BR9711948A - Composto processo para produzir um composto composi-Æo farmac-utica e uso de um composto - Google Patents

Composto processo para produzir um composto composi-Æo farmac-utica e uso de um composto

Info

Publication number
BR9711948A
BR9711948A BR9711948A BR9711948A BR9711948A BR 9711948 A BR9711948 A BR 9711948A BR 9711948 A BR9711948 A BR 9711948A BR 9711948 A BR9711948 A BR 9711948A BR 9711948 A BR9711948 A BR 9711948A
Authority
BR
Brazil
Prior art keywords
compound
pct
alkyl
different
same
Prior art date
Application number
BR9711948A
Other languages
English (en)
Inventor
William Alexander Denny
Swarnalatha Akuritaya Gamage
Julie Ann Spicer
Bruce Charles Baguley
Graeme John Finlay
Original Assignee
Xenova Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Xenova Ltd filed Critical Xenova Ltd
Publication of BR9711948A publication Critical patent/BR9711948A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/14Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
    • C07C227/18Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions involving amino or carboxyl groups, e.g. hydrolysis of esters or amides, by formation of halides, salts or esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D219/00Heterocyclic compounds containing acridine or hydrogenated acridine ring systems
    • C07D219/04Heterocyclic compounds containing acridine or hydrogenated acridine ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polishing Bodies And Polishing Tools (AREA)
  • Multicomponent Fibers (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Liquid Crystal (AREA)
BR9711948A 1996-10-18 1997-10-17 Composto processo para produzir um composto composi-Æo farmac-utica e uso de um composto BR9711948A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9621795.5A GB9621795D0 (en) 1996-10-18 1996-10-18 Pharmaceutical compounds
PCT/GB1997/002886 WO1998017650A1 (en) 1996-10-18 1997-10-17 Bis(acridinecarboxamide) and bis(phenazinecarboxamide) as antitumour agents

Publications (1)

Publication Number Publication Date
BR9711948A true BR9711948A (pt) 1999-08-24

Family

ID=10801674

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9711948A BR9711948A (pt) 1996-10-18 1997-10-17 Composto processo para produzir um composto composi-Æo farmac-utica e uso de um composto

Country Status (30)

Country Link
US (1) US6114332A (pt)
EP (1) EP0934278B1 (pt)
JP (1) JP2001503399A (pt)
KR (1) KR20000049252A (pt)
CN (1) CN1116285C (pt)
AT (1) ATE223381T1 (pt)
AU (1) AU717724B2 (pt)
BG (1) BG64555B1 (pt)
BR (1) BR9711948A (pt)
CA (1) CA2268411C (pt)
CZ (1) CZ295302B6 (pt)
DE (1) DE69715230T2 (pt)
DK (1) DK0934278T3 (pt)
ES (1) ES2183142T3 (pt)
GB (2) GB9621795D0 (pt)
HK (1) HK1018773A1 (pt)
HU (1) HU221953B1 (pt)
ID (1) ID22444A (pt)
MY (1) MY122017A (pt)
NO (1) NO313381B1 (pt)
NZ (1) NZ335055A (pt)
PL (1) PL193669B1 (pt)
PT (1) PT934278E (pt)
RO (1) RO120636B1 (pt)
RU (1) RU2179972C2 (pt)
SK (1) SK285121B6 (pt)
TW (1) TW432060B (pt)
UA (1) UA67729C2 (pt)
WO (1) WO1998017650A1 (pt)
ZA (2) ZA979331B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6974878B2 (en) 2001-03-21 2005-12-13 Symyx Technologies, Inc. Catalyst ligands, catalytic metal complexes and processes using same
EP1131283A1 (en) * 1999-09-10 2001-09-12 Symyx Technologies Catalyst ligands, catalytic metal complexes and processes using and methods of making same
GB2424884B (en) * 2003-12-31 2008-06-11 Council Scient Ind Res C-8 linked pyrrolo[2,1-c][1,4]benzodiazepine-acridone/acridine hybrids
EP3086791A4 (en) * 2013-12-24 2017-06-14 University of Florida Research Foundation, Inc. Phenazine derivatives as antimicrobial agents
CN104961801B (zh) * 2015-07-13 2018-01-19 兰州大学 一种具有多靶点的抗菌多肽偶联物及其二聚物的合成和应用
CN106554321B (zh) * 2015-09-25 2019-05-28 陆源 一种吩嗪类物质、其制备方法及其应用
KR20230087154A (ko) * 2021-12-09 2023-06-16 한국해양과학기술원 신규 다이페나진 화합물 및 이의 암 또는 신경염증질환 예방 또는 치료 용도

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ201084A (en) * 1982-06-25 1985-10-11 New Zealand Dev Finance 4-carboxamidoacridine derivatives and pharmaceutical compositions containing such
EP0172744A2 (en) * 1984-08-16 1986-02-26 Development Finance Corporation Of New Zealand Phenazinecarboxamide compounds
IT1293525B1 (it) * 1997-08-01 1999-03-01 Uni Degli Studi Camerino Bis-acridincarbossiammidi aventi attivita' antitumorale

Also Published As

Publication number Publication date
NO991833L (no) 1999-06-03
ATE223381T1 (de) 2002-09-15
JP2001503399A (ja) 2001-03-13
GB2334032B (en) 2000-11-08
CZ127199A3 (cs) 1999-09-15
NO991833D0 (no) 1999-04-16
GB9621795D0 (en) 1996-12-11
GB2334032A (en) 1999-08-11
CN1116285C (zh) 2003-07-30
DK0934278T3 (da) 2003-01-06
HK1018773A1 (en) 2000-01-07
CA2268411C (en) 2008-07-22
PL193669B1 (pl) 2007-03-30
ZA979331B (en) 1998-05-21
TW432060B (en) 2001-05-01
RU2179972C2 (ru) 2002-02-27
US6114332A (en) 2000-09-05
KR20000049252A (ko) 2000-07-25
AU717724B2 (en) 2000-03-30
HU221953B1 (hu) 2003-03-28
HUP9902883A3 (en) 2001-01-29
CA2268411A1 (en) 1998-04-30
SK50499A3 (en) 2000-05-16
NZ335055A (en) 2000-09-29
MY122017A (en) 2006-03-31
ES2183142T3 (es) 2003-03-16
DE69715230D1 (de) 2002-10-10
BG64555B1 (bg) 2005-07-29
WO1998017650A1 (en) 1998-04-30
SK285121B6 (sk) 2006-06-01
BG103329A (en) 2000-11-30
CN1240430A (zh) 2000-01-05
PT934278E (pt) 2003-01-31
NO313381B1 (no) 2002-09-23
RO120636B1 (ro) 2006-05-30
DE69715230T2 (de) 2009-09-17
EP0934278B1 (en) 2002-09-04
GB9908192D0 (en) 1999-06-02
EP0934278A1 (en) 1999-08-11
CZ295302B6 (cs) 2005-07-13
ZA979328B (en) 1998-07-06
AU4713797A (en) 1998-05-15
ID22444A (id) 1999-10-14
UA67729C2 (uk) 2004-07-15
PL332877A1 (en) 1999-10-25

Similar Documents

Publication Publication Date Title
HUP0004076A2 (hu) C-4"-Szubsztituált-makrolid-származékok
HUP9802694A1 (hu) Benzamidszármazékok, eljárás előállításukra és ezeket tartalmazó gyógyszerkészítmények
CA2054619A1 (en) Aminocoumaran derivatives, their production and use
MX9504287A (es) Derivados de camptotecina y proceso para su preparacion.
HRP20070194T3 (en) N-thiazol-2-yl-benzamide derivatives
EP0353955A3 (en) Novel compounds
EP0765865A4 (en) 2-ACYLAMINOPROPANOL COMPOUND AND MEDICINAL COMPOSITION
ES2177656T3 (es) Derivados de antraciclinona y su utilizacion en el tratamiento de la amiloidosis.
BR9711948A (pt) Composto processo para produzir um composto composi-Æo farmac-utica e uso de um composto
DE68926981D1 (de) Cephemverbindungen und Verfahren zu ihrer Herstellung
HUP0203275A2 (hu) 1-(Gyűrűs amino)-alkilciklohexán-származékok, ezeket tartalmazó görcsoldó hatású gyógyszerkészítmények, valamint ezek alkalmazása
ES472290A1 (es) Un procedimiento para preparar un compuesto de benceno di- sustituido en orto
PT92540A (pt) Processo para a preparacao de derivados de anfotericina b
DE69330601T2 (de) Serotoninergische ergolin derivate
ES2103131T3 (es) Nuevos agentes de nucleosido carbociclico utiles como inhibidores selectivos de citoquinas proinflamatorias.
ES2002036A6 (es) Un procedimiento para la preparacion de derivados de dicloroanilina.
RU99109978A (ru) Бис(акридинкарбоксамид) и бис(феназинкарбоксамид), полезные в качестве противоопухолевых агентов
IL115085A0 (en) Bicyclic carboxamide derivatives their preparation and pharmaceutical compositions containing them
RU96120092A (ru) Новые производные пиперазина и способы их получения и содержащие их композиции
RU92004544A (ru) Замещенные производные бензоилмочевины, способ их получения, противоопухолевая композиция и способ лечения
PT89483A (pt) Processo para a preparacao de derivados da 2-amino acetamida
TH18165A (th) สารยับยั้งการเกิดคีโมแทกซิของอีโอซีโนฟีล
KR940014381A (ko) 신규한 퀴놀론계 화합물 및 그의 제조방법

Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PRESENTE PEDIDO DE PATENTE DE ACORDO COM ART. 36 DA LPI