BR112015020823A2 - 1-hidróxi-benzooxaboróis como agentes antiparasíticos - Google Patents
1-hidróxi-benzooxaboróis como agentes antiparasíticosInfo
- Publication number
- BR112015020823A2 BR112015020823A2 BR112015020823A BR112015020823A BR112015020823A2 BR 112015020823 A2 BR112015020823 A2 BR 112015020823A2 BR 112015020823 A BR112015020823 A BR 112015020823A BR 112015020823 A BR112015020823 A BR 112015020823A BR 112015020823 A2 BR112015020823 A2 BR 112015020823A2
- Authority
- BR
- Brazil
- Prior art keywords
- benzooxaborols
- hydroxy
- control
- antiparasitic agents
- compounds
- Prior art date
Links
- 239000003096 antiparasitic agent Substances 0.000 title abstract 2
- 229940125687 antiparasitic agent Drugs 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 5
- 241001465754 Metazoa Species 0.000 abstract 3
- 244000079386 endoparasite Species 0.000 abstract 3
- 206010061217 Infestation Diseases 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 238000009472 formulation Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
- A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Dentistry (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Tropical Medicine & Parasitology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epidemiology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
resumo patente de invenção: "1-hidróxi-benzooxaboróis como agentes antiparasíticos". são fornecidos compostos úteis para o controle de endoparasitas tanto em animais quanto em agricultura. são também fornecidos métodos para o controle de infestações por endoparasita de um animal administrando uma quantidade efetiva de um composto como descrito acima, ou um sal farmaceuticamente aceitável do mesmo, a um animal, bem como formulações para o controle de infestações por endoparasita, usando os compostos descritos acima ou um sal aceitável do mesmo, e um veículo aceitável. os compostos reivindicados são descritos pela seguinte fórmula markush: um exemplo típico para um composto de acordo com a fórmula acima é:
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361786839P | 2013-03-15 | 2013-03-15 | |
| PCT/US2014/020966 WO2014149793A1 (en) | 2013-03-15 | 2014-03-06 | 1 -hydroxy-benzooxaboroles as antiparasitic agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BR112015020823A2 true BR112015020823A2 (pt) | 2017-07-18 |
| BR112015020823A8 BR112015020823A8 (pt) | 2019-09-17 |
Family
ID=50382679
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112015020823A BR112015020823A8 (pt) | 2013-03-15 | 2014-03-06 | 1-hidróxi-benzooxaboróis como agentes antiparasíticos, seus usos, e formulação". |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US9617285B2 (pt) |
| EP (1) | EP2970339B1 (pt) |
| JP (1) | JP6121043B2 (pt) |
| KR (1) | KR101727421B1 (pt) |
| CN (1) | CN105051048B (pt) |
| AR (1) | AR094961A1 (pt) |
| AU (1) | AU2014237862B2 (pt) |
| BR (1) | BR112015020823A8 (pt) |
| CA (1) | CA2899972A1 (pt) |
| CY (1) | CY1119473T1 (pt) |
| DK (1) | DK2970339T3 (pt) |
| EA (1) | EA027430B1 (pt) |
| ES (1) | ES2645687T3 (pt) |
| HR (1) | HRP20171517T1 (pt) |
| HU (1) | HUE035545T2 (pt) |
| LT (1) | LT2970339T (pt) |
| MX (1) | MX2015013051A (pt) |
| NO (1) | NO2904426T3 (pt) |
| PL (1) | PL2970339T3 (pt) |
| PT (1) | PT2970339T (pt) |
| RS (1) | RS56532B1 (pt) |
| SI (1) | SI2970339T1 (pt) |
| TW (1) | TW201506031A (pt) |
| WO (1) | WO2014149793A1 (pt) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
| US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
| KR20170024068A (ko) | 2014-07-01 | 2017-03-06 | 다이이찌 산쿄 가부시키가이샤 | 항박테리아제로서의 삼환식 벤즈옥사보롤 |
| TW201735792A (zh) | 2016-03-07 | 2017-10-16 | 農業保鮮股份有限公司 | 使用苯并氧雜硼雜環戊烯化合物和防腐氣體作為作物的抗微生物劑之協同方法 |
| UA122609C2 (uk) | 2016-06-03 | 2020-12-10 | Басф Се | Сполуки бензоксаборолу |
| WO2018156554A1 (en) * | 2017-02-21 | 2018-08-30 | Dow Agrosciences Llc | 1-HYDROXY-1,3-DIHYDROBENZO[c][1,2]OXABOROLES AND THEIR USE AS HERBICIDES |
| CN108864160A (zh) * | 2017-05-16 | 2018-11-23 | 苏州旺山旺水生物医药有限公司 | 含硼小分子的制备方法 |
| WO2019025250A1 (en) | 2017-08-04 | 2019-02-07 | Basf Se | SUBSTITUTED TRIFLUOROMETHYLOXADIAZOLES FOR COMBATING PHYTOPATHOGENIC FUNGI |
| WO2019108982A1 (en) | 2017-11-30 | 2019-06-06 | Boragen, Inc. | Benzoxaborole compounds and formulations thereof |
| EP3836938A4 (en) | 2018-08-18 | 2022-05-11 | Boragen, Inc. | SOLID FORMS OF SUBSTITUTED BENZOXAZOLE AND COMPOSITIONS THEREOF |
| EP4204012A1 (en) | 2020-08-31 | 2023-07-05 | Pfizer Inc. | Methods of protecting rna |
| CN112321510A (zh) * | 2020-10-27 | 2021-02-05 | 无锡双启科技有限公司 | 一种4-溴-5-甲基-1h-吲唑的制备方法 |
| CN112745270B (zh) * | 2020-12-30 | 2023-02-24 | 河北医科大学 | 新化合物及其制备苯唑草酮中间体的方法 |
| EP4137485A1 (en) * | 2021-08-20 | 2023-02-22 | Henkel AG & Co. KGaA | Vinyl ethers |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6239077B1 (en) | 1998-05-01 | 2001-05-29 | Nihon Nohyaku Co., Ltd. | Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof |
| TWI292712B (en) | 2000-12-20 | 2008-01-21 | Novartis Ag | Aminoacetonitrile compounds for use in the control of endoparasites |
| AR035531A1 (es) | 2001-01-22 | 2004-06-02 | Novartis Ag | Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos |
| AR036054A1 (es) | 2001-06-15 | 2004-08-04 | Novartis Ag | Uso de compuestos de aminoacetonitrilo para el control de plagas, una composicion y un proceso para dicho control y una composicion farmaceutica contra parasitos |
| AR038156A1 (es) | 2002-01-21 | 2004-12-29 | Novartis Ag | Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica |
| AR039020A1 (es) | 2002-03-21 | 2005-02-02 | Novartis Ag | Compuestos de aminoacetonitrilo |
| AR040082A1 (es) | 2002-05-22 | 2005-03-16 | Novartis Ag | Derivados de n-acilaminoacetonitrilo y su uso para el control de parasitos |
| TW200400931A (en) | 2002-05-22 | 2004-01-16 | Novartis Ag | Organic compounds |
| AR039961A1 (es) | 2002-06-06 | 2005-03-09 | Novartis Ag | Derivados de amidoacetonitrilo y su uso como pesticida |
| TW200400932A (en) | 2002-06-19 | 2004-01-16 | Novartis Ag | Organic compounds |
| GB0402677D0 (en) | 2003-11-06 | 2004-03-10 | Novartis Ag | Organic compounds |
| AR046757A1 (es) | 2003-12-10 | 2005-12-21 | Novartis Ag | Amidoacetonitrilos utiles como pesticidas |
| TW200613251A (en) | 2004-06-10 | 2006-05-01 | Novartis Ag | Organic compounds |
| US7767657B2 (en) | 2005-02-16 | 2010-08-03 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| EP2987796B1 (en) | 2005-02-16 | 2018-08-08 | Anacor Pharmaceuticals, Inc. | Halogen-substituted boronophthalides for the treatment of infections |
| JP2009502834A (ja) | 2005-07-25 | 2009-01-29 | ノバルティス アクチエンゲゼルシャフト | アミドニトリル化合物 |
| CA2678149C (en) | 2007-02-21 | 2013-04-16 | Pfizer Limited | Benzofuran antiparasitic agents |
| US20100026457A1 (en) * | 2008-08-04 | 2010-02-04 | Cooper Technologies Company | Location of Tagged Boxes |
| EP2358687B9 (en) | 2008-10-21 | 2013-04-17 | Merial Ltd. | Thioamide compounds, method of making and method of using thereof |
| BR112012001987A2 (pt) | 2009-07-28 | 2015-09-01 | Anacor Pharmaceuticals Inc | Composto, combinação, formulação farmacêutica, uso de um composto, uma combinação ou um sal farmaceuticamente aceitável dos mesmos, e, métodos para tratar uma infecção bacteriana, para matar ou inibir o crescimento de uma bactéria, e para inibir uma beta-lactamase. |
| WO2011019612A1 (en) * | 2009-08-14 | 2011-02-17 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| WO2011049971A1 (en) * | 2009-10-20 | 2011-04-28 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| EP2314292A1 (en) | 2009-10-20 | 2011-04-27 | Novartis AG | Endoparasiticidal compositions |
| UY32992A (es) | 2009-11-23 | 2011-04-29 | Novartis Ag | Compuestos orgánicos |
| HRP20220384T1 (hr) * | 2013-08-09 | 2022-07-22 | Glaxosmithkline Intellectual Property (No. 2) Limited | Triciklički benzoksaborol spojevi i njihove uporabe |
-
2014
- 2014-02-28 AR ARP140100676A patent/AR094961A1/es unknown
- 2014-03-06 CN CN201480014758.9A patent/CN105051048B/zh not_active Expired - Fee Related
- 2014-03-06 RS RS20171064A patent/RS56532B1/sr unknown
- 2014-03-06 JP JP2016500695A patent/JP6121043B2/ja active Active
- 2014-03-06 DK DK14712939.9T patent/DK2970339T3/en active
- 2014-03-06 ES ES14712939.9T patent/ES2645687T3/es active Active
- 2014-03-06 PT PT147129399T patent/PT2970339T/pt unknown
- 2014-03-06 SI SI201430345T patent/SI2970339T1/sl unknown
- 2014-03-06 LT LTEP14712939.9T patent/LT2970339T/lt unknown
- 2014-03-06 MX MX2015013051A patent/MX2015013051A/es unknown
- 2014-03-06 KR KR1020157024782A patent/KR101727421B1/ko active IP Right Grant
- 2014-03-06 AU AU2014237862A patent/AU2014237862B2/en not_active Ceased
- 2014-03-06 CA CA2899972A patent/CA2899972A1/en not_active Abandoned
- 2014-03-06 BR BR112015020823A patent/BR112015020823A8/pt active Search and Examination
- 2014-03-06 HU HUE14712939A patent/HUE035545T2/en unknown
- 2014-03-06 US US14/760,208 patent/US9617285B2/en not_active Expired - Fee Related
- 2014-03-06 TW TW103107747A patent/TW201506031A/zh unknown
- 2014-03-06 WO PCT/US2014/020966 patent/WO2014149793A1/en active Application Filing
- 2014-03-06 PL PL14712939T patent/PL2970339T3/pl unknown
- 2014-03-06 EP EP14712939.9A patent/EP2970339B1/en active Active
- 2014-03-06 EA EA201591512A patent/EA027430B1/ru not_active IP Right Cessation
- 2014-11-18 NO NO14799476A patent/NO2904426T3/no unknown
-
2017
- 2017-10-09 HR HRP20171517TT patent/HRP20171517T1/hr unknown
- 2017-10-20 CY CY20171101096T patent/CY1119473T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| SI2970339T1 (sl) | 2017-10-30 |
| JP6121043B2 (ja) | 2017-04-26 |
| EA201591512A9 (ru) | 2016-04-29 |
| CN105051048B (zh) | 2017-03-15 |
| RS56532B1 (sr) | 2018-02-28 |
| PL2970339T3 (pl) | 2018-01-31 |
| EP2970339A1 (en) | 2016-01-20 |
| MX2015013051A (es) | 2016-05-05 |
| BR112015020823A8 (pt) | 2019-09-17 |
| NO2904426T3 (pt) | 2018-02-10 |
| EA027430B1 (ru) | 2017-07-31 |
| EA201591512A1 (ru) | 2016-01-29 |
| CA2899972A1 (en) | 2014-09-25 |
| CN105051048A (zh) | 2015-11-11 |
| KR20150119154A (ko) | 2015-10-23 |
| LT2970339T (lt) | 2017-11-10 |
| AR094961A1 (es) | 2015-09-09 |
| TW201506031A (zh) | 2015-02-16 |
| KR101727421B1 (ko) | 2017-04-14 |
| DK2970339T3 (en) | 2017-10-02 |
| CY1119473T1 (el) | 2018-03-07 |
| HRP20171517T1 (hr) | 2017-11-17 |
| WO2014149793A1 (en) | 2014-09-25 |
| AU2014237862A1 (en) | 2015-08-13 |
| JP2016516032A (ja) | 2016-06-02 |
| US9617285B2 (en) | 2017-04-11 |
| US20150353581A1 (en) | 2015-12-10 |
| PT2970339T (pt) | 2017-11-14 |
| ES2645687T3 (es) | 2017-12-07 |
| AU2014237862B2 (en) | 2017-01-12 |
| HUE035545T2 (en) | 2018-05-28 |
| EP2970339B1 (en) | 2017-08-16 |
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Legal Events
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| B06F | Objections, documents and/or translations needed after an examination request according art. 34 industrial property law | ||
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Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS. |
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| B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTE A 6A ANUIDADE. |
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| B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2556 DE 31/12/2019. |
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| B07E | Notice of approval relating to section 229 industrial property law |