DK2661261T3 - Immunsuppressive formuleringer - Google Patents

Immunsuppressive formuleringer Download PDF

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Publication number
DK2661261T3
DK2661261T3 DK12700262.4T DK12700262T DK2661261T3 DK 2661261 T3 DK2661261 T3 DK 2661261T3 DK 12700262 T DK12700262 T DK 12700262T DK 2661261 T3 DK2661261 T3 DK 2661261T3
Authority
DK
Denmark
Prior art keywords
immunosuppressive
formulations
immunosuppressive formulations
Prior art date
Application number
DK12700262.4T
Other languages
English (en)
Inventor
Philippe Bouillot
Emeric Reynaud
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44022942&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK2661261(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Application granted granted Critical
Publication of DK2661261T3 publication Critical patent/DK2661261T3/da

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Biomedical Technology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
DK12700262.4T 2011-01-07 2012-01-05 Immunsuppressive formuleringer DK2661261T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP11150431 2011-01-07
PCT/EP2012/050151 WO2012093161A1 (en) 2011-01-07 2012-01-05 Immunosuppressant formulations

Publications (1)

Publication Number Publication Date
DK2661261T3 true DK2661261T3 (da) 2019-10-21

Family

ID=44022942

Family Applications (1)

Application Number Title Priority Date Filing Date
DK12700262.4T DK2661261T3 (da) 2011-01-07 2012-01-05 Immunsuppressive formuleringer

Country Status (35)

Country Link
US (3) US20130273161A1 (da)
EP (2) EP2661261B1 (da)
JP (2) JP6111202B2 (da)
KR (2) KR101951966B1 (da)
CN (1) CN103458877B (da)
AR (2) AR084801A1 (da)
AU (1) AU2012204835B2 (da)
BR (1) BR112013017302B1 (da)
CA (1) CA2823616C (da)
CL (1) CL2013001979A1 (da)
CO (1) CO6761402A2 (da)
CY (1) CY1122182T1 (da)
DK (1) DK2661261T3 (da)
EA (1) EA026144B9 (da)
EC (1) ECSP13012812A (da)
ES (1) ES2751920T3 (da)
GT (1) GT201300178A (da)
HR (1) HRP20191842T1 (da)
HU (1) HUE045612T2 (da)
IL (1) IL227094B (da)
JO (1) JO3619B1 (da)
LT (1) LT2661261T (da)
MA (1) MA34897B1 (da)
MX (2) MX357304B (da)
MY (1) MY161162A (da)
PE (1) PE20140216A1 (da)
PL (1) PL2661261T3 (da)
PT (1) PT2661261T (da)
SG (1) SG191286A1 (da)
SI (1) SI2661261T1 (da)
TN (1) TN2013000257A1 (da)
TW (2) TWI583380B (da)
UA (1) UA114283C2 (da)
WO (1) WO2012093161A1 (da)
ZA (1) ZA201304465B (da)

Families Citing this family (14)

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SI3129006T1 (sl) * 2014-04-10 2021-08-31 Novartis Ag Formulacija imunosupresivov
CA2973540A1 (en) 2015-02-26 2016-09-01 Novartis Ag Treatment of autoimmune disease in a patient receiving additionally a beta-blocker
WO2017006855A1 (ja) 2015-07-03 2017-01-12 アステラス製薬株式会社 安定な経口投与用医薬組成物
US11629124B2 (en) 2017-03-09 2023-04-18 Novartis Ag Solid forms comprising an oxime ether compound, compositions and methods of use thereof
US11434200B2 (en) 2017-03-09 2022-09-06 Novartis Ag Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof
AU2018341136A1 (en) 2017-09-27 2020-03-12 Novartis Ag Parenteral formulation comprising siponimod
RU2020114751A (ru) 2017-09-29 2021-10-29 Новартис Аг Схема введения доз сипонимода
MX2020007268A (es) 2017-09-29 2020-08-17 Novartis Ag Regimen de dosificacion de siponimod.
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WO2021214717A1 (en) 2020-04-23 2021-10-28 Novartis Ag Dosing regimen for the use of siponimod for the treatment of acute respiratory distress syndrome
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WO2024126409A1 (en) 2022-12-12 2024-06-20 Synthon B.V. Pharmaceutical composition of siponimod

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JP5657565B2 (ja) 2008-12-22 2015-01-21 ノバルティス アーゲー S1p受容体アゴニストの投与レジメン
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CA2773330C (en) 2009-09-29 2021-11-02 Novartis Ag Dosage regimen of an s1p receptor modulator
CA2823616C (en) 2011-01-07 2019-01-29 Novartis Ag Immunosuppressant formulations
WO2012095853A1 (en) 2011-01-10 2012-07-19 Novartis Pharma Ag Modified release formulations comprising sip receptor modulators
TW201320994A (zh) 2011-10-11 2013-06-01 Novartis Ag 投藥療程
CA3149287A1 (en) 2013-04-04 2014-10-09 Novartis Ag Identifying patient response to s1p receptor modulator administration
SI3129006T1 (sl) 2014-04-10 2021-08-31 Novartis Ag Formulacija imunosupresivov

Also Published As

Publication number Publication date
MX371290B (es) 2020-01-24
EA201391018A1 (ru) 2013-11-29
WO2012093161A1 (en) 2012-07-12
MA34897B1 (fr) 2014-02-01
ECSP13012812A (es) 2013-09-30
EP2661261A1 (en) 2013-11-13
CN103458877B (zh) 2016-06-08
CY1122182T1 (el) 2020-11-25
BR112013017302B1 (pt) 2021-12-07
AU2012204835A1 (en) 2013-08-01
AR084801A1 (es) 2013-06-26
SI2661261T1 (sl) 2019-11-29
JP6111202B2 (ja) 2017-04-05
LT2661261T (lt) 2019-10-25
NZ612420A (en) 2015-05-29
KR101951966B1 (ko) 2019-02-25
KR102166885B1 (ko) 2020-10-19
GT201300178A (es) 2014-12-30
US12071402B2 (en) 2024-08-27
IL227094B (en) 2019-03-31
JP2017141248A (ja) 2017-08-17
EP2661261B1 (en) 2019-07-31
CL2013001979A1 (es) 2013-11-22
CA2823616A1 (en) 2012-07-12
EP3590507A1 (en) 2020-01-08
CA2823616C (en) 2019-01-29
PE20140216A1 (es) 2014-03-01
AU2012204835B2 (en) 2015-07-09
US20220064110A1 (en) 2022-03-03
ZA201304465B (en) 2014-02-26
KR20190025727A (ko) 2019-03-11
CN103458877A (zh) 2013-12-18
JP6324569B2 (ja) 2018-05-16
MX357304B (es) 2018-07-04
KR20140037815A (ko) 2014-03-27
EA026144B1 (ru) 2017-03-31
ES2751920T3 (es) 2020-04-02
BR112013017302A2 (pt) 2016-10-25
AR124662A2 (es) 2023-04-19
JO3619B1 (ar) 2020-08-27
CO6761402A2 (es) 2013-09-30
HUE045612T2 (hu) 2020-01-28
TW201609092A (zh) 2016-03-16
US20200199069A1 (en) 2020-06-25
PT2661261T (pt) 2019-10-25
TN2013000257A1 (en) 2014-11-10
TWI583380B (zh) 2017-05-21
PL2661261T3 (pl) 2020-01-31
TW201249438A (en) 2012-12-16
HRP20191842T1 (hr) 2019-12-27
MX2013007909A (es) 2013-08-29
EA026144B9 (ru) 2021-10-26
US20130273161A1 (en) 2013-10-17
JP2014501770A (ja) 2014-01-23
MY161162A (en) 2017-04-14
TWI610672B (zh) 2018-01-11
SG191286A1 (en) 2013-07-31
UA114283C2 (uk) 2017-05-25

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