BR9904082A - Processo para a preparação de sais de ácido de trovafloxacina - Google Patents
Processo para a preparação de sais de ácido de trovafloxacinaInfo
- Publication number
- BR9904082A BR9904082A BR9904082-4A BR9904082A BR9904082A BR 9904082 A BR9904082 A BR 9904082A BR 9904082 A BR9904082 A BR 9904082A BR 9904082 A BR9904082 A BR 9904082A
- Authority
- BR
- Brazil
- Prior art keywords
- acid
- preparation
- trovafloxacin
- acid salts
- salts
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Indole Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Peptides Or Proteins (AREA)
Abstract
Patente de Invenção: <B>"PROCESSO PARA A PREPARAçãO DE SAIS DE áCIDO DE TROVAFLOXACINA"<D>. Os sais de ácido da trovafloxacina são preparados por hidrólise de iminas intermediárias utilizando um ácido mineral, incluindo mas não se limitando a ácido metanossulfónico, ácido etanossulfónico, ácido benzenossulfónico, ácido nítrico, ácido sulfúrico, ácido fosfórico, ácido clorídrico, ácido bromídrico, ácido tartárico, ácido cítrico, ácido acético e ácido maleico. Os sais de ácido da trovafloxacinasão úteis como agentes antibióticos.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9894498P | 1998-09-03 | 1998-09-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9904082A true BR9904082A (pt) | 2000-09-12 |
Family
ID=22271674
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9904082-4A BR9904082A (pt) | 1998-09-03 | 1999-09-03 | Processo para a preparação de sais de ácido de trovafloxacina |
Country Status (40)
| Country | Link |
|---|---|
| US (1) | US6359137B1 (pt) |
| EP (1) | EP0989119A1 (pt) |
| JP (1) | JP3354526B2 (pt) |
| KR (1) | KR20000022858A (pt) |
| CN (1) | CN1248580A (pt) |
| AP (1) | AP1118A (pt) |
| AR (1) | AR021475A1 (pt) |
| AU (1) | AU761035B2 (pt) |
| BG (1) | BG103703A (pt) |
| BR (1) | BR9904082A (pt) |
| CA (1) | CA2281244C (pt) |
| CO (1) | CO5251466A1 (pt) |
| EA (1) | EA002340B1 (pt) |
| EE (1) | EE04118B1 (pt) |
| GE (1) | GEP20022785B (pt) |
| GT (1) | GT199900142A (pt) |
| HN (1) | HN1999000141A (pt) |
| HR (1) | HRP990274A2 (pt) |
| HU (1) | HUP9902967A3 (pt) |
| ID (1) | ID23718A (pt) |
| IL (1) | IL131614A0 (pt) |
| IN (1) | IN191583B (pt) |
| IS (1) | IS5168A (pt) |
| MA (1) | MA24966A1 (pt) |
| MY (1) | MY130800A (pt) |
| NO (1) | NO994261L (pt) |
| NZ (1) | NZ337605A (pt) |
| OA (1) | OA11152A (pt) |
| PA (1) | PA8481001A1 (pt) |
| PE (1) | PE20001026A1 (pt) |
| PL (1) | PL335246A1 (pt) |
| SG (1) | SG74748A1 (pt) |
| SK (1) | SK116599A3 (pt) |
| SV (1) | SV1999000144A (pt) |
| TN (1) | TNSN99164A1 (pt) |
| TR (1) | TR199902138A2 (pt) |
| TW (1) | TW520369B (pt) |
| UY (1) | UY25686A1 (pt) |
| YU (1) | YU43199A (pt) |
| ZA (1) | ZA995630B (pt) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104892507B (zh) * | 2015-05-26 | 2018-08-28 | 徐州天意动物药业股份有限公司 | 水溶性甲磺酸沙拉沙星及其制备方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5164402A (en) * | 1989-08-16 | 1992-11-17 | Pfizer Inc | Azabicyclo quinolone and naphthyridinone carboxylic acids |
| WO1995019361A1 (en) * | 1994-01-18 | 1995-07-20 | Pfizer Inc. | Process and intermediates for preparing naphthyridonecarboxylic acid salts |
| EP0789697B1 (en) * | 1995-06-06 | 1998-06-17 | Pfizer Inc. | CRYSTAL FORM OF ANHYDROUS 7-((1a,5a, 6a)-6-AMINO-3-AZABICYCLO ( 3.1. 0]HEX-3-YL)-6-FLUORO-1-(2,4-DIFLUOROPHENYL)-1,4-DIHYDRO-4-OXO-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID, METHANESULFONIC ACID SALT |
| JPH0912547A (ja) * | 1995-06-23 | 1997-01-14 | Chisso Corp | ニューキノロン系化合物中間体の製造方法 |
| JPH0912546A (ja) * | 1995-06-23 | 1997-01-14 | Chisso Corp | アザビシクロ環化合物および製造方法 |
| WO1997007800A1 (en) * | 1995-08-29 | 1997-03-06 | Pfizer Inc. | Zwitterionic forms of trovafloxacin |
| PA8464701A1 (es) * | 1998-01-16 | 2000-09-29 | Pfizer Prod Inc | Procedimiento e intermedios para preparar naftiridonas |
| US6184380B1 (en) * | 1999-01-25 | 2001-02-06 | Pfizer Inc. | Process for preparing naphthyridones and intermediates |
-
1999
- 1999-08-17 HN HN1999000141A patent/HN1999000141A/es unknown
- 1999-08-25 GT GT199900142A patent/GT199900142A/es unknown
- 1999-08-25 SK SK1165-99A patent/SK116599A3/sk unknown
- 1999-08-26 US US09/383,320 patent/US6359137B1/en not_active Expired - Fee Related
- 1999-08-26 IL IL13161499A patent/IL131614A0/xx unknown
- 1999-08-27 AU AU44826/99A patent/AU761035B2/en not_active Ceased
- 1999-08-30 TW TW088114861A patent/TW520369B/zh active
- 1999-08-30 IS IS5168A patent/IS5168A/is unknown
- 1999-08-31 OA OA9900199A patent/OA11152A/en unknown
- 1999-08-31 PA PA19998481001A patent/PA8481001A1/es unknown
- 1999-08-31 UY UY25686A patent/UY25686A1/es not_active Application Discontinuation
- 1999-09-01 PE PE1999000878A patent/PE20001026A1/es not_active Application Discontinuation
- 1999-09-01 MA MA25749A patent/MA24966A1/fr unknown
- 1999-09-01 IN IN1171DE1999 patent/IN191583B/en unknown
- 1999-09-01 EP EP99306947A patent/EP0989119A1/en not_active Withdrawn
- 1999-09-01 ZA ZA9905630A patent/ZA995630B/xx unknown
- 1999-09-01 TN TNTNSN99164A patent/TNSN99164A1/fr unknown
- 1999-09-01 SG SG1999004240A patent/SG74748A1/en unknown
- 1999-09-01 BG BG103703A patent/BG103703A/bg unknown
- 1999-09-01 EA EA199900708A patent/EA002340B1/ru not_active IP Right Cessation
- 1999-09-01 CA CA002281244A patent/CA2281244C/en not_active Expired - Fee Related
- 1999-09-01 MY MYPI99003775A patent/MY130800A/en unknown
- 1999-09-01 JP JP24737399A patent/JP3354526B2/ja not_active Expired - Fee Related
- 1999-09-02 CN CN99118470A patent/CN1248580A/zh active Pending
- 1999-09-02 NO NO994261A patent/NO994261L/no unknown
- 1999-09-02 EE EEP199900457A patent/EE04118B1/xx not_active IP Right Cessation
- 1999-09-02 ID IDP990831D patent/ID23718A/id unknown
- 1999-09-02 SV SV1999000144A patent/SV1999000144A/es not_active Application Discontinuation
- 1999-09-02 YU YU43199A patent/YU43199A/sh unknown
- 1999-09-02 KR KR1019990037060A patent/KR20000022858A/ko active IP Right Grant
- 1999-09-02 TR TR1999/02138A patent/TR199902138A2/xx unknown
- 1999-09-02 NZ NZ337605A patent/NZ337605A/xx unknown
- 1999-09-02 AP APAP/P/1999/001667A patent/AP1118A/en active
- 1999-09-02 HU HU9902967A patent/HUP9902967A3/hu unknown
- 1999-09-02 AR ARP990104424A patent/AR021475A1/es unknown
- 1999-09-03 BR BR9904082-4A patent/BR9904082A/pt not_active Application Discontinuation
- 1999-09-03 PL PL99335246A patent/PL335246A1/xx not_active Application Discontinuation
- 1999-09-03 GE GEAP19994978A patent/GEP20022785B/en unknown
- 1999-09-03 HR HR990274A patent/HRP990274A2/hr not_active Application Discontinuation
- 1999-09-03 CO CO99055924A patent/CO5251466A1/es not_active Application Discontinuation
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BR0111947A (pt) | Composto, composição farmacêutica, método para o tratamento de um distúrbio em um mamìfero, uso de um composto e processo para preparar, um composto | |
| BR0107425A (pt) | Processo para a preparação compostos de derivados de ácido 3-hidróxi picolìnico e uso dos compostos | |
| BR0308967A (pt) | Derivados de quinolina e isoquinolina, um processo para a sua preparação e sua aplicação como inibidores de inflamação | |
| BR0209241A (pt) | Processo para preparação de derivados de9-deoxo-9a-aza-9a-homoeritromicina a 4-substituida | |
| BR0009411A (pt) | Composto de anilina substituìda, e, processo para a preparação e uso de compostos | |
| BR0210531A (pt) | Derivados de ácido sulfÈnico | |
| PT1265888E (pt) | Processo para producao de derivados de (s)-nicotina 6-substituida e compost0s intermediarios | |
| BR9912556A (pt) | Triazolpiridinas para o tratamento de distúrbios trombóticos | |
| BR0108990A (pt) | Processo para preparação de derivados de pirimidona com atividade antifungos | |
| BR0210664A (pt) | Processo de sìntese técnico para produção de tropenol | |
| BR0011996A (pt) | Preparação de piperidin-4-onas substituìdas | |
| BR9904082A (pt) | Processo para a preparação de sais de ácido de trovafloxacina | |
| BR0317665A (pt) | 1-alquil-3-aminoindazóis | |
| BR0007982A (pt) | Processo para a preparação de um composto, e,composto | |
| DK1174418T3 (da) | Fremgangsmåde til fremstilling af vandfrit gabapentin af farmaceutisk kvalitet | |
| ITMI20002187A0 (it) | Processo per la produzione dell'acido r(+) -lipico | |
| BRPI0013751B8 (pt) | processo para produção de derivados de ácido naftiridina-3-carboxílico. | |
| BR9909151A (pt) | processos para preparação de intermediários | |
| BRPI0000967A (pt) | processos para preparação de compostos secretagogos de hormônio de crescimento | |
| BR0212451A (pt) | Antagonistas de receptores de ccr-3 v | |
| BR0315762A (pt) | Utilização de derivados de ácidos piperazino-sulfónicos como antagonistas ccr1 para o tratamento de fibrose, doença de alzheimer e outras doenças | |
| BR0309037A (pt) | Processo para a preparação de sais ácidos de gemifloxacina, e, intermediário | |
| BR9914775A (pt) | Processo quìmico para preparação deintermediários | |
| BR9900797A (pt) | Processo para a preparação de piridinas substituìdas. | |
| BR9910603A (pt) | Método aprimorado paraa preparar derivados de norbenzomorfano valiosos farmaceuticamente |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFIRO O PRESENTE PEDIDO DE ACORDO COM ART. 8O, 11,13, E 25 DA LPI. |
|
| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL. |