BRPI0710095A2 - inibidores de renina para o tratamento de hipertensão - Google Patents
inibidores de renina para o tratamento de hipertensão Download PDFInfo
- Publication number
- BRPI0710095A2 BRPI0710095A2 BRPI0710095-7A BRPI0710095A BRPI0710095A2 BR PI0710095 A2 BRPI0710095 A2 BR PI0710095A2 BR PI0710095 A BRPI0710095 A BR PI0710095A BR PI0710095 A2 BRPI0710095 A2 BR PI0710095A2
- Authority
- BR
- Brazil
- Prior art keywords
- hypertension
- cessation
- renin inhibitor
- refers
- blood pressure
- Prior art date
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- 125000000623 heterocyclic group Chemical group 0.000 description 1
- 125000003707 hexyloxy group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])O* 0.000 description 1
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- 235000013980 iron oxide Nutrition 0.000 description 1
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- 239000000813 peptide hormone Substances 0.000 description 1
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- NBIIXXVUZAFLBC-UHFFFAOYSA-K phosphate Chemical compound [O-]P([O-])([O-])=O NBIIXXVUZAFLBC-UHFFFAOYSA-K 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
- A61K31/175—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine having the group, >N—C(O)—N=N— or, e.g. carbonohydrazides, carbazones, semicarbazides, semicarbazones; Thioanalogues thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Heart & Thoracic Surgery (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US78884206P | 2006-04-03 | 2006-04-03 | |
| US60/788,842 | 2006-04-03 | ||
| PCT/US2007/065564 WO2007118023A1 (en) | 2006-04-03 | 2007-03-30 | Renin inhibitors for the treatment of hypertension |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0710095A2 true BRPI0710095A2 (pt) | 2011-08-02 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0710095-7A BRPI0710095A2 (pt) | 2006-04-03 | 2007-03-30 | inibidores de renina para o tratamento de hipertensão |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20090062395A1 (enExample) |
| EP (1) | EP2004167A1 (enExample) |
| JP (1) | JP2009532494A (enExample) |
| KR (1) | KR20080108515A (enExample) |
| CN (1) | CN101415413A (enExample) |
| AU (1) | AU2007234917B2 (enExample) |
| BR (1) | BRPI0710095A2 (enExample) |
| CA (1) | CA2645260A1 (enExample) |
| CL (1) | CL2007000912A1 (enExample) |
| IL (1) | IL193905A0 (enExample) |
| MA (1) | MA30387B1 (enExample) |
| MX (1) | MX2008012729A (enExample) |
| NO (1) | NO20084625L (enExample) |
| NZ (1) | NZ571251A (enExample) |
| RU (1) | RU2008143055A (enExample) |
| SG (1) | SG170830A1 (enExample) |
| TN (1) | TNSN08383A1 (enExample) |
| TW (1) | TW200806283A (enExample) |
| WO (1) | WO2007118023A1 (enExample) |
| ZA (1) | ZA200807615B (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009087116A1 (en) * | 2008-01-11 | 2009-07-16 | Novartis Ag | Use of spp100 for the treatment of acute mi |
| CN102212012A (zh) * | 2010-04-12 | 2011-10-12 | 上海源力生物技术有限公司 | 一种合成阿利克伦的中间体及其制备方法 |
| EP2768971A1 (en) | 2011-10-20 | 2014-08-27 | Institut National de la Santé et de la Recherche Médicale (INSERM) | Methods for the detection and the treatment of cardiac remodeling |
| CA3137138A1 (en) * | 2019-04-18 | 2020-10-22 | EyePoint Pharmaceuticals, Inc. | Methods of treating hypertension with activators of tie-2 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY119161A (en) * | 1994-04-18 | 2005-04-30 | Novartis Ag | Delta-amino-gamma-hydroxy-omega-aryl-alkanoic acid amides with enzyme especially renin inhibiting activities |
| US5659065A (en) * | 1994-04-18 | 1997-08-19 | Novartis Corporation | Alpha-aminoalkanoic acids and reduction products |
| US5606078A (en) * | 1994-04-18 | 1997-02-25 | Ciba-Geigy Corporation | 3,5-Disubstituted tetrahydrofuran-2-ones |
| AU2003250858A1 (en) * | 2002-06-28 | 2004-01-19 | Novartis Ag | Use of organic compounds |
| US20040266743A1 (en) * | 2003-05-09 | 2004-12-30 | Pharmacia Corporation | Combination of an aldosterone receptor antagonist and a renin inhibitor |
| WO2005037317A2 (en) * | 2003-10-17 | 2005-04-28 | Cornell Research Foundation, Inc. | Mast cell-derived renin |
| PE20110121A1 (es) * | 2004-03-17 | 2011-02-28 | Novartis Ag | Composiciones farmaceuticas de aliskiren |
| EP1796725B1 (en) * | 2004-09-27 | 2008-07-23 | Pantarhei Bioscience B.V. | Treatment or prevention of unscheluded bleeding in women on progestogen containing medication |
-
2007
- 2007-03-30 CA CA002645260A patent/CA2645260A1/en not_active Abandoned
- 2007-03-30 AU AU2007234917A patent/AU2007234917B2/en not_active Ceased
- 2007-03-30 JP JP2009504386A patent/JP2009532494A/ja active Pending
- 2007-03-30 BR BRPI0710095-7A patent/BRPI0710095A2/pt not_active IP Right Cessation
- 2007-03-30 WO PCT/US2007/065564 patent/WO2007118023A1/en not_active Ceased
- 2007-03-30 SG SG201102387-6A patent/SG170830A1/en unknown
- 2007-03-30 KR KR1020087024219A patent/KR20080108515A/ko not_active Withdrawn
- 2007-03-30 EP EP07759755A patent/EP2004167A1/en not_active Withdrawn
- 2007-03-30 RU RU2008143055/14A patent/RU2008143055A/ru unknown
- 2007-03-30 CN CNA2007800124642A patent/CN101415413A/zh active Pending
- 2007-03-30 NZ NZ571251A patent/NZ571251A/en not_active IP Right Cessation
- 2007-03-30 US US12/293,107 patent/US20090062395A1/en not_active Abandoned
- 2007-03-30 MX MX2008012729A patent/MX2008012729A/es not_active Application Discontinuation
- 2007-04-02 TW TW096111640A patent/TW200806283A/zh unknown
- 2007-04-02 CL CL200700912A patent/CL2007000912A1/es unknown
-
2008
- 2008-09-04 ZA ZA200807615A patent/ZA200807615B/xx unknown
- 2008-09-04 IL IL193905A patent/IL193905A0/en unknown
- 2008-09-26 TN TNP2008000383A patent/TNSN08383A1/en unknown
- 2008-10-23 MA MA31327A patent/MA30387B1/fr unknown
- 2008-11-03 NO NO20084625A patent/NO20084625L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AU2007234917A1 (en) | 2007-10-18 |
| WO2007118023A1 (en) | 2007-10-18 |
| NZ571251A (en) | 2011-12-22 |
| AU2007234917B2 (en) | 2011-05-12 |
| MA30387B1 (fr) | 2009-05-04 |
| CN101415413A (zh) | 2009-04-22 |
| CA2645260A1 (en) | 2007-10-18 |
| EP2004167A1 (en) | 2008-12-24 |
| TNSN08383A1 (en) | 2009-12-29 |
| TW200806283A (en) | 2008-02-01 |
| SG170830A1 (en) | 2011-05-30 |
| CL2007000912A1 (es) | 2008-03-14 |
| RU2008143055A (ru) | 2010-05-10 |
| ZA200807615B (en) | 2009-10-28 |
| US20090062395A1 (en) | 2009-03-05 |
| JP2009532494A (ja) | 2009-09-10 |
| NO20084625L (no) | 2008-11-03 |
| IL193905A0 (en) | 2009-08-03 |
| KR20080108515A (ko) | 2008-12-15 |
| MX2008012729A (es) | 2008-10-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2260 DE 29/04/2014. |