BR112015020823A2 - 1-hidróxi-benzooxaboróis como agentes antiparasíticos - Google Patents

1-hidróxi-benzooxaboróis como agentes antiparasíticos

Info

Publication number
BR112015020823A2
BR112015020823A2 BR112015020823A BR112015020823A BR112015020823A2 BR 112015020823 A2 BR112015020823 A2 BR 112015020823A2 BR 112015020823 A BR112015020823 A BR 112015020823A BR 112015020823 A BR112015020823 A BR 112015020823A BR 112015020823 A2 BR112015020823 A2 BR 112015020823A2
Authority
BR
Brazil
Prior art keywords
benzooxaborols
hydroxy
control
antiparasitic agents
compounds
Prior art date
Application number
BR112015020823A
Other languages
English (en)
Other versions
BR112015020823A8 (pt
Inventor
J Plattner Jacob
Jarnagin Kurt
Roland Pulley Shon
Akama Tsutomu
Hunter White William
Zhou Yasheen
Zhang Yong-Kang
Original Assignee
Anacor Pharmaceuticals Inc
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anacor Pharmaceuticals Inc, Lilly Co Eli filed Critical Anacor Pharmaceuticals Inc
Publication of BR112015020823A2 publication Critical patent/BR112015020823A2/pt
Publication of BR112015020823A8 publication Critical patent/BR112015020823A8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epidemiology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)

Abstract

resumo patente de invenção: "1-hidróxi-benzooxaboróis como agentes antiparasíticos". são fornecidos compostos úteis para o controle de endoparasitas tanto em animais quanto em agricultura. são também fornecidos métodos para o controle de infestações por endoparasita de um animal administrando uma quantidade efetiva de um composto como descrito acima, ou um sal farmaceuticamente aceitável do mesmo, a um animal, bem como formulações para o controle de infestações por endoparasita, usando os compostos descritos acima ou um sal aceitável do mesmo, e um veículo aceitável. os compostos reivindicados são descritos pela seguinte fórmula markush: um exemplo típico para um composto de acordo com a fórmula acima é:
BR112015020823A 2013-03-15 2014-03-06 1-hidróxi-benzooxaboróis como agentes antiparasíticos, seus usos, e formulação". BR112015020823A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361786839P 2013-03-15 2013-03-15
PCT/US2014/020966 WO2014149793A1 (en) 2013-03-15 2014-03-06 1 -hydroxy-benzooxaboroles as antiparasitic agents

Publications (2)

Publication Number Publication Date
BR112015020823A2 true BR112015020823A2 (pt) 2017-07-18
BR112015020823A8 BR112015020823A8 (pt) 2019-09-17

Family

ID=50382679

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015020823A BR112015020823A8 (pt) 2013-03-15 2014-03-06 1-hidróxi-benzooxaboróis como agentes antiparasíticos, seus usos, e formulação".

Country Status (24)

Country Link
US (1) US9617285B2 (pt)
EP (1) EP2970339B1 (pt)
JP (1) JP6121043B2 (pt)
KR (1) KR101727421B1 (pt)
CN (1) CN105051048B (pt)
AR (1) AR094961A1 (pt)
AU (1) AU2014237862B2 (pt)
BR (1) BR112015020823A8 (pt)
CA (1) CA2899972A1 (pt)
CY (1) CY1119473T1 (pt)
DK (1) DK2970339T3 (pt)
EA (1) EA027430B1 (pt)
ES (1) ES2645687T3 (pt)
HR (1) HRP20171517T1 (pt)
HU (1) HUE035545T2 (pt)
LT (1) LT2970339T (pt)
MX (1) MX2015013051A (pt)
NO (1) NO2904426T3 (pt)
PL (1) PL2970339T3 (pt)
PT (1) PT2970339T (pt)
RS (1) RS56532B1 (pt)
SI (1) SI2970339T1 (pt)
TW (1) TW201506031A (pt)
WO (1) WO2014149793A1 (pt)

Families Citing this family (14)

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US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
EP3164404B1 (en) 2014-07-01 2019-04-03 Daiichi Sankyo Company, Limited Tricyclic benzoxaboroles as antibacterial agents
CA3015662A1 (en) 2016-03-07 2017-09-14 Agrofresh Inc. Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops
AU2017275599B2 (en) 2016-06-03 2021-09-02 Basf Se Benzoxaborole compounds
WO2018156554A1 (en) * 2017-02-21 2018-08-30 Dow Agrosciences Llc 1-HYDROXY-1,3-DIHYDROBENZO[c][1,2]OXABOROLES AND THEIR USE AS HERBICIDES
CN108864160A (zh) * 2017-05-16 2018-11-23 苏州旺山旺水生物医药有限公司 含硼小分子的制备方法
WO2019025250A1 (en) 2017-08-04 2019-02-07 Basf Se SUBSTITUTED TRIFLUOROMETHYLOXADIAZOLES FOR COMBATING PHYTOPATHOGENIC FUNGI
US11834466B2 (en) 2017-11-30 2023-12-05 5Metis, Inc. Benzoxaborole compounds and formulations thereof
CA3148168A1 (en) 2018-08-18 2020-02-27 Chun Yu Liu Solid forms of substituted benzoxaborole and compositions thereof
EP4204012A1 (en) 2020-08-31 2023-07-05 Pfizer Inc. Methods of protecting rna
CN112321510A (zh) * 2020-10-27 2021-02-05 无锡双启科技有限公司 一种4-溴-5-甲基-1h-吲唑的制备方法
CN112745270B (zh) * 2020-12-30 2023-02-24 河北医科大学 新化合物及其制备苯唑草酮中间体的方法
EP4137485A1 (en) * 2021-08-20 2023-02-22 Henkel AG & Co. KGaA Vinyl ethers

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US6239077B1 (en) 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
NZ526538A (en) 2000-12-20 2005-12-23 Novartis Ag Anti-endoparasitic amidoacetonitrils
AR035531A1 (es) 2001-01-22 2004-06-02 Novartis Ag Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos
TWI236341B (en) 2001-06-15 2005-07-21 Novartis Ag Aminoacetonitrile compounds for use in the control of endoparasites
AR038156A1 (es) 2002-01-21 2004-12-29 Novartis Ag Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica
TW200305556A (en) 2002-03-21 2003-11-01 Novartis Ag Organic compounds
AR040082A1 (es) 2002-05-22 2005-03-16 Novartis Ag Derivados de n-acilaminoacetonitrilo y su uso para el control de parasitos
TW200400931A (en) 2002-05-22 2004-01-16 Novartis Ag Organic compounds
AR039961A1 (es) 2002-06-06 2005-03-09 Novartis Ag Derivados de amidoacetonitrilo y su uso como pesticida
TW200400932A (en) 2002-06-19 2004-01-16 Novartis Ag Organic compounds
GB0402677D0 (en) 2003-11-06 2004-03-10 Novartis Ag Organic compounds
AR046757A1 (es) 2003-12-10 2005-12-21 Novartis Ag Amidoacetonitrilos utiles como pesticidas
AR049391A1 (es) 2004-06-10 2006-07-26 Novartis Ag Derivados de aminoacetonitrilo y su uso para controlar parasitos en animales de sangre caliente
NZ560448A (en) 2005-02-16 2009-08-28 Anacor Pharmaceuticals Inc Boron-containing small molecules
EP1910278A1 (en) 2005-07-25 2008-04-16 Novartis AG Amidonitrile compounds
CN106008571A (zh) 2005-12-30 2016-10-12 安纳考尔医药公司 含硼的小分子
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Also Published As

Publication number Publication date
MX2015013051A (es) 2016-05-05
HUE035545T2 (en) 2018-05-28
TW201506031A (zh) 2015-02-16
CA2899972A1 (en) 2014-09-25
KR101727421B1 (ko) 2017-04-14
EP2970339A1 (en) 2016-01-20
KR20150119154A (ko) 2015-10-23
DK2970339T3 (en) 2017-10-02
WO2014149793A1 (en) 2014-09-25
PT2970339T (pt) 2017-11-14
US9617285B2 (en) 2017-04-11
PL2970339T3 (pl) 2018-01-31
ES2645687T3 (es) 2017-12-07
AR094961A1 (es) 2015-09-09
CN105051048A (zh) 2015-11-11
EP2970339B1 (en) 2017-08-16
US20150353581A1 (en) 2015-12-10
LT2970339T (lt) 2017-11-10
SI2970339T1 (sl) 2017-10-30
JP2016516032A (ja) 2016-06-02
JP6121043B2 (ja) 2017-04-26
EA201591512A9 (ru) 2016-04-29
CN105051048B (zh) 2017-03-15
EA201591512A1 (ru) 2016-01-29
HRP20171517T1 (hr) 2017-11-17
AU2014237862B2 (en) 2017-01-12
BR112015020823A8 (pt) 2019-09-17
RS56532B1 (sr) 2018-02-28
EA027430B1 (ru) 2017-07-31
CY1119473T1 (el) 2018-03-07
NO2904426T3 (pt) 2018-02-10
AU2014237862A1 (en) 2015-08-13

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Legal Events

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B06F Objections, documents and/or translations needed after an examination request according art. 34 industrial property law
B07D Technical examination (opinion) related to article 229 of industrial property law

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B08F Application fees: dismissal - article 86 of industrial property law

Free format text: REFERENTE A 6A ANUIDADE.

B08K Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87)

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2556 DE 31/12/2019.

B07E Notice of approval relating to section 229 industrial property law