BR112012012584A2 - "processo para preparar sais de 4,5-diidroisoxazol-3-tiocarboxamidina 5,5-dissubstituídos de fórmula (i)" - Google Patents

"processo para preparar sais de 4,5-diidroisoxazol-3-tiocarboxamidina 5,5-dissubstituídos de fórmula (i)"

Info

Publication number
BR112012012584A2
BR112012012584A2 BR112012012584A BR112012012584A BR112012012584A2 BR 112012012584 A2 BR112012012584 A2 BR 112012012584A2 BR 112012012584 A BR112012012584 A BR 112012012584A BR 112012012584 A BR112012012584 A BR 112012012584A BR 112012012584 A2 BR112012012584 A2 BR 112012012584A2
Authority
BR
Brazil
Prior art keywords
dihydroisoxazole
disubstituted
preparing
formula
thiocarboxamidine salts
Prior art date
Application number
BR112012012584A
Other languages
English (en)
Other versions
BR112012012584B1 (pt
Inventor
Timo Frassetto
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of BR112012012584A2 publication Critical patent/BR112012012584A2/pt
Publication of BR112012012584B1 publication Critical patent/BR112012012584B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BR112012012584-2A 2009-11-26 2009-11-26 A process for preparing 5,5-disubstituted 4,5-dihydroisoxazol-3-thiocarboxamidine salts BR112012012584B1 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/EP2009/065925 WO2011063842A1 (de) 2009-11-26 2009-11-26 Verfahren zur herstellung 5,5-disubstituierter 4,5-dihydroisoxazol-3-thiocarboxamidin-salze

Publications (2)

Publication Number Publication Date
BR112012012584A2 true BR112012012584A2 (pt) 2015-09-08
BR112012012584B1 BR112012012584B1 (pt) 2017-10-31

Family

ID=42357887

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012012584-2A BR112012012584B1 (pt) 2009-11-26 2009-11-26 A process for preparing 5,5-disubstituted 4,5-dihydroisoxazol-3-thiocarboxamidine salts

Country Status (13)

Country Link
US (1) US8921572B2 (pt)
EP (1) EP2504322B1 (pt)
JP (1) JP5650237B2 (pt)
KR (1) KR20120086364A (pt)
CN (1) CN102666502B (pt)
AU (1) AU2009355793A1 (pt)
BR (1) BR112012012584B1 (pt)
CA (1) CA2781404A1 (pt)
DK (1) DK2504322T3 (pt)
ES (1) ES2466322T3 (pt)
IL (1) IL219796A (pt)
MX (1) MX2012005884A (pt)
WO (1) WO2011063842A1 (pt)

Families Citing this family (28)

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JP6525991B2 (ja) * 2013-07-17 2019-06-05 サノフイＳａｎｏｆｉ 薬物送達デバイス用のアセンブリおよびその動作方法
EP3476594A1 (en) 2017-10-24 2019-05-01 Renolit SE Laminate structure for biocompatible barrier packaging
EP3476593A1 (en) 2017-10-24 2019-05-01 Renolit SE Laminate structure for barrier packaging
WO2019131715A1 (ja) * 2017-12-27 2019-07-04 クミアイ化学工業株式会社 チオカルボキサミジン塩化合物の製造方法
WO2020240392A1 (en) * 2019-05-24 2020-12-03 Pi Industries Limited Process for preparation of pyroxasulfone
JPWO2020251006A1 (pt) * 2019-06-14 2020-12-17
WO2021019537A1 (en) * 2019-07-30 2021-02-04 Adama Agan Ltd. Process and intermediates for the preparation of pyroxasulfone
CA3156419C (en) * 2019-10-31 2023-12-12 Yukio Uchida Process for producing herbicide and intermediate thereof
WO2021085550A1 (ja) 2019-11-01 2021-05-06 ユニマテック株式会社 含フッ素ピリミジン化合物およびその製造方法
AR121018A1 (es) * 2020-01-15 2022-04-06 Adama Agan Ltd Forma en estado sólido de piroxasulfona
BR112022017794A2 (pt) * 2020-03-05 2022-10-25 Adama Agan Ltd Processo e intermediários para a preparação de piroxassulfona
CN111393427B (zh) * 2020-04-30 2021-11-30 安徽久易农业股份有限公司 一种砜吡草唑的合成方法
CN113754647B (zh) * 2020-06-02 2023-02-17 山东润博生物科技有限公司 一种砜吡草唑及其中间体的合成方法
CN113135867B (zh) * 2020-06-02 2022-09-23 山东润博生物科技有限公司 S-（5,5-二甲基-4,5-二氢异恶唑-3-基）乙硫酸乙酯及其合成方法和应用
CN111574511A (zh) * 2020-06-28 2020-08-25 安徽久易农业股份有限公司 一种砜吡草唑的合成方法及其应用
EP4177244A3 (en) * 2020-07-10 2023-08-09 Adama Agan Ltd. Process and intermediates for the preparation of pyroxasulfone and fenoxasulfone
CN114315747A (zh) * 2020-09-30 2022-04-12 山东润博生物科技有限公司 一种5,5-二甲基异噁唑烷-3-硫酮的制备方法
CN112645894B (zh) * 2020-11-30 2022-04-15 江苏中旗科技股份有限公司 制备砜吡草唑中间体5,5-二甲基-4,5-二氢异恶唑-3-硫代甲脒盐酸盐的方法
CN114644602A (zh) * 2020-12-17 2022-06-21 帕潘纳(北京)科技有限公司 二氢异噁唑类化合物的制备方法
WO2022137370A1 (ja) * 2020-12-23 2022-06-30 クミアイ化学工業株式会社 スルホン誘導体の製造方法
GB2603771A (en) * 2021-02-11 2022-08-17 Rotam Agrochem Int Co Ltd Novel crystalline form of pyroxa-sulfone, methods for its preparation and use of the same
JPWO2022191292A1 (pt) * 2021-03-11 2022-09-15
CN114213402A (zh) * 2021-12-01 2022-03-22 芮城华农生物化学有限公司 一种砜吡草唑亚稳态、稳定态晶型、制备方法及应用
CN114716428B (zh) * 2022-05-06 2024-02-06 山东潍坊润丰化工股份有限公司 制备砜吡草唑中间体的方法
CN114989157A (zh) * 2022-06-28 2022-09-02 安徽久易农业股份有限公司 一种砜吡草唑的晶型a及其制备方法和应用
CN116514792B (zh) * 2023-07-04 2023-10-27 潍坊新绿化工有限公司 一种砜吡草唑的制备方法
CN118221663A (zh) * 2024-05-24 2024-06-21 吉林凯莱英医药化学有限公司 砜吡草唑的连续化合成方法
CN118255757A (zh) * 2024-05-28 2024-06-28 吉林凯莱英医药化学有限公司 砜吡草唑的连续化合成方法

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Publication number Priority date Publication date Assignee Title
WO2000050410A1 (fr) 1999-02-25 2000-08-31 Nippon Soda Co., Ltd. Composes d'isoxazoline et leurs procedes de preparation
EP1203768B1 (en) 1999-08-10 2006-03-01 Kumiai Chemical Industry Co., Ltd. Isoxazoline derivatives and herbicides containing the same as the active ingredient
JP4465133B2 (ja) 2001-02-08 2010-05-19 クミアイ化学工業株式会社 イソオキサゾリン誘導体及びこれを有効成分とする除草剤
JP4621939B2 (ja) * 2004-03-31 2011-02-02 イハラケミカル工業株式会社 ５−ヒドロキシ−４−チオメチルピラゾール化合物の製造方法
JP2008001597A (ja) 2004-10-06 2008-01-10 Ihara Chem Ind Co Ltd ３−ブロモ−５，５−ジメチル−４，５−ジヒドロイソオキサゾールの製造方法
BRPI0519138B1 (pt) 2004-12-20 2016-05-10 Ihara Chemical Ind Co método para produção de um composto do sal (4,5- diidroisoxazol-3-il) tiocarboxamidina, e compostos do sal (4,5-diidroisoxazol-3-il)tiocarboxamidina
GB0603891D0 (en) 2006-02-27 2006-04-05 Syngenta Ltd Novel herbicides
WO2011063843A1 (de) * 2009-11-26 2011-06-03 Basf Se Verfahren zur herstellung 5,5-disubstituierter 2-isoxazoline

Also Published As

Publication number Publication date
US8921572B2 (en) 2014-12-30
IL219796A (en) 2015-09-24
JP5650237B2 (ja) 2015-01-07
DK2504322T3 (da) 2014-06-16
KR20120086364A (ko) 2012-08-02
CA2781404A1 (en) 2011-06-03
EP2504322A1 (de) 2012-10-03
IL219796A0 (en) 2012-07-31
MX2012005884A (es) 2012-06-19
WO2011063842A1 (de) 2011-06-03
ES2466322T3 (es) 2014-06-10
BR112012012584B1 (pt) 2017-10-31
JP2013512201A (ja) 2013-04-11
AU2009355793A1 (en) 2012-07-05
CN102666502B (zh) 2015-01-07
EP2504322B1 (de) 2014-04-02
US20120264947A1 (en) 2012-10-18
CN102666502A (zh) 2012-09-12

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Legal Events

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B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 3A ANUIDADE

B08G Application fees: restoration [chapter 8.7 patent gazette]
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]