CY1122182T1 - Ανοσοκατασταλτικες φαρμακοτεχνικες μορφες - Google Patents
Ανοσοκατασταλτικες φαρμακοτεχνικες μορφεςInfo
- Publication number
- CY1122182T1 CY1122182T1 CY20191101097T CY191101097T CY1122182T1 CY 1122182 T1 CY1122182 T1 CY 1122182T1 CY 20191101097 T CY20191101097 T CY 20191101097T CY 191101097 T CY191101097 T CY 191101097T CY 1122182 T1 CY1122182 T1 CY 1122182T1
- Authority
- CY
- Cyprus
- Prior art keywords
- pharmaceutical forms
- api
- pharmaceutically acceptable
- immunosuppressant
- immunosuppressant pharmaceutical
- Prior art date
Links
- 229960003444 immunosuppressant agent Drugs 0.000 title 1
- 230000001861 immunosuppressant effect Effects 0.000 title 1
- 239000003018 immunosuppressive agent Substances 0.000 title 1
- 239000008186 active pharmaceutical agent Substances 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000007790 solid phase Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Organic Chemistry (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Transplantation (AREA)
- Physical Education & Sports Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Biomedical Technology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Abstract
Η παρούσα εφεύρεση αναφέρεται σε μια φαρμακευτική σύνθεση στερεάς φάσης, η οποία αποτελείται από ένα ή περισσότερα φαρμακευτικώς αποδεκτά έκδοχα και ένα δραστικό φαρμακευτικό συστατικό ("API"), το οποίο είναι μια ένωση του τύπου Α1 ή Α2 ή ένα φαρμακευτικώς αποδεκτό άλας, επιδιαλύτωμα ή υδρίτης αυτής, όπου το API δεν εκτίθεται σε μια βασική ένωση.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11150431 | 2011-01-07 | ||
| EP12700262.4A EP2661261B1 (en) | 2011-01-07 | 2012-01-05 | Immunosuppressant formulations |
| PCT/EP2012/050151 WO2012093161A1 (en) | 2011-01-07 | 2012-01-05 | Immunosuppressant formulations |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CY1122182T1 true CY1122182T1 (el) | 2020-11-25 |
Family
ID=44022942
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CY20191101097T CY1122182T1 (el) | 2011-01-07 | 2019-10-22 | Ανοσοκατασταλτικες φαρμακοτεχνικες μορφες |
Country Status (35)
| Country | Link |
|---|---|
| US (3) | US20130273161A1 (el) |
| EP (2) | EP2661261B1 (el) |
| JP (2) | JP6111202B2 (el) |
| KR (2) | KR102166885B1 (el) |
| CN (1) | CN103458877B (el) |
| AR (2) | AR084801A1 (el) |
| AU (1) | AU2012204835B2 (el) |
| BR (1) | BR112013017302B1 (el) |
| CA (1) | CA2823616C (el) |
| CL (1) | CL2013001979A1 (el) |
| CO (1) | CO6761402A2 (el) |
| CY (1) | CY1122182T1 (el) |
| DK (1) | DK2661261T3 (el) |
| EA (1) | EA026144B9 (el) |
| EC (1) | ECSP13012812A (el) |
| ES (1) | ES2751920T3 (el) |
| GT (1) | GT201300178A (el) |
| HR (1) | HRP20191842T1 (el) |
| HU (1) | HUE045612T2 (el) |
| IL (1) | IL227094B (el) |
| JO (1) | JO3619B1 (el) |
| LT (1) | LT2661261T (el) |
| MA (1) | MA34897B1 (el) |
| MX (2) | MX357304B (el) |
| MY (1) | MY161162A (el) |
| PE (1) | PE20140216A1 (el) |
| PL (1) | PL2661261T3 (el) |
| PT (1) | PT2661261T (el) |
| SG (1) | SG191286A1 (el) |
| SI (1) | SI2661261T1 (el) |
| TN (1) | TN2013000257A1 (el) |
| TW (2) | TWI583380B (el) |
| UA (1) | UA114283C2 (el) |
| WO (1) | WO2012093161A1 (el) |
| ZA (1) | ZA201304465B (el) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2943598C (en) * | 2014-04-10 | 2023-03-07 | Novartis Ag | S1p modulator immediate release dosage regimen |
| PE20161385A1 (es) * | 2014-04-10 | 2017-01-05 | Novartis Ag | Formulacion inmunosupresora |
| CA2973540A1 (en) | 2015-02-26 | 2016-09-01 | Novartis Ag | Treatment of autoimmune disease in a patient receiving additionally a beta-blocker |
| SI3318259T1 (sl) * | 2015-07-03 | 2023-06-30 | Astellas Pharma Inc. | Stabilni farmacevtski sestavki za oralno dajanje |
| US11629124B2 (en) | 2017-03-09 | 2023-04-18 | Novartis Ag | Solid forms comprising an oxime ether compound, compositions and methods of use thereof |
| EP3687498A1 (en) | 2017-09-27 | 2020-08-05 | Novartis AG | Parenteral formulation comprising siponimod |
| AU2018343239A1 (en) | 2017-09-29 | 2020-03-12 | Novartis Ag | Dosing regimen of siponimod |
| US20200316021A1 (en) | 2017-09-29 | 2020-10-08 | Novartis Ag | Dosing Regimen of Siponimod |
| CN109908095A (zh) * | 2019-04-08 | 2019-06-21 | 肇庆学院 | 一种西尼莫德片剂及制备方法 |
| WO2021214717A1 (en) | 2020-04-23 | 2021-10-28 | Novartis Ag | Dosing regimen for the use of siponimod for the treatment of acute respiratory distress syndrome |
| WO2023172508A1 (en) * | 2022-03-09 | 2023-09-14 | Isp Investments Llc | Co-processed excipient composition |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU225964B1 (en) | 1994-07-12 | 2008-01-28 | Berwind Pharma Service | Moisture barrier film coating composition, method, and coated form |
| ATE527986T1 (de) * | 2002-11-07 | 2011-10-15 | Taisho Pharmaceutical Co Ltd | Grundlage für orale zusammensetzung und orale zusammensetzung |
| MY150088A (en) | 2003-05-19 | 2013-11-29 | Irm Llc | Immunosuppressant compounds and compositions |
| GT200600350A (es) | 2005-08-09 | 2007-03-28 | Formulaciones líquidas | |
| EP3120833A1 (en) * | 2007-10-12 | 2017-01-25 | Novartis Ag | Compositions comprising sphingosine 1 phosphate (s1p) receptor modulators |
| ES2526119T3 (es) | 2008-08-18 | 2015-01-07 | Novartis Ag | Derivado de azetidina para el tratamiento de neuropatías periféricas |
| PE20120336A1 (es) * | 2008-12-18 | 2012-04-30 | Novartis Ag | Sal de hemi-fumarato del acido 1-[4-[1-(4-ciclohexil-3-triflouro-metil-benciloxi-imino)-etil)-2-etil-bencil]-azetidin-3-carboxilico |
| AU2009335887A1 (en) | 2008-12-18 | 2011-06-30 | Novartis Ag | New salts |
| BRPI0922457A2 (pt) | 2008-12-18 | 2015-12-15 | Novartis Ag | forma polimórfica de ácido 1-(4-{1-[(e)-4-ciclo-hexil-3-trifluormetil-benziloxi-imino]-etil)-2-etil-benzil)-azetidino-3-carboxílico" |
| KR101660555B1 (ko) | 2008-12-22 | 2016-09-27 | 노파르티스 아게 | Ｓ１ｐ 수용체 효능제의 투여 요법 |
-
2012
- 2012-01-05 MX MX2013007909A patent/MX357304B/es active IP Right Grant
- 2012-01-05 EA EA201391018A patent/EA026144B9/ru active Protection Beyond IP Right Term
- 2012-01-05 MX MX2017007300A patent/MX371290B/es unknown
- 2012-01-05 HU HUE12700262A patent/HUE045612T2/hu unknown
- 2012-01-05 BR BR112013017302-5A patent/BR112013017302B1/pt active IP Right Grant
- 2012-01-05 LT LT12700262T patent/LT2661261T/lt unknown
- 2012-01-05 WO PCT/EP2012/050151 patent/WO2012093161A1/en active Application Filing
- 2012-01-05 ES ES12700262T patent/ES2751920T3/es active Active
- 2012-01-05 MA MA36170A patent/MA34897B1/fr unknown
- 2012-01-05 PE PE2013001522A patent/PE20140216A1/es active IP Right Grant
- 2012-01-05 CA CA2823616A patent/CA2823616C/en active Active
- 2012-01-05 JP JP2013547861A patent/JP6111202B2/ja active Active
- 2012-01-05 AU AU2012204835A patent/AU2012204835B2/en active Active
- 2012-01-05 SG SG2013047923A patent/SG191286A1/en unknown
- 2012-01-05 EP EP12700262.4A patent/EP2661261B1/en active Active
- 2012-01-05 PT PT127002624T patent/PT2661261T/pt unknown
- 2012-01-05 KR KR1020197004860A patent/KR102166885B1/ko active IP Right Grant
- 2012-01-05 DK DK12700262.4T patent/DK2661261T3/da active
- 2012-01-05 UA UAA201307576A patent/UA114283C2/uk unknown
- 2012-01-05 KR KR1020137020755A patent/KR101951966B1/ko active IP Right Grant
- 2012-01-05 JO JOP/2012/0005A patent/JO3619B1/ar active
- 2012-01-05 SI SI201231683T patent/SI2661261T1/sl unknown
- 2012-01-05 CN CN201280004869.2A patent/CN103458877B/zh active Active
- 2012-01-05 PL PL12700262T patent/PL2661261T3/pl unknown
- 2012-01-05 EP EP19188018.6A patent/EP3590507A1/en active Pending
- 2012-01-06 MY MYPI2013002251A patent/MY161162A/en unknown
- 2012-01-06 TW TW104142389A patent/TWI583380B/zh active
- 2012-01-06 AR ARP120100047A patent/AR084801A1/es not_active Application Discontinuation
- 2012-01-06 TW TW101100702A patent/TWI610672B/zh active
-
2013
- 2013-06-14 US US13/917,730 patent/US20130273161A1/en not_active Abandoned
- 2013-06-14 TN TNP2013000257A patent/TN2013000257A1/fr unknown
- 2013-06-18 ZA ZA2013/04465A patent/ZA201304465B/en unknown
- 2013-06-20 IL IL227094A patent/IL227094B/en active IP Right Grant
- 2013-07-05 GT GT201300178A patent/GT201300178A/es unknown
- 2013-07-05 CL CL2013001979A patent/CL2013001979A1/es unknown
- 2013-07-16 CO CO13168667A patent/CO6761402A2/es unknown
- 2013-08-07 EC ECSP13012812 patent/ECSP13012812A/es unknown
-
2017
- 2017-03-13 JP JP2017047220A patent/JP6324569B2/ja active Active
-
2019
- 2019-10-11 HR HRP20191842TT patent/HRP20191842T1/hr unknown
- 2019-10-22 CY CY20191101097T patent/CY1122182T1/el unknown
-
2020
- 2020-02-28 US US16/804,926 patent/US20200199069A1/en not_active Abandoned
-
2021
- 2021-04-14 US US17/230,175 patent/US20220064110A1/en active Pending
-
2022
- 2022-01-17 AR ARP220100086A patent/AR124662A2/es unknown
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