BRPI0409951A - derivados de anilina, sua produção e uso como agentes farmacêuticos - Google Patents

derivados de anilina, sua produção e uso como agentes farmacêuticos

Info

Publication number
BRPI0409951A
BRPI0409951A BRPI0409951-6A BRPI0409951A BRPI0409951A BR PI0409951 A BRPI0409951 A BR PI0409951A BR PI0409951 A BRPI0409951 A BR PI0409951A BR PI0409951 A BRPI0409951 A BR PI0409951A
Authority
BR
Brazil
Prior art keywords
production
pharmaceutical agents
aniline derivatives
above compounds
compounds
Prior art date
Application number
BRPI0409951-6A
Other languages
English (en)
Inventor
Birgit Bossenmaier
Walter-Gunar Friebe
Ulrike Reiff
Matthias Rueth
Edgar Voss
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33395779&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0409951(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BRPI0409951A publication Critical patent/BRPI0409951A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

"DERIVADOS DE ANILINA, SUA PRODUçãO E USO COMO AGENTES FARMACêUTICOS". São objeto da presente invenção os compostos da fórmula (I), seus sais farmaceuticamente aceitáveis, formas enantioméricas, diastereoisómeros e racematos, a preparação dos compostos acima mencionados, medicamentos que contêm os mesmos e produção dos mesmos, bem como o uso dos compostos acima mencionados no controle ou prevenção de doenças, tal como câncer.
BRPI0409951-6A 2003-04-30 2004-04-29 derivados de anilina, sua produção e uso como agentes farmacêuticos BRPI0409951A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP03009908 2003-04-30
PCT/EP2004/004520 WO2004096796A1 (en) 2003-04-30 2004-04-29 Novel aniline derivatives, their manufacture and use as pharmaceutical agents

Publications (1)

Publication Number Publication Date
BRPI0409951A true BRPI0409951A (pt) 2006-04-25

Family

ID=33395779

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0409951-6A BRPI0409951A (pt) 2003-04-30 2004-04-29 derivados de anilina, sua produção e uso como agentes farmacêuticos

Country Status (20)

Country Link
US (1) US7205326B2 (pt)
EP (1) EP1622896B1 (pt)
JP (1) JP2006515347A (pt)
KR (1) KR100763293B1 (pt)
CN (1) CN100345845C (pt)
AR (1) AR044098A1 (pt)
AT (1) ATE366252T1 (pt)
AU (1) AU2004234060A1 (pt)
BR (1) BRPI0409951A (pt)
CA (1) CA2522809A1 (pt)
CL (1) CL2004000898A1 (pt)
CO (1) CO5640050A2 (pt)
DE (1) DE602004007374T2 (pt)
ES (1) ES2290701T3 (pt)
MX (1) MXPA05011671A (pt)
NO (1) NO20054495L (pt)
RU (1) RU2005137033A (pt)
TW (1) TW200423931A (pt)
WO (1) WO2004096796A1 (pt)
ZA (1) ZA200508694B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200612914A (en) * 2004-03-05 2006-05-01 Hoffmann La Roche Novel oxidized thioether derivatives, their manufacture and use as pharmaceutical agents
FR2876692B1 (fr) 2004-10-19 2007-02-23 Sanofi Aventis Sa Derives de 2-amido-4-phenylthiazole, leur preparation et leur application en therapeutique
US20060116407A1 (en) * 2004-11-22 2006-06-01 Birgit Bossenmaier Amide derivatives
US20090264485A1 (en) * 2005-08-08 2009-10-22 Hans-Willi Krell Pyrazole Derivatives, Their Manufacture and Their Use as Pharmaceutical Agents
CN112920133B (zh) * 2021-01-29 2022-09-16 中国医科大学 (e)-4-甲基-2-(4-(三氟甲基)苯乙烯基)噁唑类化合物及其制备方法与用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69736642T2 (de) 1996-07-19 2007-09-20 Takeda Pharmaceutical Co. Ltd. Heterocyclische Verbindungen, ihre Herstellung und Verwendung
PE20011178A1 (es) 2000-04-07 2001-11-19 Takeda Chemical Industries Ltd Compuestos heterociclicos y su produccion

Also Published As

Publication number Publication date
CA2522809A1 (en) 2004-11-11
WO2004096796A1 (en) 2004-11-11
NO20054495D0 (no) 2005-09-28
US20040254217A1 (en) 2004-12-16
NO20054495L (no) 2005-11-23
CL2004000898A1 (es) 2005-03-04
EP1622896A1 (en) 2006-02-08
KR100763293B1 (ko) 2007-10-04
AR044098A1 (es) 2005-08-24
JP2006515347A (ja) 2006-05-25
US7205326B2 (en) 2007-04-17
DE602004007374D1 (de) 2007-08-16
ZA200508694B (en) 2007-06-27
CN1780830A (zh) 2006-05-31
TW200423931A (en) 2004-11-16
ES2290701T3 (es) 2008-02-16
DE602004007374T2 (de) 2008-03-20
CO5640050A2 (es) 2006-05-31
KR20060006070A (ko) 2006-01-18
ATE366252T1 (de) 2007-07-15
RU2005137033A (ru) 2006-06-27
MXPA05011671A (es) 2005-12-15
CN100345845C (zh) 2007-10-31
AU2004234060A1 (en) 2004-11-11
EP1622896B1 (en) 2007-07-04

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 6A, 7A E 8A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2159 DE 22/05/2012.