BRPI0413361A - forma de dosagem protegida contra abusos - Google Patents

forma de dosagem protegida contra abusos

Info

Publication number
BRPI0413361A
BRPI0413361A BRPI0413361-7A BRPI0413361A BRPI0413361A BR PI0413361 A BRPI0413361 A BR PI0413361A BR PI0413361 A BRPI0413361 A BR PI0413361A BR PI0413361 A BRPI0413361 A BR PI0413361A
Authority
BR
Brazil
Prior art keywords
dosage form
protected against
against abuse
abuse
form protected
Prior art date
Application number
BRPI0413361-7A
Other languages
English (en)
Inventor
Johannes Bartholomous
Heinrich Kugelmann
Elisabeth Arkenau-Meriae
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34199050&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0413361(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10336400A external-priority patent/DE10336400A1/de
Priority claimed from DE10361596A external-priority patent/DE10361596A1/de
Priority claimed from DE102004020220A external-priority patent/DE102004020220A1/de
Priority claimed from DE102004032051A external-priority patent/DE102004032051A1/de
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Priority to BR122018068298A priority Critical patent/BR122018068298B8/pt
Publication of BRPI0413361A publication Critical patent/BRPI0413361A/pt
Publication of BRPI0413361B1 publication Critical patent/BRPI0413361B1/pt
Publication of BRPI0413361B8 publication Critical patent/BRPI0413361B8/pt

Links

Classifications

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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
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    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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  • Health & Medical Sciences (AREA)
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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

"FORMA DE DOSAGEM PROTEGIDA CONTRA ABUSOS". A invenção relaciona-se a uma forma de dosagem termo-formada sem ser expulsa e protegida contra abusos, compreendendo ao menos um polímero natural ou sintético que tem uma força de ruptura de pelo menos de 500 N além de uma ou mais substâncias ativas que poderiam ser sujeitas ao abuso e opcionalmente adjuvantes fisiologicamente aceitáveis. A invenção relaciona-se também a um método correspondente para produzir a dita forma de dosagem.
BRPI0413361A 2003-08-06 2004-08-05 comprimido seguro contra abuso termo-moldado por extrusão sem descoramento BRPI0413361B8 (pt)

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DE102004020220A DE102004020220A1 (de) 2004-04-22 2004-04-22 Verfahren zur Herstellung einer gegen Missbrauch gesicherten, festen Darreichungsform
DE102004032051A DE102004032051A1 (de) 2004-07-01 2004-07-01 Verfahren zur Herstellung einer gegen Missbrauch gesicherten, festen Darreichungsform
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PL1842533T3 (pl) 2013-08-30
HK1113744A1 (en) 2008-10-17
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BRPI0413361B8 (pt) 2021-05-25
EP1658054A1 (de) 2006-05-24
WO2005016313A1 (de) 2005-02-24
PE20050728A1 (es) 2005-11-10
US20160374963A1 (en) 2016-12-29
IL173558A0 (en) 2006-07-05
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US20150150978A1 (en) 2015-06-04
AR045353A1 (es) 2005-10-26
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US20140356294A1 (en) 2014-12-04
PT1658054E (pt) 2007-09-18
US20160166517A1 (en) 2016-06-16
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AU2004264666A1 (en) 2005-02-24
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EP1842533A2 (de) 2007-10-10
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