BRPI0509394A - derivados de diazina, sua manufatura e uso como agentes farmacêuticos - Google Patents
derivados de diazina, sua manufatura e uso como agentes farmacêuticosInfo
- Publication number
- BRPI0509394A BRPI0509394A BRPI0509394-5A BRPI0509394A BRPI0509394A BR PI0509394 A BRPI0509394 A BR PI0509394A BR PI0509394 A BRPI0509394 A BR PI0509394A BR PI0509394 A BRPI0509394 A BR PI0509394A
- Authority
- BR
- Brazil
- Prior art keywords
- manufacture
- pharmaceutical agents
- compounds
- diazine derivatives
- diazine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Catalysts (AREA)
Abstract
"DERIVADOS DE DIAZINA, SUA MANUFATURA E USO COMO AGENTES FARMACêUTICOS". Os objetivos da presente invenção são os compostos de fórmula (I), os seus sais farmaceuticamente aceitáveis, formas enantioméricas, diastereoisómeros e racematos, a preparação dos compostos acima mencionados, os medicamentos que os contêm e a sua manufatura, bem como o usa dos compostos acima mencionados no controle ou na prevenção de doenças, tais como o câncer.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP04008130 | 2004-04-02 | ||
PCT/EP2005/003347 WO2005097785A1 (en) | 2004-04-02 | 2005-03-31 | Novel diazine derivatives, their manufacture and use as pharmaceutical agents |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0509394A true BRPI0509394A (pt) | 2007-09-18 |
Family
ID=34924554
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0509360-0A BRPI0509360A (pt) | 2004-04-02 | 2005-03-31 | processo para preparação de derivados de diazina |
BRPI0509394-5A BRPI0509394A (pt) | 2004-04-02 | 2005-03-31 | derivados de diazina, sua manufatura e uso como agentes farmacêuticos |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0509360-0A BRPI0509360A (pt) | 2004-04-02 | 2005-03-31 | processo para preparação de derivados de diazina |
Country Status (12)
Country | Link |
---|---|
US (2) | US7179812B2 (pt) |
EP (2) | EP1758897A1 (pt) |
JP (2) | JP2007530626A (pt) |
KR (2) | KR100843533B1 (pt) |
CN (2) | CN1934106A (pt) |
AR (1) | AR048455A1 (pt) |
AU (2) | AU2005231937A1 (pt) |
BR (2) | BRPI0509360A (pt) |
CA (2) | CA2561203A1 (pt) |
RU (2) | RU2006138424A (pt) |
TW (1) | TW200602329A (pt) |
WO (2) | WO2005097785A1 (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0413605D0 (en) * | 2004-06-17 | 2004-07-21 | Addex Pharmaceuticals Sa | Novel compounds |
WO2010064134A2 (en) * | 2008-12-05 | 2010-06-10 | Cadila Pharmaceuticals Ltd. | Process of synthesis of paliperidone |
US20200077658A1 (en) | 2016-12-16 | 2020-03-12 | Basf Se | Pesticidal Compounds |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2952141B2 (ja) * | 1993-01-08 | 1999-09-20 | キヤノン株式会社 | 液晶性化合物、それを含む液晶組成物、及びこれを用いた液晶素子 |
DE19517186A1 (de) * | 1995-05-11 | 1996-11-14 | Bayer Ag | Verfahren zur Herstellung substituierter 2-Fluor-pyrimidine |
ATE338754T1 (de) | 1996-07-19 | 2006-09-15 | Takeda Pharmaceutical | Heterocyclische verbindungen, ihre herstellung und verwendung |
PE20011178A1 (es) * | 2000-04-07 | 2001-11-19 | Takeda Chemical Industries Ltd | Compuestos heterociclicos y su produccion |
EP1310491A1 (en) * | 2000-07-19 | 2003-05-14 | Takeda Chemical Industries, Ltd. | Method for producing 1-substituted-1,2,3-triazole derivative |
US6984653B2 (en) | 2001-10-05 | 2006-01-10 | Takeda Pharmaceutical Company Limited | Heterocyclic compounds, oxazole derivatives, process for preparation of the same and use thereof |
JP2003277379A (ja) * | 2002-01-17 | 2003-10-02 | Takeda Chem Ind Ltd | 含窒素複素環化合物、その製造法および用途 |
WO2003059907A1 (fr) | 2002-01-17 | 2003-07-24 | Takeda Chemical Industries, Ltd. | Composes heterocycliques azotes : procede de preparation et d'utilisation |
WO2003091247A2 (en) | 2002-04-25 | 2003-11-06 | Pharmacia Corporation | Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors |
-
2005
- 2005-03-31 CN CNA2005800095299A patent/CN1934106A/zh active Pending
- 2005-03-31 AU AU2005231937A patent/AU2005231937A1/en not_active Abandoned
- 2005-03-31 AU AU2005231936A patent/AU2005231936A1/en not_active Abandoned
- 2005-03-31 EP EP05779891A patent/EP1758897A1/en not_active Withdrawn
- 2005-03-31 CN CNA2005800095119A patent/CN1934102A/zh active Pending
- 2005-03-31 TW TW094110174A patent/TW200602329A/zh unknown
- 2005-03-31 KR KR1020067020532A patent/KR100843533B1/ko not_active IP Right Cessation
- 2005-03-31 CA CA002561203A patent/CA2561203A1/en not_active Abandoned
- 2005-03-31 BR BRPI0509360-0A patent/BRPI0509360A/pt not_active IP Right Cessation
- 2005-03-31 BR BRPI0509394-5A patent/BRPI0509394A/pt not_active IP Right Cessation
- 2005-03-31 RU RU2006138424/04A patent/RU2006138424A/ru not_active Application Discontinuation
- 2005-03-31 US US11/096,286 patent/US7179812B2/en not_active Expired - Fee Related
- 2005-03-31 US US10/592,820 patent/US20080132699A1/en not_active Abandoned
- 2005-03-31 JP JP2007505494A patent/JP2007530626A/ja active Pending
- 2005-03-31 JP JP2007505495A patent/JP2007530627A/ja active Pending
- 2005-03-31 WO PCT/EP2005/003347 patent/WO2005097785A1/en not_active Application Discontinuation
- 2005-03-31 CA CA002561206A patent/CA2561206A1/en not_active Abandoned
- 2005-03-31 KR KR1020067020524A patent/KR20060131958A/ko active IP Right Grant
- 2005-03-31 RU RU2006138425/04A patent/RU2006138425A/ru not_active Application Discontinuation
- 2005-03-31 AR ARP050101274A patent/AR048455A1/es unknown
- 2005-03-31 WO PCT/EP2005/003346 patent/WO2005097777A1/en active Application Filing
- 2005-03-31 EP EP05716459A patent/EP1737846A1/en not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
KR100843533B1 (ko) | 2008-07-03 |
US20050222228A1 (en) | 2005-10-06 |
RU2006138425A (ru) | 2008-06-20 |
AR048455A1 (es) | 2006-04-26 |
JP2007530626A (ja) | 2007-11-01 |
TW200602329A (en) | 2006-01-16 |
RU2006138424A (ru) | 2008-05-10 |
WO2005097785A1 (en) | 2005-10-20 |
AU2005231937A1 (en) | 2005-10-20 |
KR20070006822A (ko) | 2007-01-11 |
CA2561206A1 (en) | 2005-10-20 |
CN1934106A (zh) | 2007-03-21 |
EP1758897A1 (en) | 2007-03-07 |
KR20060131958A (ko) | 2006-12-20 |
WO2005097777A1 (en) | 2005-10-20 |
CN1934102A (zh) | 2007-03-21 |
US20080132699A1 (en) | 2008-06-05 |
CA2561203A1 (en) | 2005-10-20 |
JP2007530627A (ja) | 2007-11-01 |
BRPI0509360A (pt) | 2007-09-11 |
EP1737846A1 (en) | 2007-01-03 |
AU2005231936A1 (en) | 2005-10-20 |
US7179812B2 (en) | 2007-02-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 5A, 6A E 7A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012. |