BR112012011780A2 - peptídeo linear,composição farmacêutica,métodopara tratamento de umadoença,indicação,condição ou sídrome mediadsa por receptor de melanocortina emum mamífero humano ou não humano e método para tratamento de uma condição responsiva ás alterações em função de receptor de melanocortina em um mamifero humano ou não humano - Google Patents
peptídeo linear,composição farmacêutica,métodopara tratamento de umadoença,indicação,condição ou sídrome mediadsa por receptor de melanocortina emum mamífero humano ou não humano e método para tratamento de uma condição responsiva ás alterações em função de receptor de melanocortina em um mamifero humano ou não humanoInfo
- Publication number
- BR112012011780A2 BR112012011780A2 BR112012011780A BR112012011780A BR112012011780A2 BR 112012011780 A2 BR112012011780 A2 BR 112012011780A2 BR 112012011780 A BR112012011780 A BR 112012011780A BR 112012011780 A BR112012011780 A BR 112012011780A BR 112012011780 A2 BR112012011780 A2 BR 112012011780A2
- Authority
- BR
- Brazil
- Prior art keywords
- human
- treating
- melanocortin receptor
- condition
- human mammal
- Prior art date
Links
- 102000004378 Melanocortin Receptors Human genes 0.000 title 2
- 108090000950 Melanocortin Receptors Proteins 0.000 title 2
- 201000010099 disease Diseases 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 1
- 230000001404 mediated effect Effects 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 108090000765 processed proteins & peptides Proteins 0.000 title 1
- 208000011580 syndromic disease Diseases 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/68—Melanocyte-stimulating hormone [MSH]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Endocrinology (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Toxicology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US26348609P | 2009-11-23 | 2009-11-23 | |
| PCT/US2010/057700 WO2011063367A1 (en) | 2009-11-23 | 2010-11-23 | Melanocortin-1 receptor-specific linear peptides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112012011780A2 true BR112012011780A2 (pt) | 2019-09-24 |
Family
ID=44060072
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112012011780A BR112012011780A2 (pt) | 2009-11-23 | 2010-11-23 | peptídeo linear,composição farmacêutica,métodopara tratamento de umadoença,indicação,condição ou sídrome mediadsa por receptor de melanocortina emum mamífero humano ou não humano e método para tratamento de uma condição responsiva ás alterações em função de receptor de melanocortina em um mamifero humano ou não humano |
Country Status (13)
| Country | Link |
|---|---|
| US (3) | US8933194B2 (https=) |
| EP (1) | EP2504351A4 (https=) |
| JP (1) | JP2013511554A (https=) |
| KR (1) | KR20120102716A (https=) |
| CN (1) | CN102712674A (https=) |
| AU (1) | AU2010321739A1 (https=) |
| BR (1) | BR112012011780A2 (https=) |
| CA (1) | CA2781405A1 (https=) |
| EA (1) | EA201290295A1 (https=) |
| IL (1) | IL219946A0 (https=) |
| MX (1) | MX2012005859A (https=) |
| WO (1) | WO2011063367A1 (https=) |
| ZA (1) | ZA201203331B (https=) |
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| WO2011063366A1 (en) * | 2009-11-23 | 2011-05-26 | Palatin Technologies, Inc. | Melanocortin-1 receptor-specific cyclic peptides |
| IT1404931B1 (it) * | 2010-06-11 | 2013-12-09 | Medivis S R L | Composizioni oftalmiche per la somministrazione di principi attivi liposolubili . |
| US9441013B2 (en) | 2011-05-17 | 2016-09-13 | H. Lee Moffitt Cancer Center And Research Institute, Inc. | Melanocortin 1 receptor ligands and methods of use |
| US9290539B2 (en) | 2011-05-17 | 2016-03-22 | The Arizona Board Of Regents On Behalf Of The University Of Arizona | Melanotropin ligands for skin care |
| US9402877B2 (en) * | 2011-11-04 | 2016-08-02 | Xion Pharmaceuticals Corporation | Methods and compositions for oral administration of melanocortin receptor agonist compounds |
| EP2814501A4 (en) | 2012-03-13 | 2016-03-02 | Tensive Controls Inc | MELANOCORTINANALOGA WITH INCREASED EFFECTIVENESS AND TRANSPORTATION OF THEREOF |
| US9814755B2 (en) | 2014-06-10 | 2017-11-14 | The Arizona Board Of Regents On Behalf Of The University Of Arizona | Methods for the treatment of depression and anxiety |
| US9821023B2 (en) | 2014-06-10 | 2017-11-21 | The Arizona Board Of Regents On Behalf Of The University Of Arizona | Methods for the treatment of central nervous system (CNS) disorders and mood disorders |
| US20170022252A1 (en) | 2014-06-10 | 2017-01-26 | The Arizona Board Of Regents On Behalf Of The University Of Arizona | Novel modulators of melanocortin receptors |
| CN104436159A (zh) * | 2014-12-09 | 2015-03-25 | 天津医科大学眼科医院 | 一种新型滴眼液对治疗干眼的用途 |
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| EP3328372A4 (en) | 2015-07-28 | 2019-03-20 | University Of Iowa Research Foundation | COMPOSITIONS AND METHOD FOR THE TREATMENT OF CANCER |
| US10550157B2 (en) | 2015-10-16 | 2020-02-04 | Arizona Board Of Regent On Behalf Of The University Of Arizona | Compositions and methods for treating central nervous system (CNS) disorders and mood disorders |
| AU2017281940C1 (en) | 2016-06-24 | 2024-11-07 | University Of Iowa Research Foundation | Compositions and methods of treating melanoma |
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| US11819520B2 (en) * | 2018-02-23 | 2023-11-21 | Duke University | Cultured thymus tissue transplantation promotes donor-specific tolerance to allogeneic solid organ transplants |
| US11529335B2 (en) | 2020-07-31 | 2022-12-20 | University Of Iowa Research Foundation | Compositions and methods for treating cancer |
| WO2023091689A1 (en) | 2021-11-19 | 2023-05-25 | University Of Iowa Research Foundation | Combined use of mcr1-directed radiotherapy and immune checkpoint inhibition in the treatment of melanoma |
| US20260049105A1 (en) * | 2022-08-18 | 2026-02-19 | Arizona Board Of Regents On Behalf Of The University Of Arizona | Selective mc4r ligand for treating obesity and cognitive loss |
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-
2010
- 2010-11-23 JP JP2012540142A patent/JP2013511554A/ja not_active Withdrawn
- 2010-11-23 CA CA 2781405 patent/CA2781405A1/en not_active Abandoned
- 2010-11-23 AU AU2010321739A patent/AU2010321739A1/en not_active Abandoned
- 2010-11-23 CN CN2010800610676A patent/CN102712674A/zh active Pending
- 2010-11-23 KR KR20127016182A patent/KR20120102716A/ko not_active Withdrawn
- 2010-11-23 BR BR112012011780A patent/BR112012011780A2/pt not_active IP Right Cessation
- 2010-11-23 MX MX2012005859A patent/MX2012005859A/es not_active Application Discontinuation
- 2010-11-23 EA EA201290295A patent/EA201290295A1/ru unknown
- 2010-11-23 WO PCT/US2010/057700 patent/WO2011063367A1/en not_active Ceased
- 2010-11-23 EP EP10832345.2A patent/EP2504351A4/en not_active Withdrawn
-
2012
- 2012-05-08 ZA ZA2012/03331A patent/ZA201203331B/en unknown
- 2012-05-16 US US13/472,955 patent/US8933194B2/en active Active
- 2012-05-23 IL IL219946A patent/IL219946A0/en unknown
-
2014
- 2014-12-30 US US14/585,686 patent/US9580466B2/en active Active
-
2017
- 2017-02-02 US US15/422,850 patent/US10106578B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| AU2010321739A1 (en) | 2012-05-31 |
| US10106578B2 (en) | 2018-10-23 |
| KR20120102716A (ko) | 2012-09-18 |
| US20120225831A1 (en) | 2012-09-06 |
| MX2012005859A (es) | 2012-12-17 |
| US20150119341A1 (en) | 2015-04-30 |
| EP2504351A1 (en) | 2012-10-03 |
| US8933194B2 (en) | 2015-01-13 |
| WO2011063367A1 (en) | 2011-05-26 |
| US9580466B2 (en) | 2017-02-28 |
| CN102712674A (zh) | 2012-10-03 |
| EA201290295A1 (ru) | 2013-01-30 |
| EP2504351A4 (en) | 2013-10-30 |
| US20170145056A1 (en) | 2017-05-25 |
| JP2013511554A (ja) | 2013-04-04 |
| ZA201203331B (en) | 2013-07-31 |
| IL219946A0 (en) | 2012-07-31 |
| CA2781405A1 (en) | 2011-05-26 |
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