BRPI0408148A - derivados de ácido benzoilureidopiridil-piperidina e -pirrolidina-carboxìlico, processos para a preparação e uso dos mesmos - Google Patents
derivados de ácido benzoilureidopiridil-piperidina e -pirrolidina-carboxìlico, processos para a preparação e uso dos mesmosInfo
- Publication number
- BRPI0408148A BRPI0408148A BRPI0408148-0A BRPI0408148A BRPI0408148A BR PI0408148 A BRPI0408148 A BR PI0408148A BR PI0408148 A BRPI0408148 A BR PI0408148A BR PI0408148 A BRPI0408148 A BR PI0408148A
- Authority
- BR
- Brazil
- Prior art keywords
- benzoylureidopyridyl
- piperidine
- carboxylic acid
- acid derivatives
- processes
- Prior art date
Links
- NMDAFFPZWCMMLW-UHFFFAOYSA-N n-[(1-pyridin-2-ylpiperidin-2-yl)carbamoyl]benzamide Chemical compound C=1C=CC=CC=1C(=O)NC(=O)NC1CCCCN1C1=CC=CC=N1 NMDAFFPZWCMMLW-UHFFFAOYSA-N 0.000 title abstract 2
- NYCVCXMSZNOGDH-UHFFFAOYSA-N pyrrolidine-1-carboxylic acid Chemical class OC(=O)N1CCCC1 NYCVCXMSZNOGDH-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 239000003814 drug Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 208000001072 type 2 diabetes mellitus Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Diabetes (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Obesity (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Emergency Medicine (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10309929A DE10309929B4 (de) | 2003-03-07 | 2003-03-07 | Substituierte Benzoylureidopyridyl-piperidin- und -pyrrolidin-carbonsäurederivate, Verfahren zu deren Herstellung und deren Verwendung |
| PCT/EP2004/001735 WO2004078743A1 (de) | 2003-03-07 | 2004-02-21 | Substituierte benzoylureidopyridyl-piperidin- und -pyrrolidin-carbonsäurederivate, verfahren zu deren herstellung und deren verwendung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0408148A true BRPI0408148A (pt) | 2006-03-01 |
Family
ID=32945839
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0408148-0A BRPI0408148A (pt) | 2003-03-07 | 2004-02-21 | derivados de ácido benzoilureidopiridil-piperidina e -pirrolidina-carboxìlico, processos para a preparação e uso dos mesmos |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP1603895B1 (enExample) |
| JP (1) | JP2006519795A (enExample) |
| KR (1) | KR20050108487A (enExample) |
| CN (1) | CN1759109A (enExample) |
| AT (1) | ATE386735T1 (enExample) |
| AU (1) | AU2004218267A1 (enExample) |
| BR (1) | BRPI0408148A (enExample) |
| CA (1) | CA2518322A1 (enExample) |
| CO (1) | CO5690587A2 (enExample) |
| DE (2) | DE10309929B4 (enExample) |
| HR (1) | HRP20050779A2 (enExample) |
| MA (1) | MA27745A1 (enExample) |
| MX (1) | MXPA05009122A (enExample) |
| NO (1) | NO20054418L (enExample) |
| PL (1) | PL377293A1 (enExample) |
| RU (1) | RU2005131011A (enExample) |
| WO (1) | WO2004078743A1 (enExample) |
| ZA (1) | ZA200506119B (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006055435A1 (en) | 2004-11-15 | 2006-05-26 | Bristol-Myers Squibb Company | 2-aminonaphthalene derivatives and related glycogen phosphorylase inhibitors |
| WO2006053274A2 (en) | 2004-11-15 | 2006-05-18 | Bristol-Myers Squibb Company | 2-amino-1-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors |
| US7226942B2 (en) | 2004-11-15 | 2007-06-05 | Bristol-Myers Squibb Company | 2-amino-4-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors |
| US7365061B2 (en) | 2004-11-15 | 2008-04-29 | Bristol-Myers Squibb Company | 2-Amino-3-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors |
| PE20110235A1 (es) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | Combinaciones farmaceuticas que comprenden linagliptina y metmorfina |
| MX2012003389A (es) * | 2009-10-06 | 2012-04-10 | Bristol Myers Squibb Co | Moduladores de gpr40 de pirrolidina. |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3034004A1 (de) * | 1980-09-10 | 1982-04-22 | Hoechst Ag, 6000 Frankfurt | Sulfonylharnstoffe, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen und ihre verwendung |
| DE10116768A1 (de) * | 2001-04-04 | 2002-10-10 | Aventis Pharma Gmbh | Acylphenylharnstoffderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| CA2411082A1 (en) * | 2000-06-09 | 2002-12-05 | Aventis Pharma Deutschland Gmbh | Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament |
| DE10125567B4 (de) * | 2001-05-25 | 2004-08-26 | Aventis Pharma Deutschland Gmbh | Carbonamid substituierte Phenylharnstoffderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| PE20021091A1 (es) * | 2001-05-25 | 2003-02-04 | Aventis Pharma Gmbh | Derivados de fenilurea sustituidos con carbonamida y procedimiento para su preparacion |
| IL164249A0 (en) * | 2002-04-11 | 2005-12-18 | Aventis Pharma Gmbh | Acyl-3-carboxphenylurea derivatives, processes forpreparing them and their use |
| CA2493373A1 (en) * | 2002-07-11 | 2004-01-22 | Aventis Pharma Deutschland Gmbh | Urea-substituted and urethane-substituted acylureas, methods for the production thereof and their use as medicaments |
| AU2003249937A1 (en) * | 2002-07-12 | 2004-02-02 | Sanofi-Aventis Deutschland Gmbh | Heterocyclically substituted benzoylureas, method for their production and their use as medicaments |
-
2003
- 2003-03-07 DE DE10309929A patent/DE10309929B4/de not_active Expired - Fee Related
-
2004
- 2004-02-21 KR KR1020057016583A patent/KR20050108487A/ko not_active Withdrawn
- 2004-02-21 CA CA002518322A patent/CA2518322A1/en not_active Abandoned
- 2004-02-21 EP EP04713467A patent/EP1603895B1/de not_active Expired - Lifetime
- 2004-02-21 BR BRPI0408148-0A patent/BRPI0408148A/pt not_active IP Right Cessation
- 2004-02-21 AT AT04713467T patent/ATE386735T1/de not_active IP Right Cessation
- 2004-02-21 WO PCT/EP2004/001735 patent/WO2004078743A1/de not_active Ceased
- 2004-02-21 HR HR20050779A patent/HRP20050779A2/xx not_active Application Discontinuation
- 2004-02-21 RU RU2005131011/04A patent/RU2005131011A/ru not_active Application Discontinuation
- 2004-02-21 DE DE502004006253T patent/DE502004006253D1/de not_active Expired - Lifetime
- 2004-02-21 AU AU2004218267A patent/AU2004218267A1/en not_active Abandoned
- 2004-02-21 CN CNA2004800062407A patent/CN1759109A/zh active Pending
- 2004-02-21 JP JP2006504448A patent/JP2006519795A/ja not_active Ceased
- 2004-02-21 MX MXPA05009122A patent/MXPA05009122A/es unknown
- 2004-02-21 PL PL377293A patent/PL377293A1/pl not_active Application Discontinuation
-
2005
- 2005-08-01 ZA ZA200506119A patent/ZA200506119B/en unknown
- 2005-09-06 CO CO05089471A patent/CO5690587A2/es not_active Application Discontinuation
- 2005-09-07 MA MA28485A patent/MA27745A1/fr unknown
- 2005-09-23 NO NO20054418A patent/NO20054418L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MA27745A1 (fr) | 2006-02-01 |
| EP1603895A1 (de) | 2005-12-14 |
| DE10309929B4 (de) | 2006-02-23 |
| PL377293A1 (pl) | 2006-01-23 |
| CA2518322A1 (en) | 2004-09-16 |
| CO5690587A2 (es) | 2006-10-31 |
| JP2006519795A (ja) | 2006-08-31 |
| RU2005131011A (ru) | 2006-05-10 |
| KR20050108487A (ko) | 2005-11-16 |
| CN1759109A (zh) | 2006-04-12 |
| WO2004078743A1 (de) | 2004-09-16 |
| HRP20050779A2 (en) | 2006-10-31 |
| ZA200506119B (en) | 2006-11-29 |
| EP1603895B1 (de) | 2008-02-20 |
| MXPA05009122A (es) | 2005-10-20 |
| AU2004218267A1 (en) | 2004-09-16 |
| NO20054418L (no) | 2005-09-23 |
| ATE386735T1 (de) | 2008-03-15 |
| DE502004006253D1 (de) | 2008-04-03 |
| DE10309929A1 (de) | 2004-12-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 5A, 6A, 7A E 8A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2159 DE 22/05/2012. |