BRPI0013751B8 - processo para produção de derivados de ácido naftiridina-3-carboxílico. - Google Patents

processo para produção de derivados de ácido naftiridina-3-carboxílico.

Info

Publication number
BRPI0013751B8
BRPI0013751B8 BRPI0013751A BR0013751A BRPI0013751B8 BR PI0013751 B8 BRPI0013751 B8 BR PI0013751B8 BR PI0013751 A BRPI0013751 A BR PI0013751A BR 0013751 A BR0013751 A BR 0013751A BR PI0013751 B8 BRPI0013751 B8 BR PI0013751B8
Authority
BR
Brazil
Prior art keywords
naphthyridine
carboxylic acid
acid derivatives
producing
formula
Prior art date
Application number
BRPI0013751A
Other languages
English (en)
Other versions
BR0013751A (pt
BR0013751B1 (pt
Inventor
Choi Hoon
David Hayler John
Cho Sungwok
Original Assignee
Lg Chemical Ltd
Sb Pharmco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lg Chemical Ltd, Sb Pharmco Inc filed Critical Lg Chemical Ltd
Publication of BR0013751A publication Critical patent/BR0013751A/pt
Publication of BR0013751B1 publication Critical patent/BR0013751B1/pt
Publication of BRPI0013751B8 publication Critical patent/BRPI0013751B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Abstract

"processo para produção de derivados de ácido naftiridina-3-carboxílico". processo para produção de derivados de ácido naftiridina-3-carboxílico de fórmula (i) possuindo atividade antibacteriana.
BRPI0013751A 1999-09-03 2000-09-01 processo para produção de derivados de ácido naftiridina-3-carboxílico. BRPI0013751B8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9920917.3A GB9920917D0 (en) 1999-09-03 1999-09-03 Novel process
PCT/GB2000/003366 WO2001018002A1 (en) 1999-09-03 2000-09-01 Process for production of naphthyridine-3-carboxylic acid derivatives

Publications (3)

Publication Number Publication Date
BR0013751A BR0013751A (pt) 2002-05-07
BR0013751B1 BR0013751B1 (pt) 2013-02-05
BRPI0013751B8 true BRPI0013751B8 (pt) 2021-05-25

Family

ID=10860353

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0013751A BRPI0013751B8 (pt) 1999-09-03 2000-09-01 processo para produção de derivados de ácido naftiridina-3-carboxílico.

Country Status (23)

Country Link
US (1) US7232907B2 (pt)
EP (1) EP1214321B1 (pt)
JP (1) JP4208464B2 (pt)
KR (1) KR100724311B1 (pt)
CN (1) CN1275963C (pt)
AR (1) AR029002A1 (pt)
AT (1) ATE271050T1 (pt)
AU (1) AU773722B2 (pt)
BR (1) BRPI0013751B8 (pt)
CA (1) CA2383753C (pt)
CO (1) CO5470281A1 (pt)
DE (1) DE60012196T2 (pt)
DK (1) DK1214321T3 (pt)
ES (1) ES2223574T3 (pt)
GB (1) GB9920917D0 (pt)
HK (1) HK1047093B (pt)
MX (1) MXPA02002355A (pt)
MY (1) MY125309A (pt)
PT (1) PT1214321E (pt)
SI (1) SI1214321T1 (pt)
TW (1) TWI274753B (pt)
WO (1) WO2001018002A1 (pt)
ZA (1) ZA200201781B (pt)

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CA2281817C (en) * 1999-06-29 2008-07-29 Smithkline Beecham Corporation Methods of use of fluoroquinolone compounds against maxillary sinus pathogenic bacteria
GB9920917D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel process
GB9920919D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel compound
US7199242B2 (en) 2001-08-02 2007-04-03 Lg Life Sciences Limited Processes for the production of amino-protected derivatives of 4-aminomethylene-pyrrolidin-3-one and/or 4-aminomethylene-pyrrolidin-3-alkoxyimino derivatives and/or gemifloxacin or a salt thereof
KR100517638B1 (ko) * 2002-04-08 2005-09-28 주식회사 엘지생명과학 게미플록사신 산염의 새로운 제조방법
KR100653334B1 (ko) * 2003-03-07 2006-12-04 주식회사 엘지생명과학 4-아미노메틸-3-알콕시이미노피롤리딘 메탄설폰산염의 신규한 제조 방법
WO2006134431A1 (en) * 2005-05-03 2006-12-21 Ranbaxy Laboratories Limited Formate salt of gemifloxacin
EP2159225A1 (en) 2005-06-15 2010-03-03 Hetero Drugs Limited Gemifloxacin process and polymorphs
WO2008053324A1 (en) * 2006-10-31 2008-05-08 Orchid Chemicals & Pharmaceuticals Limited An improved process for the preparation of gemifloxacin mesylate

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IN162769B (pt) 1984-11-13 1988-07-09 Kyorin Seiyaku Kk
NZ222047A (en) 1986-10-08 1991-01-29 Bristol Myers Co Quinoline - or naphthyridine - carboxylic acid anti-bacterial agents
JPH01100165A (ja) 1987-10-13 1989-04-18 Shionogi & Co Ltd オキシムまたはヒドロキシアミン誘導体系抗菌剤
US4920120A (en) 1988-01-25 1990-04-24 Warner-Lambert Company Antibacterial agents
JPH0356479A (ja) 1989-07-24 1991-03-12 Takeshi Yokota 水溶性キノロン誘導体のｐ‐トルエンスルホン酸塩
IE66202B1 (en) 1989-08-16 1995-12-13 Pfizer Azabicyclo quinolone carboxylic acids
US5137892A (en) 1990-12-12 1992-08-11 Abbott Laboratories Quinoline, naphthyridine and pyridobenzoxazine derivatives
US5276041A (en) 1991-11-08 1994-01-04 Kaken Pharmaceutical Co., Ltd. Oxime derivatives
JPH0673056A (ja) 1992-08-26 1994-03-15 Kaken Pharmaceut Co Ltd キノリンカルボン酸誘導体およびその塩
US5776944A (en) 1994-06-16 1998-07-07 Lg Chemical Ltd. 7-(4-aminomethyl-3-methyloxyiminopyrroplidin-1-yl)-1-cyclopropyl-6-flu oro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid and the process for the preparation thereof
EP0688772B1 (en) 1994-06-16 1999-05-06 LG Chemical Limited Quinoline carboxylic acid derivatives having 7-(4-amino-methyl-3-oxime) pyrrolidine substituents and processes for their preparation
JP3449658B2 (ja) 1994-12-21 2003-09-22 杏林製薬株式会社 安定性に優れた８−アルコキシキノロンカルボン酸水和物並びにその製造方法
ES2117426T3 (es) 1995-06-06 1998-08-01 Pfizer Forma cristalina de la sal anhidra compuesta de los acidos 7-((1a,5a,6a)-6-amino-3-azabiciclo(3.1.0.)hex-3-il)-6-fluoro-1-(2,4-difluorofenil)-1,4-dihidro-4-oxo-1,8-naftiridina-3-carboxilico y metanosulfonico.
KR100291882B1 (ko) 1995-08-11 2001-10-26 디. 제이. 우드, 스피겔 알렌 제이 (1에스,2에스)-1-(4-하이드록시페닐)-2-(4-하이드록시-4-페닐피페리딘-1-일)-1-프로판올메탄설포네이트트리하이드레이트
UA49880C2 (uk) 1996-03-29 2002-10-15 Смітклайн Бічам Корпорейшн Дигідрат ерпоcартану, фармацевтична композиція, спосіб отримання твердої дозованої форми, спосіб блокування рецепторів ангіотензину іі
MA24500A1 (fr) * 1997-03-21 1998-10-01 Lg Life Sciences Ltd Derive du sel d'acide carboxylique de naphthyridine .
KR100286874B1 (ko) 1998-03-04 2001-04-16 성재갑 보호된 4-아미노메틸-피롤리딘-3-온의 제조방법
DE69911203T2 (de) 1998-05-29 2004-07-15 Pharmacia & Upjohn Co., Kalamazoo 3-[(1'-n-methylamino)ethyl-n-benzyl]pyrrolidin-monomethanesulfonat
GB9820405D0 (en) 1998-09-18 1998-11-11 Smithkline Beecham Plc Process
PT1223935E (pt) 1999-06-29 2008-04-03 Lg Life Sciences Ltd Utilização de compostos de gemifloxacina contra bactérias
EP1401440A4 (en) 1999-09-01 2006-07-05 Lg Life Sciences Ltd METHODS OF USING FLUOROQUINOLONE COMPOUNDS AGAINST BACTERIA
GB9920917D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel process
GB9920919D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel compound
WO2001021176A1 (en) 1999-09-22 2001-03-29 Smithkline Beecham Corporation Methods of use of fluoroquinolone compounds against bacteria
KR20010091379A (ko) 2000-03-15 2001-10-23 성재갑 7-(4-아미노메틸-3-옥심)피롤리딘 치환체를 갖는 퀴놀린카르복실산 유도체의 신규 제조방법
KR20020018560A (ko) 2000-09-01 2002-03-08 성재갑 3-아미노메틸-4-ｚ-메톡시이미노피롤리딘의 신규 제조방법

Also Published As

Publication number Publication date
CO5470281A1 (es) 2004-12-30
HK1047093B (zh) 2005-05-27
CA2383753A1 (en) 2001-03-15
US20050176961A1 (en) 2005-08-11
DE60012196D1 (de) 2004-08-19
ES2223574T3 (es) 2005-03-01
CA2383753C (en) 2011-06-28
US7232907B2 (en) 2007-06-19
CN1377350A (zh) 2002-10-30
EP1214321A1 (en) 2002-06-19
PT1214321E (pt) 2004-10-29
AR029002A1 (es) 2003-06-04
MY125309A (en) 2006-07-31
WO2001018002A1 (en) 2001-03-15
EP1214321B1 (en) 2004-07-14
DK1214321T3 (da) 2004-10-25
JP2003508532A (ja) 2003-03-04
ZA200201781B (en) 2003-06-25
MXPA02002355A (es) 2004-07-16
AU7019700A (en) 2001-04-10
HK1047093A1 (en) 2003-02-07
GB9920917D0 (en) 1999-11-10
KR20020041421A (ko) 2002-06-01
BR0013751A (pt) 2002-05-07
KR100724311B1 (ko) 2007-06-04
CN1275963C (zh) 2006-09-20
TWI274753B (en) 2007-03-01
DE60012196T2 (de) 2005-08-18
BR0013751B1 (pt) 2013-02-05
SI1214321T1 (en) 2004-12-31
JP4208464B2 (ja) 2009-01-14
ATE271050T1 (de) 2004-07-15
AU773722B2 (en) 2004-06-03

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B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
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