BRPI0909211B8 - formulação oral em forma de comprimido de compostos de tetraciclina - Google Patents

formulação oral em forma de comprimido de compostos de tetraciclina

Info

Publication number
BRPI0909211B8
BRPI0909211B8 BRPI0909211A BRPI0909211A BRPI0909211B8 BR PI0909211 B8 BRPI0909211 B8 BR PI0909211B8 BR PI0909211 A BRPI0909211 A BR PI0909211A BR PI0909211 A BRPI0909211 A BR PI0909211A BR PI0909211 B8 BRPI0909211 B8 BR PI0909211B8
Authority
BR
Brazil
Prior art keywords
tetracycline compounds
oral tablet
form formulation
oral
formulations
Prior art date
Application number
BRPI0909211A
Other languages
English (en)
Inventor
Johnston Sean
Original Assignee
Paratek Pharm Innc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41114256&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0909211(B8) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Paratek Pharm Innc filed Critical Paratek Pharm Innc
Priority to BR122020011180A priority Critical patent/BR122020011180B8/pt
Publication of BRPI0909211A2 publication Critical patent/BRPI0909211A2/pt
Publication of BRPI0909211B1 publication Critical patent/BRPI0909211B1/pt
Publication of BRPI0909211B8 publication Critical patent/BRPI0909211B8/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/65—Tetracyclines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

formulações orais e injetáveis de compostos de tetraciclina são descritas formulações injetáveis e orais de um composto de tetraciclina. em uma modalidade, a invenção se refere a uma formulação oral de um composto de 9-aminometil tetraciclina, ou de um sal seu, em forma de comprimido ou cápsula. as formulações po-dem ser usadas, por exemplo, para tratar infecções.
BRPI0909211A 2008-03-28 2009-03-30 formulação oral em forma de comprimido de compostos de tetraciclina BRPI0909211B8 (pt)

Priority Applications (1)

Application Number Priority Date Filing Date Title
BR122020011180A BR122020011180B8 (pt) 2008-03-28 2009-03-30 formulações injetáveis de compostos de tetraciclina

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4039808P 2008-03-28 2008-03-28
US61/040,398 2008-03-28
PCT/US2009/001973 WO2009120389A1 (en) 2008-03-28 2009-03-30 Oral and injectable formulations of tetracycline compounds

Publications (3)

Publication Number Publication Date
BRPI0909211A2 BRPI0909211A2 (pt) 2016-11-29
BRPI0909211B1 BRPI0909211B1 (pt) 2020-08-25
BRPI0909211B8 true BRPI0909211B8 (pt) 2021-05-25

Family

ID=41114256

Family Applications (2)

Application Number Title Priority Date Filing Date
BRPI0909211A BRPI0909211B8 (pt) 2008-03-28 2009-03-30 formulação oral em forma de comprimido de compostos de tetraciclina
BR122020011180A BR122020011180B8 (pt) 2008-03-28 2009-03-30 formulações injetáveis de compostos de tetraciclina

Family Applications After (1)

Application Number Title Priority Date Filing Date
BR122020011180A BR122020011180B8 (pt) 2008-03-28 2009-03-30 formulações injetáveis de compostos de tetraciclina

Country Status (31)

Country Link
US (2) US9314475B2 (pt)
EP (3) EP3348258B1 (pt)
JP (7) JP2011515473A (pt)
KR (3) KR101893740B1 (pt)
CN (1) CN102046177B (pt)
AU (1) AU2009229174A1 (pt)
BR (2) BRPI0909211B8 (pt)
CA (2) CA2719751C (pt)
CL (1) CL2010000281A1 (pt)
CO (1) CO6300935A2 (pt)
CY (2) CY1120240T1 (pt)
DK (2) DK2271348T3 (pt)
EC (1) ECSP10010576A (pt)
ES (2) ES2674708T3 (pt)
HK (1) HK1257928A1 (pt)
HR (2) HRP20180836T1 (pt)
HU (2) HUE052201T2 (pt)
IL (1) IL208440A0 (pt)
LT (2) LT3348258T (pt)
MA (1) MA32275B1 (pt)
MX (1) MX2010010585A (pt)
NO (1) NO2271348T3 (pt)
NZ (1) NZ588428A (pt)
PL (2) PL2271348T3 (pt)
PT (2) PT2271348T (pt)
RU (1) RU2010144130A (pt)
SI (2) SI2271348T1 (pt)
TR (1) TR201806893T4 (pt)
UA (2) UA122762C2 (pt)
WO (1) WO2009120389A1 (pt)
ZA (1) ZA201007013B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102015602A (zh) 2008-03-05 2011-04-13 帕拉特克药品公司 米诺环素化合物及其使用方法
TW202216656A (zh) 2008-05-23 2022-05-01 美商Ｐｒｔｋ Ｓｐｖ２公司 四環素化合物之甲苯磺酸鹽及同素異形體
ES2613738T3 (es) 2010-05-12 2017-05-25 Rempex Pharmaceuticals, Inc. Composiciones de tetraciclina
MX2018013271A (es) * 2016-05-02 2019-03-28 Paratek Pharm Innc Compuestos 9-aminometil minociclina y metodos para utilizarlos en el tratamiento de infeccion de vias urinarias (ivu).
US10166912B2 (en) 2016-08-19 2019-01-01 Sl Corporation Automotive LED driving apparatus
CA3042514A1 (en) 2016-11-01 2018-05-11 Paratek Pharmaceuticals, Inc. 9-aminomethyl minocycline compounds and use thereof in treating community-acquired bacterial pneumonia (cabp)
MX2021002503A (es) * 2018-09-04 2021-06-15 Paratek Pharm Innc Métodos de tratamiento de infecciones micobacterianas usando compuestos de tetraciclina.
PT117254B (pt) 2021-05-26 2024-04-18 Hovione Farm S A Método de síntese de compostos 9-aminometil tetraciclinas

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Also Published As

Publication number Publication date
DK3348258T3 (da) 2020-12-07
WO2009120389A8 (en) 2009-12-30
ECSP10010576A (es) 2010-12-30
CA2719751C (en) 2018-01-02
MX2010010585A (es) 2010-11-09
EP3789030A1 (en) 2021-03-10
BR122020011180B1 (pt) 2021-03-23
JP2021167355A (ja) 2021-10-21
EP2271348B1 (en) 2018-03-28
JP2011515473A (ja) 2011-05-19
JP2023144043A (ja) 2023-10-06
JP2016145260A (ja) 2016-08-12
CY1120240T1 (el) 2019-07-10
BRPI0909211B1 (pt) 2020-08-25
DK2271348T3 (en) 2018-06-14
LT3348258T (lt) 2020-12-10
HRP20201883T1 (hr) 2021-01-22
US20100056638A1 (en) 2010-03-04
TR201806893T4 (tr) 2018-06-21
KR101893740B1 (ko) 2018-08-30
LT2271348T (lt) 2018-06-25
CA2984301A1 (en) 2009-10-01
CN102046177B (zh) 2012-12-19
IL208440A0 (en) 2010-12-30
PT2271348T (pt) 2018-04-16
EP2271348A1 (en) 2011-01-12
CL2010000281A1 (es) 2012-03-30
PL3348258T3 (pl) 2021-03-08
HRP20180836T1 (hr) 2018-07-27
BR122020011180B8 (pt) 2021-07-27
AU2009229174A1 (en) 2009-10-01
HK1257928A1 (zh) 2019-11-01
UA109627C2 (uk) 2015-09-25
PL2271348T3 (pl) 2018-08-31
KR20160105532A (ko) 2016-09-06
JP6412521B2 (ja) 2018-10-24
JP5940119B2 (ja) 2016-06-29
MA32275B1 (fr) 2011-05-02
WO2009120389A1 (en) 2009-10-01
UA122762C2 (uk) 2021-01-06
HUE038257T2 (hu) 2018-10-29
EP3348258A1 (en) 2018-07-18
US20160279151A1 (en) 2016-09-29
ES2674708T3 (es) 2018-07-03
CY1123382T1 (el) 2021-12-31
JP2019196408A (ja) 2019-11-14
BRPI0909211A2 (pt) 2016-11-29
NZ588428A (en) 2012-08-31
KR101746228B1 (ko) 2017-06-12
PT3348258T (pt) 2020-11-25
JP6577645B2 (ja) 2019-09-18
EP2271348A4 (en) 2011-05-25
CA2719751A1 (en) 2009-10-01
SI3348258T1 (sl) 2020-12-31
JP2014221820A (ja) 2014-11-27
US9314475B2 (en) 2016-04-19
EP3348258B1 (en) 2020-09-09
KR20180026799A (ko) 2018-03-13
CN102046177A (zh) 2011-05-04
JP2018203778A (ja) 2018-12-27
CO6300935A2 (es) 2011-07-21
NO2271348T3 (pt) 2018-08-25
ES2836448T3 (es) 2021-06-25
HUE052201T2 (hu) 2021-04-28
KR20110008057A (ko) 2011-01-25
KR101835574B1 (ko) 2018-03-08
ZA201007013B (en) 2013-11-27
CA2984301C (en) 2020-10-27
RU2010144130A (ru) 2012-05-10
SI2271348T1 (en) 2018-08-31

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