BRPI0616228A2 - composto, sal, composiÇço farmacÊutica, e, uso de um composto - Google Patents
composto, sal, composiÇço farmacÊutica, e, uso de um composto Download PDFInfo
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- BRPI0616228A2 BRPI0616228A2 BRPI0616228-2A BRPI0616228A BRPI0616228A2 BR PI0616228 A2 BRPI0616228 A2 BR PI0616228A2 BR PI0616228 A BRPI0616228 A BR PI0616228A BR PI0616228 A2 BRPI0616228 A2 BR PI0616228A2
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US72152705P | 2005-09-29 | 2005-09-29 | |
| US60/721527 | 2005-09-29 | ||
| PCT/US2006/036423 WO2007040982A1 (en) | 2005-09-29 | 2006-09-20 | 5- (phenylisoxazolylethoxy) -triazol- 3 -yl substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0616228A2 true BRPI0616228A2 (pt) | 2011-06-14 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0616228-2A BRPI0616228A2 (pt) | 2005-09-29 | 2006-09-20 | composto, sal, composiÇço farmacÊutica, e, uso de um composto |
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| Country | Link |
|---|---|
| US (4) | US7476684B2 (https=) |
| EP (1) | EP1934209A1 (https=) |
| JP (2) | JP2009510064A (https=) |
| KR (1) | KR20080050421A (https=) |
| CN (1) | CN101273037A (https=) |
| AR (1) | AR058807A1 (https=) |
| AU (1) | AU2006297462A1 (https=) |
| BR (1) | BRPI0616228A2 (https=) |
| CA (1) | CA2623009A1 (https=) |
| EC (1) | ECSP088283A (https=) |
| IL (1) | IL189990A0 (https=) |
| NO (1) | NO20081434L (https=) |
| RU (1) | RU2008108219A (https=) |
| TW (1) | TW200800976A (https=) |
| UA (1) | UA92503C2 (https=) |
| UY (1) | UY29796A1 (https=) |
| WO (1) | WO2007040982A1 (https=) |
| ZA (1) | ZA200802163B (https=) |
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| IL166510A0 (en) * | 2002-08-09 | 2006-01-15 | Nps Pharma Inc | 1,2,4"oxadiazole as modulators of metabotropic glutamate receptor-5 |
| US7585881B2 (en) * | 2004-02-18 | 2009-09-08 | Astrazeneca Ab | Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
| AR058807A1 (es) * | 2005-09-29 | 2008-02-27 | Astrazeneca Ab | 5-(fenilisoxazoletoxi)-triazol-3-il piridinas sustituidas, para el tratamiento de trastornos mediados por el receptor mglur5 |
| TW200821305A (en) * | 2006-10-05 | 2008-05-16 | Astrazeneca Ab | MGluR5 modulators |
| PE20090875A1 (es) | 2007-10-19 | 2009-08-08 | Astrazeneca Ab | Derivados de tetrazol como moduladores de los receptores de glutamato metabotropicos |
| EP2212316A4 (en) * | 2007-10-26 | 2012-06-27 | Astrazeneca Ab | DERIVATIVES OF AMINO1,2,4-TRIAZOLES AS MODULATORS OF MGLUR5 |
| WO2010019101A1 (en) * | 2008-08-12 | 2010-02-18 | Astrazeneca Ab | A crystalline form of 4- (5-{ (ir) -1- [5- (3- chlorophenyl) isoxazol-3-yl] ethoxy } - 4 -methyl- 4h- 1, 2,4- triazol-3-yl) pyridine |
| CN102176910A (zh) * | 2008-08-12 | 2011-09-07 | 阿斯利康(瑞典)有限公司 | 4-(5-{(1r)-1-[5-(3-氯苯基)异噁唑-3-基]乙氧基}-4-甲基-4h-1,2,4-三唑-3-基)吡啶的新晶体形式 |
| CA2751761A1 (en) * | 2008-10-22 | 2010-04-29 | House Ear Institute | Treatment and/or prevention of inner ear conditions by modulation of a metabotropic glutamate receptor |
| MX2011005981A (es) * | 2008-12-12 | 2011-06-27 | Astrazeneca Ab | Nuevo proceso para preparar 4-[4-metil-5-(alquiltio c1-10/aril c5-10-alquilto c1-6)-4h-1,2,4-triazol-3-il]piridinas. |
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| KR20160120157A (ko) | 2015-04-07 | 2016-10-17 | 주식회사 메드팩토 | 암 예방 또는 치료용 약학적 조성물 및 이를 이용한 방법 |
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| NZ517221A (en) | 1999-08-19 | 2004-01-30 | Nps Pharma Inc | Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
| CN1853630A (zh) * | 2001-02-21 | 2006-11-01 | Nps制药公司 | 杂多环化合物及其在亲代谢的谷氨酸受体拮抗剂中的应用 |
| IL166510A0 (en) * | 2002-08-09 | 2006-01-15 | Nps Pharma Inc | 1,2,4"oxadiazole as modulators of metabotropic glutamate receptor-5 |
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| AU2003264018A1 (en) | 2002-08-09 | 2004-02-25 | Astrazeneca Ab | Compounds having an activity at metabotropic glutamate receptors |
| WO2005060971A1 (en) | 2003-12-18 | 2005-07-07 | Astrazeneca Ab | Treatment of reflux-related diseases |
| BRPI0417308A (pt) | 2003-12-19 | 2007-09-11 | Astrazeneca Ab | compostos, respectivo uso, composição farmacêutica, métodos de tratamento de distúrbios mediados pelo receptor mglur5 e de inibição da ativação de receptores mglur5 e processo de produção de compostos de piridila |
| WO2005077368A2 (en) * | 2004-02-03 | 2005-08-25 | Astrazeneca Ab | Treatment of gastro-esophageal reflux disease (gerd) |
| WO2005077345A1 (en) | 2004-02-03 | 2005-08-25 | Astrazeneca Ab | Compounds for the treatment of gastro-esophageal reflux disease |
| DK1716152T3 (da) | 2004-02-18 | 2008-11-03 | Astrazeneca Ab | Kondenserade heterocykliske forbindelser og deres anvendelse som metabotrope receptorantagonister til behandling af gastrointentinde lidelser |
| US7585881B2 (en) * | 2004-02-18 | 2009-09-08 | Astrazeneca Ab | Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists |
| RU2381226C2 (ru) | 2004-02-18 | 2010-02-10 | Астразенека Аб | Полигетероциклические соединения и их применение в качестве антагонистов метаботропного рецептора глутамата |
| EP1720860A1 (en) | 2004-02-18 | 2006-11-15 | AstraZeneca AB | Triazole compounds and their use as metabotropic glutamate receptor antagonists |
| BRPI0507499A (pt) | 2004-02-18 | 2007-07-24 | Astrazeneca Ab | composto ou um sal farmaceuticamente aceitável ou hidrato dos mesmos, composição farmacêutica, uso do composto, e, métodos para tratar distúrbios mediados por mglur 5 e para inibir a ativação de receptores de mglur 5 |
| TW200533664A (en) | 2004-02-18 | 2005-10-16 | Astrazeneca Ab | Tetrazole compounds and their use as metabotropic glutamate receptor antagonists |
| AR058807A1 (es) * | 2005-09-29 | 2008-02-27 | Astrazeneca Ab | 5-(fenilisoxazoletoxi)-triazol-3-il piridinas sustituidas, para el tratamiento de trastornos mediados por el receptor mglur5 |
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- 2006-09-15 AR ARP060104038A patent/AR058807A1/es not_active Application Discontinuation
- 2006-09-15 UY UY29796A patent/UY29796A1/es not_active Application Discontinuation
- 2006-09-19 TW TW095134584A patent/TW200800976A/zh unknown
- 2006-09-20 CA CA002623009A patent/CA2623009A1/en not_active Abandoned
- 2006-09-20 US US11/523,717 patent/US7476684B2/en not_active Expired - Fee Related
- 2006-09-20 UA UAA200802884A patent/UA92503C2/ru unknown
- 2006-09-20 RU RU2008108219/04A patent/RU2008108219A/ru not_active Application Discontinuation
- 2006-09-20 JP JP2008533434A patent/JP2009510064A/ja active Pending
- 2006-09-20 EP EP06803836A patent/EP1934209A1/en not_active Withdrawn
- 2006-09-20 WO PCT/US2006/036423 patent/WO2007040982A1/en not_active Ceased
- 2006-09-20 BR BRPI0616228-2A patent/BRPI0616228A2/pt not_active IP Right Cessation
- 2006-09-20 AU AU2006297462A patent/AU2006297462A1/en not_active Abandoned
- 2006-09-20 US US12/067,270 patent/US20080227824A1/en not_active Abandoned
- 2006-09-20 KR KR1020087006537A patent/KR20080050421A/ko not_active Withdrawn
- 2006-09-20 CN CNA2006800343984A patent/CN101273037A/zh active Pending
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2007
- 2007-07-27 US US11/829,866 patent/US20070270468A1/en not_active Abandoned
- 2007-07-27 US US11/829,867 patent/US20070270469A1/en not_active Abandoned
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2008
- 2008-03-06 IL IL189990A patent/IL189990A0/en unknown
- 2008-03-07 ZA ZA200802163A patent/ZA200802163B/xx unknown
- 2008-03-14 EC EC2008008283A patent/ECSP088283A/es unknown
- 2008-03-19 NO NO20081434A patent/NO20081434L/no not_active Application Discontinuation
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2009
- 2009-09-14 JP JP2009211258A patent/JP2010013476A/ja active Pending
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| Publication number | Publication date |
|---|---|
| US20070270468A1 (en) | 2007-11-22 |
| ZA200802163B (en) | 2009-09-30 |
| JP2009510064A (ja) | 2009-03-12 |
| RU2008108219A (ru) | 2009-11-10 |
| IL189990A0 (en) | 2008-08-07 |
| KR20080050421A (ko) | 2008-06-05 |
| AR058807A1 (es) | 2008-02-27 |
| TW200800976A (en) | 2008-01-01 |
| US20070129408A1 (en) | 2007-06-07 |
| AU2006297462A1 (en) | 2007-04-12 |
| WO2007040982A1 (en) | 2007-04-12 |
| US20080227824A1 (en) | 2008-09-18 |
| NO20081434L (no) | 2008-05-19 |
| JP2010013476A (ja) | 2010-01-21 |
| EP1934209A1 (en) | 2008-06-25 |
| US7476684B2 (en) | 2009-01-13 |
| CA2623009A1 (en) | 2007-04-12 |
| UA92503C2 (ru) | 2010-11-10 |
| UY29796A1 (es) | 2007-04-30 |
| CN101273037A (zh) | 2008-09-24 |
| US20070270469A1 (en) | 2007-11-22 |
| ECSP088283A (es) | 2008-04-28 |
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