PL2661261T3 - Formulacje immunosupresyjne - Google Patents

Formulacje immunosupresyjne

Info

Publication number
PL2661261T3
PL2661261T3 PL12700262T PL12700262T PL2661261T3 PL 2661261 T3 PL2661261 T3 PL 2661261T3 PL 12700262 T PL12700262 T PL 12700262T PL 12700262 T PL12700262 T PL 12700262T PL 2661261 T3 PL2661261 T3 PL 2661261T3
Authority
PL
Poland
Prior art keywords
immunosuppressant
formulations
immunosuppressant formulations
Prior art date
Application number
PL12700262T
Other languages
English (en)
Inventor
Philippe BOUILLOT
Emeric Reynaud
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44022942&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2661261(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PL2661261T3 publication Critical patent/PL2661261T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Transplantation (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
PL12700262T 2011-01-07 2012-01-05 Formulacje immunosupresyjne PL2661261T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11150431 2011-01-07
EP12700262.4A EP2661261B1 (en) 2011-01-07 2012-01-05 Immunosuppressant formulations
PCT/EP2012/050151 WO2012093161A1 (en) 2011-01-07 2012-01-05 Immunosuppressant formulations

Publications (1)

Publication Number Publication Date
PL2661261T3 true PL2661261T3 (pl) 2020-01-31

Family

ID=44022942

Family Applications (1)

Application Number Title Priority Date Filing Date
PL12700262T PL2661261T3 (pl) 2011-01-07 2012-01-05 Formulacje immunosupresyjne

Country Status (35)

Country Link
US (3) US20130273161A1 (pl)
EP (2) EP3590507A1 (pl)
JP (2) JP6111202B2 (pl)
KR (2) KR102166885B1 (pl)
CN (1) CN103458877B (pl)
AR (2) AR084801A1 (pl)
AU (1) AU2012204835B2 (pl)
BR (1) BR112013017302B1 (pl)
CA (1) CA2823616C (pl)
CL (1) CL2013001979A1 (pl)
CO (1) CO6761402A2 (pl)
CY (1) CY1122182T1 (pl)
DK (1) DK2661261T3 (pl)
EA (1) EA026144B9 (pl)
EC (1) ECSP13012812A (pl)
ES (1) ES2751920T3 (pl)
GT (1) GT201300178A (pl)
HR (1) HRP20191842T1 (pl)
HU (1) HUE045612T2 (pl)
IL (1) IL227094B (pl)
JO (1) JO3619B1 (pl)
LT (1) LT2661261T (pl)
MA (1) MA34897B1 (pl)
MX (2) MX357304B (pl)
MY (1) MY161162A (pl)
PE (1) PE20140216A1 (pl)
PL (1) PL2661261T3 (pl)
PT (1) PT2661261T (pl)
SG (1) SG191286A1 (pl)
SI (1) SI2661261T1 (pl)
TN (1) TN2013000257A1 (pl)
TW (2) TWI583380B (pl)
UA (1) UA114283C2 (pl)
WO (1) WO2012093161A1 (pl)
ZA (1) ZA201304465B (pl)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20140216A1 (es) 2011-01-07 2014-03-01 Novartis Ag Formulaciones inmunosupresoras
RU2020107732A (ru) * 2014-04-10 2020-03-30 Новартис Аг Схема дозирования модулятора s1p с немедленным высвобождением
KR102466348B1 (ko) * 2014-04-10 2022-11-10 노파르티스 아게 면역억제제 제제
CA2973540A1 (en) 2015-02-26 2016-09-01 Novartis Ag Treatment of autoimmune disease in a patient receiving additionally a beta-blocker
SI3318259T1 (sl) * 2015-07-03 2023-06-30 Astellas Pharma Inc. Stabilni farmacevtski sestavki za oralno dajanje
US11629124B2 (en) 2017-03-09 2023-04-18 Novartis Ag Solid forms comprising an oxime ether compound, compositions and methods of use thereof
US11434200B2 (en) 2017-03-09 2022-09-06 Novartis Ag Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof
MX2020007270A (es) 2017-09-27 2020-08-17 Novartis Ag Formulacion parenteral que comprende siponimod.
JP2020535139A (ja) 2017-09-29 2020-12-03 ノバルティス アーゲー シポニモドの投与レジメン
US20200316021A1 (en) 2017-09-29 2020-10-08 Novartis Ag Dosing Regimen of Siponimod
CN109908095A (zh) * 2019-04-08 2019-06-21 肇庆学院 一种西尼莫德片剂及制备方法
WO2021214717A1 (en) 2020-04-23 2021-10-28 Novartis Ag Dosing regimen for the use of siponimod for the treatment of acute respiratory distress syndrome
WO2023172508A1 (en) * 2022-03-09 2023-09-14 Isp Investments Llc Co-processed excipient composition
WO2024126409A1 (en) 2022-12-12 2024-06-20 Synthon B.V. Pharmaceutical composition of siponimod

Family Cites Families (44)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3872113A (en) 1972-05-30 1975-03-18 Endo Lab Hydroxy- and acetoxy-phthalaldehydric acid, O-(substituted) oximes
DE122011100012I1 (de) 1992-10-21 2011-10-20 Mitsubishi Tanabe Pharma Corp 2-Amino-1, 3-propandiolverbindung und immunosuppressium.
CZ297271B6 (cs) 1994-07-12 2006-10-11 Bpsi Holdings, Inc. Suchá povlaková hmota pro výrobu filmu zabranujícímu prístupu vlhkosti, zpusob a tvorba povlaku
HU224814B1 (en) 1995-12-28 2006-02-28 Mitsubishi Pharma Corp Use of propane-1,3-diol derivative for the preparation of a medicament useful for the topical treating of inflammatory and immune diseases
MY121470A (en) 1999-05-03 2006-01-28 Ranbaxy Lab Ltd Stable solid pharmaceutical compositions containing enalapril maleate
AU2001285331B2 (en) 2000-08-31 2006-04-06 Merck & Co., Inc. Phosphate derivatives as immunoregulatory agents
AR041786A1 (es) 2002-03-15 2005-06-01 Novartis Ag Derivados de azetidina como antagonistas del receptor ccr-3, un proceso para su preparacion, una composicion farmaceutica y el uso de dichos derivados para la elaboracion de un medicamento
CN1652757B (zh) 2002-05-16 2012-02-08 诺瓦提斯公司 Edg受体结合剂在癌症中的应用
KR101030586B1 (ko) * 2002-11-07 2011-04-21 다이쇼 세이야꾸 가부시끼가이샤 구강용 조성물 기제 및 구강용 조성물
PE20130200A1 (es) 2003-04-08 2013-03-09 Novartis Ag Composicion farmaceutica que contiene un agonista del receptor s1p y un alcohol de azucar
BRPI0410746A (pt) 2003-05-19 2006-06-27 Irm Llc compostos e composições imunossupressoras
MY150088A (en) 2003-05-19 2013-11-29 Irm Llc Immunosuppressant compounds and compositions
PE20050158A1 (es) 2003-05-19 2005-05-12 Irm Llc Compuestos inmunosupresores y composiciones
JP4861177B2 (ja) 2003-09-12 2012-01-25 ニューロノバ エービー 神経系の障害の処置
TW200517106A (en) 2003-10-29 2005-06-01 Wyeth Corp Sustained release pharmaceutical compositions
JP2007536310A (ja) 2004-05-03 2007-12-13 ノバルティス アクチエンゲゼルシャフト S1p受容体アゴニストおよびjak3キナーゼ阻害剤を含む、組合せ剤
US20060002999A1 (en) 2004-06-17 2006-01-05 Forest Laboratories, Inc. Immediate release formulations of 1-aminocyclohexane compounds, memantine and neramexane
MX2007006373A (es) 2004-11-29 2007-06-20 Novartis Ag Regimen de dosificacion de un agonista del receptor s1p.
EP1688141A1 (en) 2005-01-31 2006-08-09 elbion AG The use of flupirtine for the treatment of overactive bladder and associated diseases, and for the treatment of irritable bowel syndrome
GB0504544D0 (en) 2005-03-04 2005-04-13 Novartis Ag Organic compounds
RU2296999C2 (ru) 2005-03-09 2007-04-10 Алексей Арнольдович Корженевский Способ выявления критериев для проведения адекватной иммунотерапии гнойно-септических заболеваний
GT200600350A (es) 2005-08-09 2007-03-28 Formulaciones líquidas
JP5269595B2 (ja) 2005-09-09 2013-08-21 アンジェリーニ ラボファーム リミテッド ライアビリティ カンパニー 1日1回投与用トラゾドン組成物
GB0612721D0 (en) 2006-06-27 2006-08-09 Novartis Ag Organic compounds
WO2008072056A1 (en) 2006-12-14 2008-06-19 Pfizer Limited Use of mtp inhibitors for the treatment of obesity using low doses and dose-escalation
DE102007019417A1 (de) 2007-04-23 2008-11-13 Grünenthal GmbH Tapentadol zur Schmerzbehandlung bei Arthrose
EP2142184B1 (en) 2007-05-04 2018-10-24 Novartis AG Use of s1p receptor modulator
WO2009048993A2 (en) 2007-10-12 2009-04-16 Novartis Ag Compositions comprising sphingosine 1 phosphate (s1p) receptor modulators
KR101718639B1 (ko) 2008-03-17 2017-03-21 액테리온 파마슈티칼 리미티드 선별적 s1p₁ 수용체 작동약에 대한 투약 섭생
KR20170081755A (ko) 2008-06-20 2017-07-12 노파르티스 아게 다발성 경화증을 치료하기 위한 소아용 조성물
CA2730751A1 (en) 2008-07-23 2010-01-28 Novartis Ag Sphingosine 1 phosphate receptor modulators and their use to treat muscle inflammation
JP5624037B2 (ja) * 2008-08-18 2014-11-12 ノバルティスアーゲー 末梢神経障害の治療のための化合物
MX2011006609A (es) * 2008-12-18 2011-06-30 Novartis Ag Sal de hemi-fumarato del acido 1-[4-[1-(4-ciclohexil-3-trifluoro-m etil-benciloxi-imino)-etil]-2-etil-bencil]-azetidin-3-carboxilico .
US8486930B2 (en) 2008-12-18 2013-07-16 Novartis Ag Salts
ES2531831T3 (es) 2008-12-18 2015-03-20 Novartis Ag Forma polimórfica del ácido 1-(4-{1-[(E)-4-ciclohexil-3-trifluorometil-benciloxiimino]-etil}-2-etil-bencil)-azetidin-3-carboxilico
WO2010070083A1 (en) 2008-12-19 2010-06-24 Novartis Ag Mouthpiece for an inhaler
SG171888A1 (en) 2008-12-22 2011-07-28 Novartis Ag Dosage regimen of an s1p receptor agonist
HUE026869T2 (en) 2008-12-22 2016-08-29 Novartis Ag Dosing regimen for fingolimod for the treatment of multiple sclerosis
SG178987A1 (en) 2009-09-29 2012-04-27 Novartis Ag Dosage regimen of an s1p receptor modulator
PE20140216A1 (es) 2011-01-07 2014-03-01 Novartis Ag Formulaciones inmunosupresoras
WO2012095853A1 (en) 2011-01-10 2012-07-19 Novartis Pharma Ag Modified release formulations comprising sip receptor modulators
TW201320994A (zh) 2011-10-11 2013-06-01 Novartis Ag 投藥療程
SG11201506493VA (en) 2013-04-04 2015-10-29 Novartis Ag Identifying patient response to s1p receptor modulator administration
KR102466348B1 (ko) 2014-04-10 2022-11-10 노파르티스 아게 면역억제제 제제

Also Published As

Publication number Publication date
JP2017141248A (ja) 2017-08-17
CO6761402A2 (es) 2013-09-30
EP2661261A1 (en) 2013-11-13
CA2823616C (en) 2019-01-29
TW201249438A (en) 2012-12-16
JP6324569B2 (ja) 2018-05-16
EA026144B1 (ru) 2017-03-31
TN2013000257A1 (en) 2014-11-10
DK2661261T3 (da) 2019-10-21
CA2823616A1 (en) 2012-07-12
CY1122182T1 (el) 2020-11-25
LT2661261T (lt) 2019-10-25
CN103458877B (zh) 2016-06-08
JP6111202B2 (ja) 2017-04-05
AR084801A1 (es) 2013-06-26
HUE045612T2 (hu) 2020-01-28
IL227094B (en) 2019-03-31
MA34897B1 (fr) 2014-02-01
ECSP13012812A (es) 2013-09-30
US20220064110A1 (en) 2022-03-03
TWI610672B (zh) 2018-01-11
JP2014501770A (ja) 2014-01-23
ES2751920T3 (es) 2020-04-02
SI2661261T1 (sl) 2019-11-29
NZ612420A (en) 2015-05-29
US12071402B2 (en) 2024-08-27
WO2012093161A1 (en) 2012-07-12
KR102166885B1 (ko) 2020-10-19
MY161162A (en) 2017-04-14
CL2013001979A1 (es) 2013-11-22
GT201300178A (es) 2014-12-30
KR101951966B1 (ko) 2019-02-25
JO3619B1 (ar) 2020-08-27
MX371290B (es) 2020-01-24
EP2661261B1 (en) 2019-07-31
EP3590507A1 (en) 2020-01-08
US20200199069A1 (en) 2020-06-25
AU2012204835A1 (en) 2013-08-01
MX2013007909A (es) 2013-08-29
TWI583380B (zh) 2017-05-21
US20130273161A1 (en) 2013-10-17
TW201609092A (zh) 2016-03-16
EA201391018A1 (ru) 2013-11-29
UA114283C2 (uk) 2017-05-25
BR112013017302B1 (pt) 2021-12-07
KR20190025727A (ko) 2019-03-11
HRP20191842T1 (hr) 2019-12-27
AR124662A2 (es) 2023-04-19
KR20140037815A (ko) 2014-03-27
AU2012204835B2 (en) 2015-07-09
PT2661261T (pt) 2019-10-25
EA026144B9 (ru) 2021-10-26
BR112013017302A2 (pt) 2016-10-25
PE20140216A1 (es) 2014-03-01
MX357304B (es) 2018-07-04
CN103458877A (zh) 2013-12-18
ZA201304465B (en) 2014-02-26
SG191286A1 (en) 2013-07-31

Similar Documents

Publication Publication Date Title
IL227094B (en) Immunosuppressive preparations
HRP20181896T1 (hr) Farmaceutske formulacije
EP2701734A4 (en) LIPOSOMAL FORMULATIONS
GB201111438D0 (en) Formulation
ZA201309221B (en) Formulation
ZA201306016B (en) Bendamustine formulations
HK1197193A1 (en) Sunscreen formulations
IL229700A0 (en) Dronvir formulations
GB201114725D0 (en) Ophthalmic formulations
EP2765992A4 (en) FOAM FORMULATIONS
ZA201402456B (en) Formulation
GB201110278D0 (en) Formulations
EP2782585A4 (en) ANTIVIRAL PREPARATIONS
GB201106958D0 (en) Formulation
GB201111578D0 (en) Pharmeutical formulations
GB201111013D0 (en) Formulations
GB201107626D0 (en) Formulations
GB201107627D0 (en) Formulations
GB201105410D0 (en) Formulations
GB201105360D0 (en) Formulations
GB201104049D0 (en) Formulations
GB201104048D0 (en) Formulations
GB201102795D0 (en) Formulations
GB201104284D0 (en) Formulation
GB201103769D0 (en) Cosmetic formulations