BR0013751A - Processo para produção de derivados de ácido naftiridina-3-carboxìlico - Google Patents

Processo para produção de derivados de ácido naftiridina-3-carboxìlico

Info

Publication number
BR0013751A
BR0013751A BR0013751-0A BR0013751A BR0013751A BR 0013751 A BR0013751 A BR 0013751A BR 0013751 A BR0013751 A BR 0013751A BR 0013751 A BR0013751 A BR 0013751A
Authority
BR
Brazil
Prior art keywords
production
carboxylic acid
acid derivatives
naphthyridine
naftyridine
Prior art date
Application number
BR0013751-0A
Other languages
English (en)
Other versions
BR0013751B1 (pt
BRPI0013751B8 (pt
Inventor
Sungwook Cho
Hoon Choi
John David Hayler
Original Assignee
Sb Pharmco Inc
Lg Chemical Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sb Pharmco Inc, Lg Chemical Ltd filed Critical Sb Pharmco Inc
Publication of BR0013751A publication Critical patent/BR0013751A/pt
Publication of BR0013751B1 publication Critical patent/BR0013751B1/pt
Publication of BRPI0013751B8 publication Critical patent/BRPI0013751B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

"PROCESSO PARA PRODUçãO DE DERIVADOS DE áCIDO NAFTIRIDINA-3-CARBOXìLICO". Processo para produção de derivados de ácido Naftiridina-3-carboxílico de fórmula (I) possuindo atividade antibacteriana.
BRPI0013751A 1999-09-03 2000-09-01 processo para produção de derivados de ácido naftiridina-3-carboxílico. BRPI0013751B8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9920917.3A GB9920917D0 (en) 1999-09-03 1999-09-03 Novel process
PCT/GB2000/003366 WO2001018002A1 (en) 1999-09-03 2000-09-01 Process for production of naphthyridine-3-carboxylic acid derivatives

Publications (3)

Publication Number Publication Date
BR0013751A true BR0013751A (pt) 2002-05-07
BR0013751B1 BR0013751B1 (pt) 2013-02-05
BRPI0013751B8 BRPI0013751B8 (pt) 2021-05-25

Family

ID=10860353

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0013751A BRPI0013751B8 (pt) 1999-09-03 2000-09-01 processo para produção de derivados de ácido naftiridina-3-carboxílico.

Country Status (23)

Country Link
US (1) US7232907B2 (pt)
EP (1) EP1214321B1 (pt)
JP (1) JP4208464B2 (pt)
KR (1) KR100724311B1 (pt)
CN (1) CN1275963C (pt)
AR (1) AR029002A1 (pt)
AT (1) ATE271050T1 (pt)
AU (1) AU773722B2 (pt)
BR (1) BRPI0013751B8 (pt)
CA (1) CA2383753C (pt)
CO (1) CO5470281A1 (pt)
DE (1) DE60012196T2 (pt)
DK (1) DK1214321T3 (pt)
ES (1) ES2223574T3 (pt)
GB (1) GB9920917D0 (pt)
HK (1) HK1047093B (pt)
MX (1) MXPA02002355A (pt)
MY (1) MY125309A (pt)
PT (1) PT1214321E (pt)
SI (1) SI1214321T1 (pt)
TW (1) TWI274753B (pt)
WO (1) WO2001018002A1 (pt)
ZA (1) ZA200201781B (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2281817C (en) * 1999-06-29 2008-07-29 Smithkline Beecham Corporation Methods of use of fluoroquinolone compounds against maxillary sinus pathogenic bacteria
GB9920917D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel process
GB9920919D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel compound
DE60229255D1 (de) 2001-08-02 2008-11-20 Lg Life Sciences Ltd Verfahren zur herstellung von amino-geschützten 4-aminomethylene-pyrrolidin-3-on-derivaten, gemifloxacin und deren salze
KR100517638B1 (ko) * 2002-04-08 2005-09-28 주식회사 엘지생명과학 게미플록사신 산염의 새로운 제조방법
KR100653334B1 (ko) * 2003-03-07 2006-12-04 주식회사 엘지생명과학 4-아미노메틸-3-알콕시이미노피롤리딘 메탄설폰산염의 신규한 제조 방법
WO2006134431A1 (en) * 2005-05-03 2006-12-21 Ranbaxy Laboratories Limited Formate salt of gemifloxacin
US7834027B2 (en) 2005-06-15 2010-11-16 Hetero Drugs Limited Gemifloxacin process and polymorphs
US20100076193A1 (en) * 2006-10-31 2010-03-25 Chandrasekaran Ramasubbu process for the preparation of gemifloxacin

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57134482A (en) 1981-02-13 1982-08-19 Dainippon Pharmaceut Co Ltd 1-ethyl-6-fluoro-1,4-dihydro-4-oxo-7-(1-piperazinyl)-1,8- naphthyridine-3-carboxylic acid-3/2 hydrate and its preparation
IN162769B (pt) 1984-11-13 1988-07-09 Kyorin Seiyaku Kk
NZ222047A (en) 1986-10-08 1991-01-29 Bristol Myers Co Quinoline - or naphthyridine - carboxylic acid anti-bacterial agents
JPH01100165A (ja) 1987-10-13 1989-04-18 Shionogi & Co Ltd オキシムまたはヒドロキシアミン誘導体系抗菌剤
US4920120A (en) 1988-01-25 1990-04-24 Warner-Lambert Company Antibacterial agents
JPH0356479A (ja) 1989-07-24 1991-03-12 Takeshi Yokota 水溶性キノロン誘導体のｐ‐トルエンスルホン酸塩
WO1991002526A1 (en) 1989-08-16 1991-03-07 Pfizer Inc. Azabicyclo quinolone carboxylic acids
US5137892A (en) 1990-12-12 1992-08-11 Abbott Laboratories Quinoline, naphthyridine and pyridobenzoxazine derivatives
US5276041A (en) 1991-11-08 1994-01-04 Kaken Pharmaceutical Co., Ltd. Oxime derivatives
JPH0673056A (ja) 1992-08-26 1994-03-15 Kaken Pharmaceut Co Ltd キノリンカルボン酸誘導体およびその塩
EP0688772B1 (en) * 1994-06-16 1999-05-06 LG Chemical Limited Quinoline carboxylic acid derivatives having 7-(4-amino-methyl-3-oxime) pyrrolidine substituents and processes for their preparation
US5776944A (en) * 1994-06-16 1998-07-07 Lg Chemical Ltd. 7-(4-aminomethyl-3-methyloxyiminopyrroplidin-1-yl)-1-cyclopropyl-6-flu oro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid and the process for the preparation thereof
JP3449658B2 (ja) 1994-12-21 2003-09-22 杏林製薬株式会社 安定性に優れた８−アルコキシキノロンカルボン酸水和物並びにその製造方法
EP0789697B1 (en) 1995-06-06 1998-06-17 Pfizer Inc. CRYSTAL FORM OF ANHYDROUS 7-((1a,5a, 6a)-6-AMINO-3-AZABICYCLO ( 3.1. 0]HEX-3-YL)-6-FLUORO-1-(2,4-DIFLUOROPHENYL)-1,4-DIHYDRO-4-OXO-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID, METHANESULFONIC ACID SALT
DK0843661T3 (da) 1995-08-11 2002-07-22 Pfizer (1S,2S)-1-(4-hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)-1-propanolmethansulfonat-trihydrat
AU726694B2 (en) 1996-03-29 2000-11-16 Smithkline Beecham Corporation Eprosartan dihydrate and a process for its production and formulation
MA24500A1 (fr) * 1997-03-21 1998-10-01 Lg Life Sciences Ltd Derive du sel d'acide carboxylique de naphthyridine .
KR100286874B1 (ko) 1998-03-04 2001-04-16 성재갑 보호된 4-아미노메틸-피롤리딘-3-온의 제조방법
ES2207229T3 (es) 1998-05-29 2004-05-16 PHARMACIA & UPJOHN COMPANY Monometanosulfonato de 3-((1'-n-metilamino)etil-n-bencil)pirrolidina.
GB9820405D0 (en) 1998-09-18 1998-11-11 Smithkline Beecham Plc Process
ES2299430T3 (es) 1999-06-29 2008-06-01 Lg Life Sciences, Ltd. Utilizacion de compuestos de gemifloxacina contra bacterias.
JP2004507440A (ja) 1999-09-01 2004-03-11 スミスクライン・ビーチャム・コーポレイション 細菌に対するフルオロキノロン化合物の使用法
GB9920917D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel process
GB9920919D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel compound
EP1242079A4 (en) 1999-09-22 2003-01-22 Smithkline Beecham Methods of anti-bacterial use of fluoroquinolonic compounds
KR20010091379A (ko) 2000-03-15 2001-10-23 성재갑 7-(4-아미노메틸-3-옥심)피롤리딘 치환체를 갖는 퀴놀린카르복실산 유도체의 신규 제조방법
KR20020018560A (ko) 2000-09-01 2002-03-08 성재갑 3-아미노메틸-4-ｚ-메톡시이미노피롤리딘의 신규 제조방법

Also Published As

Publication number Publication date
US7232907B2 (en) 2007-06-19
SI1214321T1 (en) 2004-12-31
WO2001018002A1 (en) 2001-03-15
AU7019700A (en) 2001-04-10
ES2223574T3 (es) 2005-03-01
GB9920917D0 (en) 1999-11-10
ZA200201781B (en) 2003-06-25
DE60012196T2 (de) 2005-08-18
JP2003508532A (ja) 2003-03-04
HK1047093B (zh) 2005-05-27
KR100724311B1 (ko) 2007-06-04
BR0013751B1 (pt) 2013-02-05
CO5470281A1 (es) 2004-12-30
ATE271050T1 (de) 2004-07-15
AU773722B2 (en) 2004-06-03
MY125309A (en) 2006-07-31
JP4208464B2 (ja) 2009-01-14
DK1214321T3 (da) 2004-10-25
EP1214321A1 (en) 2002-06-19
EP1214321B1 (en) 2004-07-14
US20050176961A1 (en) 2005-08-11
KR20020041421A (ko) 2002-06-01
DE60012196D1 (de) 2004-08-19
PT1214321E (pt) 2004-10-29
CN1377350A (zh) 2002-10-30
CA2383753A1 (en) 2001-03-15
HK1047093A1 (en) 2003-02-07
AR029002A1 (es) 2003-06-04
BRPI0013751B8 (pt) 2021-05-25
MXPA02002355A (es) 2004-07-16
TWI274753B (en) 2007-03-01
CN1275963C (zh) 2006-09-20
CA2383753C (en) 2011-06-28

Similar Documents

Publication Publication Date Title
BR9900177A (pt) Inibidores de metaloprotease.
PT1177176E (pt) Derivados de acidos triarilicos como ligandos de receptores ppar.
BR0112693A (pt) (derivados) de ácido sulfonilaminometilbenzóico substituìdos e processo para preparação do mesmo
ES2122076T3 (es) Derivados de nor-acidos biliares, procedimiento para su preparacion y utilizacion de estos compuestos como medicamentos.
NO178969C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive, substituerte kinazolinoner
HUP0102465A3 (en) Process for the production of an aqueous monoester peroxycarboxylic acid solution, the solution obtainable by this process, and its use as disinfectant
EA200000826A1 (ru) Галоидированные производные амидиноаминокислот, применимые в качестве ингибиторов no-синтазы
ES2150808T3 (es) Forma cristalina de (4-trifluorometil)-anilida de acido 5-metilisoxazol-4-carboxilico.
YU94103A (sh) Novi derivati sulfonske kiseline
TR200201168T2 (tr) CGRP-Antagonistleri-yeni siklopropanlar içeren ilaçlar ve üretim yöntemleri.
FI98067B (fi) Uusia alkyleenidiammoniumdiklavulanaattijohdannaisia, menetelmä niidenvalmistamiseksi samoin kuin niiden käyttö kalvulaanihapon puhdistamiseksi
BR0013751A (pt) Processo para produção de derivados de ácido naftiridina-3-carboxìlico
EA200000204A1 (ru) Производные пирролопирролона в качестве ингибиторов эластазы нейтрофилов
ES2131313T3 (es) Derivados de acido nipecotico como compuestos antitromboticos.
BR9909898A (pt) Processo para purificação de um derivado de cefalosporina
BR9811855A (pt) Processo para preparação de ácido l-ascórbico
ES2178301T3 (es) Derivados del acido penicilanico 2-beta-sustituido-6-alquilideno como inhibidores de la beta-lactama.
BR0013750A (pt) Intermediários para a produção de derivados de ácido naftiridina-3-carboxìlico
PT1165485E (pt) Processo para a preparacao de produtos intermediarios pesticidas
PT1206452E (pt) Processo de preparacao de compostos benzoper-hidroisoindole
BR9907340A (pt) Ciclo-heptenos substituìdos, e processo para a produção de um composto
PT1133495E (pt) Semi-hidrocloreto do acido 8-ciano-1-ciclopropil-7-(1s,6s-2,8-diazabiciclo-¬4.3.0|-nonano-8-il)-6-fluoro-1,4-diidro-4-oxo-3-quinolinocarboxilico
ES2134971T3 (es) Derivado de acido octahidro-2-naftaleno-carboxilico, su produccion y uso.
PT818464E (pt) Metilsulfomicina i processo para a sua producao e utilizacao
CO5200841A1 (es) Derivados de bencimidazol sustituidos, procedimiento para su preparacion y su empleo como medicamentos

Legal Events

Date Code Title Description
B15G Petition not considered as such [chapter 15.7 patent gazette]

Free format text: DESCONHECIDAS AS PETICOES DE TRANSFERENCIA E ALTERACAO DE NOME NO 050668/RJ DE 12/09/2002 E 020040017093/RJ DE 15/12/2004, BEM COMO AS PETICOES DE ADITAMENTO NO 020050009719/RJ DE 14/02/2005 E 020050025961/RJ DE 15/04/2005, UMA VEZ QUE NAO FOI APRESENTADA A DOCUMENTACAO EXIGIDA PARA TAIS ATOS.

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 05/02/2013, OBSERVADAS AS CONDICOES LEGAIS.

B16C Correction of notification of the grant [chapter 16.3 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 01/09/2000 OBSERVADAS AS CONDICOES LEGAIS. PATENTE CONCEDIDA CONFORME ADI 5.529/DF

B21A Patent or certificate of addition expired [chapter 21.1 patent gazette]

Free format text: PATENTE EXTINTA EM 01/09/2020