BR9713087A - Composição farmacêutica estabilizada, utilização e processo para preparar a mesma, e, utilização de ácido metanossulfÈnico ou ácido clorìdrico - Google Patents

Composição farmacêutica estabilizada, utilização e processo para preparar a mesma, e, utilização de ácido metanossulfÈnico ou ácido clorìdrico

Info

Publication number
BR9713087A
BR9713087A BR9713087-7A BR9713087A BR9713087A BR 9713087 A BR9713087 A BR 9713087A BR 9713087 A BR9713087 A BR 9713087A BR 9713087 A BR9713087 A BR 9713087A
Authority
BR
Brazil
Prior art keywords
pharmaceutical composition
acid
prepare
stabilized pharmaceutical
hydrochloric acid
Prior art date
Application number
BR9713087-7A
Other languages
English (en)
Portuguese (pt)
Inventor
Jean-Paul Bounine
Guillaume Conrath
Original Assignee
Rh Ne Poulenc Rorer S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rh Ne Poulenc Rorer S A filed Critical Rh Ne Poulenc Rorer S A
Publication of BR9713087A publication Critical patent/BR9713087A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08Peptides having 5 to 11 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/20Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Inorganic Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BR9713087-7A 1996-11-19 1997-11-14 Composição farmacêutica estabilizada, utilização e processo para preparar a mesma, e, utilização de ácido metanossulfÈnico ou ácido clorìdrico BR9713087A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9614062A FR2755857B1 (fr) 1996-11-19 1996-11-19 Compositions pharmaceutiques stabilisees, a base de quinupristine et de dalfopristine et leur preparation
PCT/FR1997/002047 WO1998022107A1 (fr) 1996-11-19 1997-11-14 Compositions pharmaceutiques stabilisees, a base de quinupristine et de dalfopristine et leur preparation

Publications (1)

Publication Number Publication Date
BR9713087A true BR9713087A (pt) 2000-03-28

Family

ID=9497744

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9713087-7A BR9713087A (pt) 1996-11-19 1997-11-14 Composição farmacêutica estabilizada, utilização e processo para preparar a mesma, e, utilização de ácido metanossulfÈnico ou ácido clorìdrico

Country Status (45)

Country Link
US (1) US5994338A (de)
EP (1) EP0949923B1 (de)
JP (1) JP4278115B2 (de)
KR (1) KR100530836B1 (de)
CN (1) CN1146417C (de)
AP (1) AP998A (de)
AR (1) AR008695A1 (de)
AT (1) ATE223217T1 (de)
AU (1) AU740291B2 (de)
BG (1) BG63621B1 (de)
BR (1) BR9713087A (de)
CA (1) CA2271095C (de)
CO (1) CO4910113A1 (de)
CZ (1) CZ299913B6 (de)
DE (1) DE69715247T2 (de)
DK (1) DK0949923T3 (de)
DZ (1) DZ2349A1 (de)
EA (1) EA002025B1 (de)
EE (1) EE03668B1 (de)
ES (1) ES2179375T3 (de)
FR (1) FR2755857B1 (de)
HK (1) HK1022832A1 (de)
HR (1) HRP970615B1 (de)
HU (1) HUP9904327A3 (de)
IL (2) IL129607A0 (de)
IN (1) IN187038B (de)
JO (1) JO1992B1 (de)
MA (1) MA26448A1 (de)
MY (1) MY123805A (de)
NO (1) NO992399D0 (de)
NZ (1) NZ334949A (de)
OA (1) OA11047A (de)
PE (1) PE13999A1 (de)
PL (1) PL190164B1 (de)
PT (1) PT949923E (de)
RS (1) RS49608B (de)
SA (1) SA97180645B1 (de)
SK (1) SK284311B6 (de)
TN (1) TNSN97184A1 (de)
TR (1) TR199901096T2 (de)
TW (1) TW474816B (de)
UA (1) UA59376C2 (de)
UY (1) UY24780A1 (de)
WO (1) WO1998022107A1 (de)
ZA (1) ZA9710435B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2772272B1 (fr) * 1997-12-16 2000-01-14 Rhone Poulenc Rorer Sa Compositions pharmaceutiques a base de dalfopristine et de quinupristine et leur preparation
EP1115417B1 (de) * 1998-09-25 2006-04-05 Cubist Pharmaceuticals, Inc. Verwendung von daptomycin
CN100335122C (zh) * 1999-03-03 2007-09-05 伊莱利利公司 含有成胶束表面活性剂的棘白菌素药物制剂
TWI233805B (en) * 1999-07-01 2005-06-11 Fujisawa Pharmaceutical Co Stabilized pharmaceutical composition in lyophilized form as antifungal agent
US6119269A (en) * 1999-09-23 2000-09-19 Imler; Jack Fishing vest with removable storage container system
US6696412B1 (en) 2000-01-20 2004-02-24 Cubist Pharmaceuticals, Inc. High purity lipopeptides, Lipopeptide micelles and processes for preparing same
FR2812549B1 (fr) * 2000-08-03 2003-03-21 Aventis Pharma Sa Associations dalfopristine/quinupristine avec le cefpirome
US20060014674A1 (en) 2000-12-18 2006-01-19 Dennis Keith Methods for preparing purified lipopeptides

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2549065B1 (fr) * 1983-07-13 1985-10-25 Rhone Poulenc Sante Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2576022B1 (fr) * 1985-01-11 1987-09-11 Rhone Poulenc Sante Nouveaux derives de la pristinamycine ii b, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2599036B1 (fr) * 1986-05-22 1988-09-09 Rhone Poulenc Sante Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
CZ174899A3 (cs) 1999-08-11
BG63621B1 (bg) 2002-07-31
CA2271095C (fr) 2004-08-03
NZ334949A (en) 2000-12-22
TNSN97184A1 (fr) 2005-03-15
AP998A (en) 2001-08-09
IN187038B (de) 2001-12-29
NO992399L (no) 1999-05-19
JP2001504475A (ja) 2001-04-03
YU22499A (sh) 2002-03-18
ES2179375T3 (es) 2003-01-16
HRP970615B1 (en) 2002-12-31
WO1998022107A1 (fr) 1998-05-28
CO4910113A1 (es) 2000-04-24
PE13999A1 (es) 1999-05-05
DK0949923T3 (da) 2002-12-23
EA002025B1 (ru) 2001-12-24
US5994338A (en) 1999-11-30
DE69715247T2 (de) 2003-04-30
HK1022832A1 (en) 2000-08-25
EE03668B1 (et) 2002-04-15
HUP9904327A3 (en) 2002-03-28
PT949923E (pt) 2003-01-31
EP0949923A1 (de) 1999-10-20
CN1146417C (zh) 2004-04-21
DE69715247D1 (de) 2002-10-10
CZ299913B6 (cs) 2008-12-29
SK66099A3 (en) 2000-01-18
EE9900127A (et) 1999-12-15
SK284311B6 (sk) 2005-01-03
OA11047A (fr) 2003-03-07
KR100530836B1 (ko) 2005-11-23
EA199900479A1 (ru) 2000-02-28
AU5125698A (en) 1998-06-10
PL190164B1 (pl) 2005-11-30
ZA9710435B (en) 1998-06-10
IL129607A0 (en) 2000-02-29
NO992399D0 (no) 1999-05-19
AU740291B2 (en) 2001-11-01
BG103412A (en) 2000-06-30
CN1233959A (zh) 1999-11-03
HUP9904327A2 (hu) 2000-06-28
TW474816B (en) 2002-02-01
TR199901096T2 (xx) 1999-07-21
CA2271095A1 (fr) 1998-05-28
SA97180645B1 (ar) 2005-12-12
UA59376C2 (uk) 2003-09-15
EP0949923B1 (de) 2002-09-04
KR20000053343A (ko) 2000-08-25
JP4278115B2 (ja) 2009-06-10
DZ2349A1 (fr) 2002-12-28
AR008695A1 (es) 2000-02-09
UY24780A1 (es) 2001-08-27
MA26448A1 (fr) 2004-12-20
JO1992B1 (en) 1999-05-15
RS49608B (sr) 2007-06-04
HRP970615A2 (en) 1998-08-31
MY123805A (en) 2006-06-30
ATE223217T1 (de) 2002-09-15
FR2755857A1 (fr) 1998-05-22
IL129607A (en) 2006-08-20
FR2755857B1 (fr) 1998-12-24

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Legal Events

Date Code Title Description
B25D Requested change of name of applicant approved
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PRESENTE PEDIDO DE PATENTE DE ACORDO COM ART. 8O DA LPI.