CA1105037A - N-(4-pyrazolidinyl) benzamides - Google Patents

N-(4-pyrazolidinyl) benzamides

Info

Publication number
CA1105037A
CA1105037A CA309,651A CA309651A CA1105037A CA 1105037 A CA1105037 A CA 1105037A CA 309651 A CA309651 A CA 309651A CA 1105037 A CA1105037 A CA 1105037A
Authority
CA
Canada
Prior art keywords
amino
chloro
methoxy
pyrazolidinyl
process according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA309,651A
Other languages
English (en)
French (fr)
Inventor
Carl D. Lunsford
Albert D. Cale, Jr.
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AH Robins Co Inc
Original Assignee
AH Robins Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AH Robins Co Inc filed Critical AH Robins Co Inc
Priority to CA362,371A priority Critical patent/CA1109880A/en
Application granted granted Critical
Publication of CA1105037A publication Critical patent/CA1105037A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/04—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Otolaryngology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA309,651A 1977-08-19 1978-08-18 N-(4-pyrazolidinyl) benzamides Expired CA1105037A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CA362,371A CA1109880A (en) 1977-08-19 1980-10-14 N-(4-pyrazolidinyl) benzamides

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US82603177A 1977-08-19 1977-08-19
US826,031 1977-08-19
US90036978A 1978-04-26 1978-04-26
US900,369 1978-04-26
US93012578A 1978-08-01 1978-08-01
US930,125 1992-08-14

Publications (1)

Publication Number Publication Date
CA1105037A true CA1105037A (en) 1981-07-14

Family

ID=27420183

Family Applications (1)

Application Number Title Priority Date Filing Date
CA309,651A Expired CA1105037A (en) 1977-08-19 1978-08-18 N-(4-pyrazolidinyl) benzamides

Country Status (21)

Country Link
JP (1) JPS5441873A (sv)
AU (1) AU521421B2 (sv)
BR (1) BR7805288A (sv)
CA (1) CA1105037A (sv)
CH (2) CH639374A5 (sv)
DE (1) DE2836062A1 (sv)
DK (1) DK152361C (sv)
ES (1) ES472686A1 (sv)
FI (1) FI68044C (sv)
FR (1) FR2400511A1 (sv)
GB (2) GB2017678B (sv)
HK (1) HK42282A (sv)
IE (1) IE47430B1 (sv)
MX (1) MX5469E (sv)
NL (1) NL7808596A (sv)
NO (1) NO149107C (sv)
NZ (1) NZ188189A (sv)
PH (1) PH13331A (sv)
PT (1) PT68442A (sv)
SE (2) SE444434B (sv)
YU (1) YU41116B (sv)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4309552A (en) * 1980-08-07 1982-01-05 A. H. Robins Company, Inc. Synthesis of 4-nitro-1,2-hydrocarbyl pyrazolidines and process for preparation thereof
US5126343A (en) * 1989-09-11 1992-06-30 G. D. Searle & Co. N-azabicyclo [3.3.0]octane amides of aromatic acids
JP3065506B2 (ja) * 1995-04-03 2000-07-17 株式会社資生堂 ピラゾリジン誘導体及びラジカルスカベンジャー、脳梗塞抑制剤、脳浮腫抑制剤
AR086587A1 (es) 2011-05-31 2014-01-08 Syngenta Participations Ag Compuestos insecticidas

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3966957A (en) * 1972-04-03 1976-06-29 A. H. Robins Company, Incorporated Method for controlling emesis with N-(1-substituted-3-pyrrolidinyl)benzamides and thiobenzamides

Also Published As

Publication number Publication date
DK366978A (da) 1979-02-20
FR2400511A1 (fr) 1979-03-16
GB2017678B (en) 1982-03-10
BR7805288A (pt) 1979-04-10
YU198678A (en) 1983-01-21
SE444434B (sv) 1986-04-14
GB2003153B (en) 1982-02-24
NO149107B (no) 1983-11-07
NO782812L (no) 1979-02-20
DK152361C (da) 1988-07-25
YU41116B (en) 1986-12-31
ES472686A1 (es) 1979-03-16
FR2400511B1 (sv) 1981-09-04
NO149107C (no) 1984-02-22
FI782507A (fi) 1979-02-20
CH645356A5 (fr) 1984-09-28
NL7808596A (nl) 1979-02-21
PT68442A (en) 1978-09-01
FI68044C (fi) 1985-07-10
GB2017678A (en) 1979-10-10
FI68044B (fi) 1985-03-29
SE8303564D0 (sv) 1983-06-21
AU521421B2 (en) 1982-04-01
IE47430B1 (en) 1984-03-21
HK42282A (en) 1982-10-08
DE2836062A1 (de) 1979-03-01
JPS6315273B2 (sv) 1988-04-04
JPS5441873A (en) 1979-04-03
GB2003153A (en) 1979-03-07
SE8303564L (sv) 1983-06-21
SE7808694L (sv) 1979-02-20
PH13331A (en) 1980-03-13
SE451723B (sv) 1987-10-26
IE781682L (en) 1979-02-19
NZ188189A (en) 1984-07-06
DK152361B (da) 1988-02-22
CH639374A5 (fr) 1983-11-15
AU3906178A (en) 1980-02-21
MX5469E (es) 1983-08-16

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Legal Events

Date Code Title Description
MKEX Expiry