CY1119473T1 - 1-υδροξυ-βενζοοξαβορολια ως αντιπαρασιτικοι παραγοντες - Google Patents
1-υδροξυ-βενζοοξαβορολια ως αντιπαρασιτικοι παραγοντεςInfo
- Publication number
- CY1119473T1 CY1119473T1 CY20171101096T CY171101096T CY1119473T1 CY 1119473 T1 CY1119473 T1 CY 1119473T1 CY 20171101096 T CY20171101096 T CY 20171101096T CY 171101096 T CY171101096 T CY 171101096T CY 1119473 T1 CY1119473 T1 CY 1119473T1
- Authority
- CY
- Cyprus
- Prior art keywords
- benzoxavorola
- hydroxy
- compounds
- intra
- animal
- Prior art date
Links
- 230000002141 anti-parasite Effects 0.000 title 1
- 239000003096 antiparasitic agent Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 6
- 241001465754 Metazoa Species 0.000 abstract 3
- 150000003839 salts Chemical class 0.000 abstract 2
- 244000079386 endoparasite Species 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
- A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Dentistry (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Tropical Medicine & Parasitology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Epidemiology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Steroid Compounds (AREA)
Abstract
Εδώ παρέχονται ενώσεις χρήσιμες για την καταπολέμηση ενδοπαρασίτων και σε ζώα και στη γεωργία. Περαιτέρω παρέχονται μέθοδοι για την καταπολέμηση ενδοπαρασιτικών προσβολών ενός ζώου διά της χορήγησης μιας αποτελεσματικής ποσότητας μιας ένωσης όπως περιγράφεται παραπάνω, ή ενός φαρμακευτικώς αποδεκτού άλατος αυτής, σε ένα ζώο, καθώς και σκευάσματα για την καταπολέμηση ενδοπαρασιτικών προσβολών με τη χρησιμοποίηση των ενώσεων που περιγράφονται παραπάνω ή ενός αποδεκτού άλατος αυτών, και ενός αποδεκτού φορέα. Οι αξιούμενες ενώσεις περιγράφονται διά του ακόλουθου τύπου Markush: Ένα τυπικό παράδειγμα για μια ένωση σύμφωνα με τον παραπάνω τύπο είναι: Ένα τυπικό παράδειγμα για μια ένωση σύμφωνα με τον παραπάνω τύπο είναι:
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361786839P | 2013-03-15 | 2013-03-15 | |
| PCT/US2014/020966 WO2014149793A1 (en) | 2013-03-15 | 2014-03-06 | 1 -hydroxy-benzooxaboroles as antiparasitic agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CY1119473T1 true CY1119473T1 (el) | 2018-03-07 |
Family
ID=50382679
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CY20171101096T CY1119473T1 (el) | 2013-03-15 | 2017-10-20 | 1-υδροξυ-βενζοοξαβορολια ως αντιπαρασιτικοι παραγοντες |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US9617285B2 (el) |
| EP (1) | EP2970339B1 (el) |
| JP (1) | JP6121043B2 (el) |
| KR (1) | KR101727421B1 (el) |
| CN (1) | CN105051048B (el) |
| AR (1) | AR094961A1 (el) |
| AU (1) | AU2014237862B2 (el) |
| BR (1) | BR112015020823A8 (el) |
| CA (1) | CA2899972A1 (el) |
| CY (1) | CY1119473T1 (el) |
| DK (1) | DK2970339T3 (el) |
| EA (1) | EA027430B1 (el) |
| ES (1) | ES2645687T3 (el) |
| HR (1) | HRP20171517T1 (el) |
| HU (1) | HUE035545T2 (el) |
| LT (1) | LT2970339T (el) |
| MX (1) | MX2015013051A (el) |
| NO (1) | NO2904426T3 (el) |
| PL (1) | PL2970339T3 (el) |
| PT (1) | PT2970339T (el) |
| RS (1) | RS56532B1 (el) |
| SI (1) | SI2970339T1 (el) |
| TW (1) | TW201506031A (el) |
| WO (1) | WO2014149793A1 (el) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
| US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
| CA2953881A1 (en) | 2014-07-01 | 2016-01-07 | Daiichi Sankyo Company, Limited | Tricyclic benzoxaboroles as antibacterial agents |
| EP3426029B1 (en) | 2016-03-07 | 2023-08-30 | AgroFresh Inc. | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
| CA3026316A1 (en) | 2016-06-03 | 2017-12-07 | Basf Se | Benzoxaborole compounds |
| WO2018156554A1 (en) * | 2017-02-21 | 2018-08-30 | Dow Agrosciences Llc | 1-HYDROXY-1,3-DIHYDROBENZO[c][1,2]OXABOROLES AND THEIR USE AS HERBICIDES |
| CN108864160A (zh) * | 2017-05-16 | 2018-11-23 | 苏州旺山旺水生物医药有限公司 | 含硼小分子的制备方法 |
| WO2019025250A1 (en) | 2017-08-04 | 2019-02-07 | Basf Se | SUBSTITUTED TRIFLUOROMETHYLOXADIAZOLES FOR COMBATING PHYTOPATHOGENIC FUNGI |
| BR112020010927A2 (pt) | 2017-11-30 | 2020-12-01 | Boragen, Inc. | compostos de benzoxaborol e formulações dos mesmos |
| JP2021534247A (ja) | 2018-08-18 | 2021-12-09 | ボラゲン，インコーポレーテッド | 置換ベンゾキサボロールの固体形態およびその組成物 |
| US20230340530A1 (en) | 2020-08-31 | 2023-10-26 | Pfizer Inc. | Methods of Protecting RNA |
| CN112321510A (zh) * | 2020-10-27 | 2021-02-05 | 无锡双启科技有限公司 | 一种4-溴-5-甲基-1h-吲唑的制备方法 |
| CN112745270B (zh) * | 2020-12-30 | 2023-02-24 | 河北医科大学 | 新化合物及其制备苯唑草酮中间体的方法 |
| EP4137485A1 (en) * | 2021-08-20 | 2023-02-22 | Henkel AG & Co. KGaA | Vinyl ethers |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6239077B1 (en) | 1998-05-01 | 2001-05-29 | Nihon Nohyaku Co., Ltd. | Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof |
| PT1392281E (pt) | 2000-12-20 | 2007-05-31 | Novartis Ag | Amidoacetonitrilos anti-endoparasitários |
| AR035531A1 (es) | 2001-01-22 | 2004-06-02 | Novartis Ag | Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos |
| TWI236341B (en) | 2001-06-15 | 2005-07-21 | Novartis Ag | Aminoacetonitrile compounds for use in the control of endoparasites |
| AR038156A1 (es) | 2002-01-21 | 2004-12-29 | Novartis Ag | Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica |
| AR039020A1 (es) | 2002-03-21 | 2005-02-02 | Novartis Ag | Compuestos de aminoacetonitrilo |
| AR040229A1 (es) | 2002-05-22 | 2005-03-23 | Novartis Ag | Amidoacetonitrilos |
| AR040082A1 (es) | 2002-05-22 | 2005-03-16 | Novartis Ag | Derivados de n-acilaminoacetonitrilo y su uso para el control de parasitos |
| AR039961A1 (es) | 2002-06-06 | 2005-03-09 | Novartis Ag | Derivados de amidoacetonitrilo y su uso como pesticida |
| TW200400932A (en) | 2002-06-19 | 2004-01-16 | Novartis Ag | Organic compounds |
| GB0402677D0 (en) | 2003-11-06 | 2004-03-10 | Novartis Ag | Organic compounds |
| AR046757A1 (es) | 2003-12-10 | 2005-12-21 | Novartis Ag | Amidoacetonitrilos utiles como pesticidas |
| TW200613251A (en) | 2004-06-10 | 2006-05-01 | Novartis Ag | Organic compounds |
| ES2540966T3 (es) * | 2005-02-16 | 2015-07-15 | Anacor Pharmaceuticals, Inc. | Compuestos biocidas de boronoftalida |
| EP1910278A1 (en) | 2005-07-25 | 2008-04-16 | Novartis AG | Amidonitrile compounds |
| BRPI0621279B1 (pt) | 2005-12-30 | 2021-07-20 | Anacor Pharmaceuticals, Inc | Moléculas pequenas contendo boro |
| ES2367332T3 (es) | 2007-02-21 | 2011-11-02 | Pfizer Limited | Agentes antiparasitarios de benzofurano. |
| US20100026457A1 (en) * | 2008-08-04 | 2010-02-04 | Cooper Technologies Company | Location of Tagged Boxes |
| ES2393965T3 (es) | 2008-10-21 | 2013-01-03 | Merial Ltd. | Compuestos de tioamida, procedimiento de preparación y procedimiento de uso de los mismos |
| US8343944B2 (en) * | 2009-07-28 | 2013-01-01 | Anacor Pharmaceuticals, Inc. | Trisubstituted boron-containing molecules |
| WO2011019612A1 (en) * | 2009-08-14 | 2011-02-17 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| WO2011049971A1 (en) * | 2009-10-20 | 2011-04-28 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| EP2314292A1 (en) | 2009-10-20 | 2011-04-27 | Novartis AG | Endoparasiticidal compositions |
| UY32992A (es) | 2009-11-23 | 2011-04-29 | Novartis Ag | Compuestos orgánicos |
| LT3030519T (lt) * | 2013-08-09 | 2022-04-11 | Glaxosmithkline Intellectual Property (No. 2) Limited | Tricikliniai benzoksaborolo junginiai ir jų naudojimas |
-
2014
- 2014-02-28 AR ARP140100676A patent/AR094961A1/es unknown
- 2014-03-06 RS RS20171064A patent/RS56532B1/sr unknown
- 2014-03-06 AU AU2014237862A patent/AU2014237862B2/en not_active Ceased
- 2014-03-06 MX MX2015013051A patent/MX2015013051A/es unknown
- 2014-03-06 ES ES14712939.9T patent/ES2645687T3/es active Active
- 2014-03-06 PT PT147129399T patent/PT2970339T/pt unknown
- 2014-03-06 CN CN201480014758.9A patent/CN105051048B/zh not_active Expired - Fee Related
- 2014-03-06 EP EP14712939.9A patent/EP2970339B1/en active Active
- 2014-03-06 EA EA201591512A patent/EA027430B1/ru not_active IP Right Cessation
- 2014-03-06 PL PL14712939T patent/PL2970339T3/pl unknown
- 2014-03-06 CA CA2899972A patent/CA2899972A1/en not_active Abandoned
- 2014-03-06 US US14/760,208 patent/US9617285B2/en not_active Expired - Fee Related
- 2014-03-06 LT LTEP14712939.9T patent/LT2970339T/lt unknown
- 2014-03-06 TW TW103107747A patent/TW201506031A/zh unknown
- 2014-03-06 KR KR1020157024782A patent/KR101727421B1/ko active IP Right Grant
- 2014-03-06 JP JP2016500695A patent/JP6121043B2/ja active Active
- 2014-03-06 HU HUE14712939A patent/HUE035545T2/en unknown
- 2014-03-06 BR BR112015020823A patent/BR112015020823A8/pt active Search and Examination
- 2014-03-06 DK DK14712939.9T patent/DK2970339T3/en active
- 2014-03-06 SI SI201430345T patent/SI2970339T1/sl unknown
- 2014-03-06 WO PCT/US2014/020966 patent/WO2014149793A1/en active Application Filing
- 2014-11-18 NO NO14799476A patent/NO2904426T3/no unknown
-
2017
- 2017-10-09 HR HRP20171517TT patent/HRP20171517T1/hr unknown
- 2017-10-20 CY CY20171101096T patent/CY1119473T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP6121043B2 (ja) | 2017-04-26 |
| DK2970339T3 (en) | 2017-10-02 |
| CN105051048B (zh) | 2017-03-15 |
| LT2970339T (lt) | 2017-11-10 |
| US20150353581A1 (en) | 2015-12-10 |
| US9617285B2 (en) | 2017-04-11 |
| RS56532B1 (sr) | 2018-02-28 |
| TW201506031A (zh) | 2015-02-16 |
| PT2970339T (pt) | 2017-11-14 |
| SI2970339T1 (sl) | 2017-10-30 |
| EP2970339B1 (en) | 2017-08-16 |
| KR20150119154A (ko) | 2015-10-23 |
| BR112015020823A8 (pt) | 2019-09-17 |
| ES2645687T3 (es) | 2017-12-07 |
| EA027430B1 (ru) | 2017-07-31 |
| AU2014237862B2 (en) | 2017-01-12 |
| WO2014149793A1 (en) | 2014-09-25 |
| PL2970339T3 (pl) | 2018-01-31 |
| CA2899972A1 (en) | 2014-09-25 |
| BR112015020823A2 (pt) | 2017-07-18 |
| AR094961A1 (es) | 2015-09-09 |
| KR101727421B1 (ko) | 2017-04-14 |
| HRP20171517T1 (hr) | 2017-11-17 |
| JP2016516032A (ja) | 2016-06-02 |
| EP2970339A1 (en) | 2016-01-20 |
| MX2015013051A (es) | 2016-05-05 |
| NO2904426T3 (el) | 2018-02-10 |
| EA201591512A9 (ru) | 2016-04-29 |
| EA201591512A1 (ru) | 2016-01-29 |
| AU2014237862A1 (en) | 2015-08-13 |
| CN105051048A (zh) | 2015-11-11 |
| HUE035545T2 (en) | 2018-05-28 |
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