MX371290B - Formulaciones inmunosupresoras. - Google Patents

Formulaciones inmunosupresoras.

Info

Publication number
MX371290B
MX371290B MX2017007300A MX2017007300A MX371290B MX 371290 B MX371290 B MX 371290B MX 2017007300 A MX2017007300 A MX 2017007300A MX 2017007300 A MX2017007300 A MX 2017007300A MX 371290 B MX371290 B MX 371290B
Authority
MX
Mexico
Prior art keywords
api
immunosuppressant
formulations
compound
immunosuppressant formulations
Prior art date
Application number
MX2017007300A
Other languages
English (en)
Inventor
Reynaud Emeric
Bouillot Philippe
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44022942&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX371290(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MX371290B publication Critical patent/MX371290B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Transplantation (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biomedical Technology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

Abstract

La presente invención se refiere a una composición farmacéutica en fase sólida, la cual comprende uno o más excipientes farmacéuticamente aceptables, y un ingrediente farmacéutico activo ("API"), el cual es un compuesto de la fórmula A1 o A2, o una sal, solvato o hidrato farmacológicamente aceptable del mismo, en donde el ingrediente farmacéutico activo (API) no se expone a un compuesto básico.
MX2017007300A 2011-01-07 2012-01-05 Formulaciones inmunosupresoras. MX371290B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP11150431 2011-01-07
PCT/EP2012/050151 WO2012093161A1 (en) 2011-01-07 2012-01-05 Immunosuppressant formulations

Publications (1)

Publication Number Publication Date
MX371290B true MX371290B (es) 2020-01-24

Family

ID=44022942

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2013007909A MX357304B (es) 2011-01-07 2012-01-05 Formulaciones inmunosupresoras.
MX2017007300A MX371290B (es) 2011-01-07 2012-01-05 Formulaciones inmunosupresoras.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
MX2013007909A MX357304B (es) 2011-01-07 2012-01-05 Formulaciones inmunosupresoras.

Country Status (35)

Country Link
US (3) US20130273161A1 (es)
EP (2) EP3590507A1 (es)
JP (2) JP6111202B2 (es)
KR (2) KR102166885B1 (es)
CN (1) CN103458877B (es)
AR (2) AR084801A1 (es)
AU (1) AU2012204835B2 (es)
BR (1) BR112013017302B1 (es)
CA (1) CA2823616C (es)
CL (1) CL2013001979A1 (es)
CO (1) CO6761402A2 (es)
CY (1) CY1122182T1 (es)
DK (1) DK2661261T3 (es)
EA (1) EA026144B9 (es)
EC (1) ECSP13012812A (es)
ES (1) ES2751920T3 (es)
GT (1) GT201300178A (es)
HR (1) HRP20191842T1 (es)
HU (1) HUE045612T2 (es)
IL (1) IL227094B (es)
JO (1) JO3619B1 (es)
LT (1) LT2661261T (es)
MA (1) MA34897B1 (es)
MX (2) MX357304B (es)
MY (1) MY161162A (es)
PE (1) PE20140216A1 (es)
PL (1) PL2661261T3 (es)
PT (1) PT2661261T (es)
SG (1) SG191286A1 (es)
SI (1) SI2661261T1 (es)
TN (1) TN2013000257A1 (es)
TW (2) TWI583380B (es)
UA (1) UA114283C2 (es)
WO (1) WO2012093161A1 (es)
ZA (1) ZA201304465B (es)

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PE20140216A1 (es) 2011-01-07 2014-03-01 Novartis Ag Formulaciones inmunosupresoras
RU2020107732A (ru) * 2014-04-10 2020-03-30 Новартис Аг Схема дозирования модулятора s1p с немедленным высвобождением
KR102466348B1 (ko) * 2014-04-10 2022-11-10 노파르티스 아게 면역억제제 제제
CA2973540A1 (en) 2015-02-26 2016-09-01 Novartis Ag Treatment of autoimmune disease in a patient receiving additionally a beta-blocker
SI3318259T1 (sl) * 2015-07-03 2023-06-30 Astellas Pharma Inc. Stabilni farmacevtski sestavki za oralno dajanje
US11629124B2 (en) 2017-03-09 2023-04-18 Novartis Ag Solid forms comprising an oxime ether compound, compositions and methods of use thereof
US11434200B2 (en) 2017-03-09 2022-09-06 Novartis Ag Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof
MX2020007270A (es) 2017-09-27 2020-08-17 Novartis Ag Formulacion parenteral que comprende siponimod.
JP2020535139A (ja) 2017-09-29 2020-12-03 ノバルティス アーゲー シポニモドの投与レジメン
US20200316021A1 (en) 2017-09-29 2020-10-08 Novartis Ag Dosing Regimen of Siponimod
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WO2021214717A1 (en) 2020-04-23 2021-10-28 Novartis Ag Dosing regimen for the use of siponimod for the treatment of acute respiratory distress syndrome
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WO2024126409A1 (en) 2022-12-12 2024-06-20 Synthon B.V. Pharmaceutical composition of siponimod

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Also Published As

Publication number Publication date
JP2017141248A (ja) 2017-08-17
CO6761402A2 (es) 2013-09-30
EP2661261A1 (en) 2013-11-13
CA2823616C (en) 2019-01-29
TW201249438A (en) 2012-12-16
JP6324569B2 (ja) 2018-05-16
EA026144B1 (ru) 2017-03-31
TN2013000257A1 (en) 2014-11-10
DK2661261T3 (da) 2019-10-21
CA2823616A1 (en) 2012-07-12
CY1122182T1 (el) 2020-11-25
LT2661261T (lt) 2019-10-25
CN103458877B (zh) 2016-06-08
JP6111202B2 (ja) 2017-04-05
AR084801A1 (es) 2013-06-26
HUE045612T2 (hu) 2020-01-28
IL227094B (en) 2019-03-31
MA34897B1 (fr) 2014-02-01
ECSP13012812A (es) 2013-09-30
US20220064110A1 (en) 2022-03-03
TWI610672B (zh) 2018-01-11
JP2014501770A (ja) 2014-01-23
ES2751920T3 (es) 2020-04-02
SI2661261T1 (sl) 2019-11-29
NZ612420A (en) 2015-05-29
US12071402B2 (en) 2024-08-27
WO2012093161A1 (en) 2012-07-12
KR102166885B1 (ko) 2020-10-19
MY161162A (en) 2017-04-14
CL2013001979A1 (es) 2013-11-22
GT201300178A (es) 2014-12-30
KR101951966B1 (ko) 2019-02-25
JO3619B1 (ar) 2020-08-27
EP2661261B1 (en) 2019-07-31
EP3590507A1 (en) 2020-01-08
US20200199069A1 (en) 2020-06-25
AU2012204835A1 (en) 2013-08-01
MX2013007909A (es) 2013-08-29
TWI583380B (zh) 2017-05-21
PL2661261T3 (pl) 2020-01-31
US20130273161A1 (en) 2013-10-17
TW201609092A (zh) 2016-03-16
EA201391018A1 (ru) 2013-11-29
UA114283C2 (uk) 2017-05-25
BR112013017302B1 (pt) 2021-12-07
KR20190025727A (ko) 2019-03-11
HRP20191842T1 (hr) 2019-12-27
AR124662A2 (es) 2023-04-19
KR20140037815A (ko) 2014-03-27
AU2012204835B2 (en) 2015-07-09
PT2661261T (pt) 2019-10-25
EA026144B9 (ru) 2021-10-26
BR112013017302A2 (pt) 2016-10-25
PE20140216A1 (es) 2014-03-01
MX357304B (es) 2018-07-04
CN103458877A (zh) 2013-12-18
ZA201304465B (en) 2014-02-26
SG191286A1 (en) 2013-07-31

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