA 002181351A CA 2181351 A CA2181351 A CA 2181351A CA 2181351 C CA2181351 C CA 2181351C
Authority
CA
Canada
Prior art keywords
formula
compound
acid
alkyl
treating
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CA002181351A
Other languages
English (en)
French (fr)
Other versions
CA2181351A1 (en
Inventor
Tamim F. Braish
Darrell E. Fox
Timothy Norris
Peter R. Rose
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of CA2181351A1 publication Critical patent/CA2181351A1/en
Application granted granted Critical
Publication of CA2181351C publication Critical patent/CA2181351C/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA002181351A 1994-01-18 1994-12-12 Process and intermediates for preparing naphthyridonecarboxylic acid salts Expired - Fee Related CA2181351C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18194294A 1994-01-18 1994-01-18
US08/181,942 1994-01-18
PCT/IB1994/000410 WO1995019361A1 (en) 1994-01-18 1994-12-12 Process and intermediates for preparing naphthyridonecarboxylic acid salts

Publications (2)

Publication Number Publication Date
CA2181351A1 CA2181351A1 (en) 1995-07-20
CA2181351C true CA2181351C (en) 1999-09-28

Family

ID=22666458

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002181351A Expired - Fee Related CA2181351C (en) 1994-01-18 1994-12-12 Process and intermediates for preparing naphthyridonecarboxylic acid salts

Country Status (19)

Country Link
EP (1) EP0740667A1 (ja)
JP (1) JP2891543B2 (ja)
KR (1) KR100221386B1 (ja)
CN (1) CN1141634A (ja)
AU (1) AU694149B2 (ja)
BR (1) BR9408490A (ja)
CA (1) CA2181351C (ja)
CZ (1) CZ286896B6 (ja)
FI (1) FI962880A (ja)
HU (1) HUT74883A (ja)
IL (1) IL112323A (ja)
MY (1) MY130510A (ja)
NO (1) NO305838B1 (ja)
NZ (1) NZ276478A (ja)
PL (1) PL179996B1 (ja)
RU (1) RU2147303C1 (ja)
TW (1) TW414791B (ja)
WO (1) WO1995019361A1 (ja)
ZA (1) ZA95340B (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK280535B6 (sk) * 1995-06-06 2000-03-13 Pfizer Inc. Kryštalická forma bezvodej soli kyseliny 7-([1a,5a
ES2095809B1 (es) * 1995-07-27 1997-12-16 Sint Quimica Sa Procedimiento para la preparacion de acidos naftiridin carboxilicos y sus sales.
GB9524466D0 (en) * 1995-11-30 1996-01-31 Pfizer Ltd Process
GB9614422D0 (en) * 1996-07-09 1996-09-04 Pfizer Ltd Novel process
JPH1087617A (ja) * 1996-07-09 1998-04-07 Pfizer Inc キノリン系抗生物質の合成に有用な中間体の製法
HN1998000106A (es) 1997-08-01 1999-01-08 Pfizer Prod Inc Composiciones parenterales de alatroflaxacino
HN1999000141A (es) * 1998-09-03 2000-06-19 Pfizer Prod Inc Procedimiento para preparar sales de trovafloxacina de adicion de acidos.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5164402A (en) * 1989-08-16 1992-11-17 Pfizer Inc Azabicyclo quinolone and naphthyridinone carboxylic acids

Also Published As

Publication number Publication date
CZ286896B6 (en) 2000-07-12
PL179996B1 (en) 2000-11-30
NO962990D0 (no) 1996-07-17
PL317043A1 (en) 1997-03-03
MY130510A (en) 2007-06-29
KR100221386B1 (ko) 1999-09-15
JPH09501182A (ja) 1997-02-04
WO1995019361A1 (en) 1995-07-20
HUT74883A (en) 1997-02-28
BR9408490A (pt) 1997-08-26
EP0740667A1 (en) 1996-11-06
FI962880A0 (fi) 1996-07-17
HU9601957D0 (en) 1996-09-30
NZ276478A (en) 1998-05-27
TW414791B (en) 2000-12-11
CN1141634A (zh) 1997-01-29
AU1075495A (en) 1995-08-01
JP2891543B2 (ja) 1999-05-17
IL112323A (en) 2001-03-19
CA2181351A1 (en) 1995-07-20
CZ211196A3 (en) 1997-01-15
AU694149B2 (en) 1998-07-16
NO305838B1 (no) 1999-08-02
IL112323A0 (en) 1995-03-30
RU2147303C1 (ru) 2000-04-10
NO962990L (no) 1996-07-17
ZA95340B (en) 1996-07-17
FI962880A (fi) 1996-07-17

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Legal Events

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