ZA200802163B - 5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders - Google Patents

5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders

Info

Publication number
ZA200802163B
ZA200802163B ZA200802163A ZA200802163A ZA200802163B ZA 200802163 B ZA200802163 B ZA 200802163B ZA 200802163 A ZA200802163 A ZA 200802163A ZA 200802163 A ZA200802163 A ZA 200802163A ZA 200802163 B ZA200802163 B ZA 200802163B
Authority
ZA
South Africa
Prior art keywords
phenylisoxazolylethoxy
psychiatric
triazol
neurological
treatment
Prior art date
Application number
ZA200802163A
Other languages
English (en)
Inventor
Minidis Alexander
Wensbo David
Slassi Abdelmalik
Isaac Methvin
Ericsson Caroline
Profir Veronica
Bergstrom Per-Olov
Edwards Louise
Arora Jalaj
Xin Tao
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of ZA200802163B publication Critical patent/ZA200802163B/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Virology (AREA)
  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Anesthesiology (AREA)
ZA200802163A 2005-09-29 2008-03-07 5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders ZA200802163B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US72152705P 2005-09-29 2005-09-29

Publications (1)

Publication Number Publication Date
ZA200802163B true ZA200802163B (en) 2009-09-30

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ZA200802163A ZA200802163B (en) 2005-09-29 2008-03-07 5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders

Country Status (18)

Country Link
US (4) US7476684B2 (https=)
EP (1) EP1934209A1 (https=)
JP (2) JP2009510064A (https=)
KR (1) KR20080050421A (https=)
CN (1) CN101273037A (https=)
AR (1) AR058807A1 (https=)
AU (1) AU2006297462A1 (https=)
BR (1) BRPI0616228A2 (https=)
CA (1) CA2623009A1 (https=)
EC (1) ECSP088283A (https=)
IL (1) IL189990A0 (https=)
NO (1) NO20081434L (https=)
RU (1) RU2008108219A (https=)
TW (1) TW200800976A (https=)
UA (1) UA92503C2 (https=)
UY (1) UY29796A1 (https=)
WO (1) WO2007040982A1 (https=)
ZA (1) ZA200802163B (https=)

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US8080568B1 (en) * 2010-06-29 2011-12-20 Ewha University - Industry Collaboration Foundation 2-pyridyl substituted imidazoles as therapeutic ALK5 and/or ALK4 inhibitors
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JP2013544874A (ja) 2010-12-08 2013-12-19 オスロ ユニヴァーシティー ホスピタル エイチエフ Ｗｎｔシグナル伝達経路阻害薬としてのトリアゾール誘導体
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KR102027368B1 (ko) * 2018-05-29 2019-10-01 서울대학교산학협력단 통증의 강도를 측정하는 방법
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EP1720860A1 (en) 2004-02-18 2006-11-15 AstraZeneca AB Triazole compounds and their use as metabotropic glutamate receptor antagonists
BRPI0507499A (pt) 2004-02-18 2007-07-24 Astrazeneca Ab composto ou um sal farmaceuticamente aceitável ou hidrato dos mesmos, composição farmacêutica, uso do composto, e, métodos para tratar distúrbios mediados por mglur 5 e para inibir a ativação de receptores de mglur 5
TW200533664A (en) 2004-02-18 2005-10-16 Astrazeneca Ab Tetrazole compounds and their use as metabotropic glutamate receptor antagonists
AR058807A1 (es) * 2005-09-29 2008-02-27 Astrazeneca Ab 5-(fenilisoxazoletoxi)-triazol-3-il piridinas sustituidas, para el tratamiento de trastornos mediados por el receptor mglur5

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US20070270468A1 (en) 2007-11-22
JP2009510064A (ja) 2009-03-12
RU2008108219A (ru) 2009-11-10
IL189990A0 (en) 2008-08-07
KR20080050421A (ko) 2008-06-05
AR058807A1 (es) 2008-02-27
TW200800976A (en) 2008-01-01
US20070129408A1 (en) 2007-06-07
AU2006297462A1 (en) 2007-04-12
WO2007040982A1 (en) 2007-04-12
US20080227824A1 (en) 2008-09-18
NO20081434L (no) 2008-05-19
JP2010013476A (ja) 2010-01-21
EP1934209A1 (en) 2008-06-25
US7476684B2 (en) 2009-01-13
CA2623009A1 (en) 2007-04-12
UA92503C2 (ru) 2010-11-10
UY29796A1 (es) 2007-04-30
CN101273037A (zh) 2008-09-24
BRPI0616228A2 (pt) 2011-06-14
US20070270469A1 (en) 2007-11-22
ECSP088283A (es) 2008-04-28

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