BR112012031667A2 - composição - Google Patents

composição

Info

Publication number
BR112012031667A2
BR112012031667A2 BR112012031667A BR112012031667A BR112012031667A2 BR 112012031667 A2 BR112012031667 A2 BR 112012031667A2 BR 112012031667 A BR112012031667 A BR 112012031667A BR 112012031667 A BR112012031667 A BR 112012031667A BR 112012031667 A2 BR112012031667 A2 BR 112012031667A2
Authority
BR
Brazil
Prior art keywords
composition
Prior art date
Application number
BR112012031667A
Other languages
English (en)
Inventor
Daniel E Dobry
David K Lyon
David T Vodak
Dwayne T Friesen
Warren K Miller
William B Caldwell
Original Assignee
Dow Global Technologies Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44627135&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112012031667(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Global Technologies Llc filed Critical Dow Global Technologies Llc
Publication of BR112012031667A2 publication Critical patent/BR112012031667A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08BPOLYSACCHARIDES; DERIVATIVES THEREOF
    • C08B13/00Preparation of cellulose ether-esters
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08LCOMPOSITIONS OF MACROMOLECULAR COMPOUNDS
    • C08L1/00Compositions of cellulose, modified cellulose or cellulose derivatives
    • C08L1/08Cellulose derivatives
    • C08L1/32Cellulose ether-esters

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Inorganic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Polymers & Plastics (AREA)
  • Organic Chemistry (AREA)
  • Materials Engineering (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BR112012031667A 2010-06-14 2011-06-13 composição BR112012031667A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35452510P 2010-06-14 2010-06-14
PCT/US2011/040222 WO2011159626A1 (en) 2010-06-14 2011-06-13 Hydroxypropyl methyl cellulose acetate succinate with enhanced acetate and succinate substitution

Publications (1)

Publication Number Publication Date
BR112012031667A2 true BR112012031667A2 (pt) 2016-11-08

Family

ID=44627135

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012031667A BR112012031667A2 (pt) 2010-06-14 2011-06-13 composição

Country Status (11)

Country Link
US (1) US9040033B2 (pt)
EP (1) EP2579896B1 (pt)
JP (1) JP5792807B2 (pt)
KR (1) KR101807338B1 (pt)
CN (1) CN103153343B (pt)
BR (1) BR112012031667A2 (pt)
CA (1) CA2801712A1 (pt)
CO (1) CO6660473A2 (pt)
IL (1) IL223607A (pt)
MX (1) MX2012014849A (pt)
WO (1) WO2011159626A1 (pt)

Families Citing this family (50)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10026698A1 (de) 2000-05-30 2001-12-06 Basf Ag Selbstemulgierende Wirkstoffformulierung und Verwendung dieser Formulierung
US8377952B2 (en) 2003-08-28 2013-02-19 Abbott Laboratories Solid pharmaceutical dosage formulation
US8025899B2 (en) 2003-08-28 2011-09-27 Abbott Laboratories Solid pharmaceutical dosage form
US20140088164A1 (en) 2010-11-24 2014-03-27 Rib-X Pharmaceuticals, Inc. Pharmaceutical Compositions
EP2802354A4 (en) * 2012-01-09 2015-07-29 Virginia Tech Intell Prop CELLULOSE DERIVATIVES FOR INHIBITING THE CRYSTALLIZATION OF MEDIALLY SOLUBLE DRUGS IN WATER
KR102041766B1 (ko) * 2012-03-27 2019-11-07 다우 글로벌 테크놀로지스 엘엘씨 셀룰로스 에테르의 에스테르의 제조방법
WO2013154607A1 (en) 2012-04-11 2013-10-17 Dow Global Technologies Llc Esterified cellulose ethers having a specific substituent distribution
CN102807625A (zh) * 2012-08-23 2012-12-05 浙江中维药业有限公司 一种醋酸羟丙甲纤维素琥珀酸酯的制备方法
US10730957B2 (en) 2012-08-24 2020-08-04 Dow Global Technologies Llc Process of preparing an esterified cellulose ether in the presence of an alkali metal carboxylate and an aliphatic carboxylic acid
BR112015002055A2 (pt) * 2012-08-24 2017-07-04 Dow Global Technologies Llc acetato succinato de hidroxialquil metil celulose, composição, dispersão sólida, processo para produzir uma dispersão sólida, forma de dosagem e cápsula de envoltório
US20150203595A1 (en) * 2012-08-24 2015-07-23 Dow Global Technologies Llc Process for preparing an ester of a cellulose ether in the presence of an alkali metal carboxylate
WO2014031447A1 (en) 2012-08-24 2014-02-27 Dow Global Technologies Llc Process for preparing an ester of a cellulose ether in the presence of an aliphatic carboxylic acid
CN104736572B (zh) 2012-08-24 2017-09-05 陶氏环球技术有限责任公司 部分交联的酯化纤维素醚
EP2961775B1 (en) 2013-03-01 2020-04-08 Hercules LLC Pharmaceutical compositions with enhanced performance and improved processability
WO2014137777A1 (en) 2013-03-07 2014-09-12 Dow Global Technologies Llc Novel esterified cellulose ethers of low viscosity
US20150368365A1 (en) * 2013-03-07 2015-12-24 Dow Global Technologies Llc Novel esterified cellulose ethers of low viscosity and high molecular weight
WO2014137778A1 (en) 2013-03-07 2014-09-12 Dow Global Technologies Llc Novel esterified cellulose ethers of very low viscosity
US9890220B2 (en) * 2013-03-07 2018-02-13 Dow Global Technologies Llc Esterified cellulose ethers of very high molecular weight
JP6306691B2 (ja) 2013-05-14 2018-04-04 ダウ グローバル テクノロジーズ エルエルシー ジカルボン酸を用いたエステル化セルロースエーテル
KR101918327B1 (ko) * 2013-06-03 2018-11-13 신에쓰 가가꾸 고교 가부시끼가이샤 가열 용융 압출용 조성물 및 이를 이용한 가열 용융 압출 성형물의 제조 방법
CN105829352B (zh) 2013-09-23 2018-04-10 陶氏环球技术有限责任公司 用于从反应产物混合物中回收酯化纤维素醚的方法
KR102286952B1 (ko) * 2013-12-31 2021-08-09 롯데정밀화학 주식회사 입도분포가 조절된 히드록시프로필 메틸셀룰로오스 아세테이트 숙시네이트(hpmcas) 입자의 제조방법 및 hpmcas 분말
US10759873B2 (en) 2014-02-20 2020-09-01 Dow Global Technologies Llc Esterified cellulose ethers of high molecular weight and homogeneity
KR20170045249A (ko) * 2014-08-27 2017-04-26 다우 글로벌 테크놀로지스 엘엘씨 낮은 아세톤-불용성 함량의 에스테르화된 셀룰로오스 에테르
AU2015317358A1 (en) * 2014-09-19 2017-04-27 Board Of Regents, The University Of Texas System Methods of preparing extrudates
CN104311674A (zh) * 2014-10-17 2015-01-28 广东东阳光药业有限公司 一种混合酯的制备方法
CN107074980A (zh) * 2014-10-31 2017-08-18 陶氏环球技术有限责任公司 制备纤维素醚的酯的方法
CN107074979B (zh) * 2014-10-31 2019-07-19 陶氏环球技术有限责任公司 用于产生乙酸纤维素醚丁二酸酯的方法
WO2016069343A1 (en) 2014-10-31 2016-05-06 Dow Global Technologies Llc Efficient process for preparing an ester of a cellulose ether
JP6203702B2 (ja) 2014-11-18 2017-09-27 信越化学工業株式会社 ヒプロメロース酢酸エステルコハク酸エステルを用いたスプレードライ用溶液及び固体分散体の製造方法
JP6295380B2 (ja) * 2015-03-16 2018-03-14 ダウ グローバル テクノロジーズ エルエルシー 脂肪族カルボン酸の存在下でエステル化セルロースエーテルを調製するためのプロセス
KR20170128350A (ko) * 2015-03-16 2017-11-22 다우 글로벌 테크놀로지스 엘엘씨 에스테르화된 셀룰로오스 에테르의 수용액
KR20170128371A (ko) * 2015-03-16 2017-11-22 다우 글로벌 테크놀로지스 엘엘씨 수용성 에스테르화된 셀룰로오스 에테르
BR112017018367A2 (pt) * 2015-03-16 2018-04-10 Dow Global Technologies Llc gelificação de éteres de celulose esterificados
WO2016148977A1 (en) 2015-03-16 2016-09-22 Dow Global Technologies Llc Water-soluble esterified cellulose ethers having a low degree of neutralization
JP6725534B2 (ja) 2015-05-15 2020-07-22 ダウ グローバル テクノロジーズ エルエルシー 極めて高い分子量及び低い粘度のエステル化セルロースエーテルの生成プロセス
BR112017023845A2 (pt) 2015-05-15 2018-07-31 Dow Global Technologies Llc processo de preparação de um éter de celulose esterificado de peso molecular elevado
EP3328899B1 (en) * 2015-07-28 2019-06-19 Dow Global Technologies LLC Process for producing dispersion of esterified cellulose ether
WO2017058973A1 (en) * 2015-10-02 2017-04-06 Dow Global Technologies Llc Aqueous composition comprising dispersed esterified cellulose ether
CN108348466A (zh) * 2015-12-08 2018-07-31 陶氏环球技术有限责任公司 包含纤维素醚和水溶性酯化纤维素醚的组合物
US9884922B2 (en) * 2016-03-11 2018-02-06 Shin-Etsu Chemical Co., Ltd. Hypromellose acetate succinate, method for producing the same and composition containing the same
AU2017248828A1 (en) 2016-04-15 2018-11-01 Janssen Sciences Ireland Uc Combinations and methods comprising a capsid assembly inhibitor
GB201609222D0 (en) 2016-05-25 2016-07-06 F2G Ltd Pharmaceutical formulation
KR20190069446A (ko) * 2016-10-18 2019-06-19 다우 글로벌 테크놀로지스 엘엘씨 에스터화된 셀룰로스 에터를 제조하는 효율적인 공정
US10888525B2 (en) * 2016-11-02 2021-01-12 Shin-Etsu Chemical Co., Ltd. Hypromellose acetate succinate and method for producing the same
MX2019010712A (es) * 2017-03-17 2019-10-21 Dow Global Technologies Llc Proceso para recuperar un eter de celulosa esterificado a partir de una mezcla de producto de reaccion.
BR112020007972A2 (pt) * 2017-10-27 2020-10-20 Plexxikon, Inc. formulações de composto que modula quinases
EA202092171A1 (ru) 2018-03-14 2020-12-01 Янссен Сайенсиз Айрлэнд Анлимитед Компани Схема дозирования модулятора сборки капсида
US11819503B2 (en) 2019-04-23 2023-11-21 F2G Ltd Method of treating coccidioides infection
CN115651085B (zh) * 2022-11-14 2023-11-17 乳源东阳光药业有限公司 一种醋酸羟丙甲纤维素琥珀酸酯的纯化方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4226981A (en) 1977-09-28 1980-10-07 Shin-Etsu Chemical Co., Ltd. Ether-ester derivatives of cellulose and their applications
JP2528706B2 (ja) 1988-05-30 1996-08-28 ゼリア新薬工業株式会社 ジヒドロピリジン化合物の製剤組成物
EP1741424B1 (en) * 1997-08-11 2018-10-03 Pfizer Products Inc. Solid pharmaceutical dispersions with enhanced bioavailabilty
EP0901786B1 (en) * 1997-08-11 2007-06-13 Pfizer Products Inc. Solid pharmaceutical dispersions with enhanced bioavailability
WO2002038126A2 (en) * 2000-11-08 2002-05-16 Aeromatic-Fielder Ag A process for production of particles for pharmaceutical compositions having increased bioavailability
WO2005115330A2 (en) * 2004-05-28 2005-12-08 Pfizer Products Inc. Pharmaceutical compositions with enhanced performance
WO2007029660A1 (ja) * 2005-09-06 2007-03-15 Astellas Pharma Inc. 腸溶性基剤が表面に吸着した難溶性薬物の微小粒子
EP1942872A2 (en) * 2005-11-04 2008-07-16 Eastman Chemical Company Carboxyalkylcellulose esters for administration of poorly soluble pharmaceutically active agents

Also Published As

Publication number Publication date
CN103153343A (zh) 2013-06-12
WO2011159626A1 (en) 2011-12-22
US9040033B2 (en) 2015-05-26
JP2013532151A (ja) 2013-08-15
IL223607A (en) 2016-04-21
CO6660473A2 (es) 2013-04-30
CN103153343B (zh) 2015-02-11
US20130102691A1 (en) 2013-04-25
KR101807338B1 (ko) 2018-01-10
CA2801712A1 (en) 2011-12-22
MX2012014849A (es) 2013-05-01
EP2579896A1 (en) 2013-04-17
JP5792807B2 (ja) 2015-10-14
KR20130109102A (ko) 2013-10-07
EP2579896B1 (en) 2016-07-20

Similar Documents

Publication Publication Date Title
BR112012031667A2 (pt) composição
DK2640893T4 (da) Sammensætninger
BR112012032683A2 (pt) composição
BR112012028556A2 (pt) Indóis
DE102011100241A8 (de) Nitridhalbleiterbauteil
DK3225404T3 (da) Fluidpatron
CR20130111A (es) Triazina-oxidiazoles
DE10170954T8 (de) Mikrowellendruckgarer
DE112011104226A5 (de) Käfigmutter
DE102011117046A8 (de) Doppelkupplungswindungsgetriebe
BR112012032980A2 (pt) composição
DE112011101226A5 (de) Linearwegmesssystem
DE112011102080A5 (de) Kupplungszentralausrücker
DK2539163T3 (da) Dækventil
DK2442899T3 (da) Rotorskive
DE112011102711A5 (de) Hydrostataktor
DK2448659T3 (da) Rotorskive
DK2447426T3 (da) Vaske-WC
DK2553004T3 (da) Sammensatte materialer
DE102010019119B8 (de) Cuttermesser
DE112010005518A5 (de) Dichtungsmanchette
DE102010038420A8 (de) Reinigungungsvorrichtung
DK2596072T3 (da) Bor-forbindelses-suspension
DK2521486T3 (da) Palpometer
CO6801789A2 (es) N-hetarilmetil pirazolilcarboxamidas

Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06T Formal requirements before examination [chapter 6.20 patent gazette]
B11E Dismissal acc. art. 34 of ipl - requirements for examination incomplete
B11T Dismissal of application maintained [chapter 11.20 patent gazette]