BR0313523A - Intermediários do esteróide 5-androsten-3(beta)-ol e processos para a sua preparação - Google Patents

Intermediários do esteróide 5-androsten-3(beta)-ol e processos para a sua preparação

Info

Publication number
BR0313523A
BR0313523A BR0313523-3A BR0313523A BR0313523A BR 0313523 A BR0313523 A BR 0313523A BR 0313523 A BR0313523 A BR 0313523A BR 0313523 A BR0313523 A BR 0313523A
Authority
BR
Brazil
Prior art keywords
androsten
processes
preparation
steroid
intermediates
Prior art date
Application number
BR0313523-3A
Other languages
English (en)
Portuguese (pt)
Inventor
Michael J White
Peter G M Wuts
Doris Beck
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of BR0313523A publication Critical patent/BR0313523A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0011—Androstane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/001—Lactones
    • C07J21/003—Lactones at position 17

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BR0313523-3A 2002-08-16 2003-03-21 Intermediários do esteróide 5-androsten-3(beta)-ol e processos para a sua preparação BR0313523A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40399002P 2002-08-16 2002-08-16
US41529302P 2002-10-01 2002-10-01
PCT/US2003/007791 WO2004016640A2 (en) 2002-08-16 2003-03-21 5 ANDROSTEN-3β-OL STEROID INTERMEDIATES AND PROCESSES FOR THEIR PREPARATION

Publications (1)

Publication Number Publication Date
BR0313523A true BR0313523A (pt) 2005-06-28

Family

ID=31891414

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0313523-3A BR0313523A (pt) 2002-08-16 2003-03-21 Intermediários do esteróide 5-androsten-3(beta)-ol e processos para a sua preparação

Country Status (12)

Country Link
US (2) US20040034215A1 (enExample)
EP (1) EP1534732B1 (enExample)
JP (1) JP2006507369A (enExample)
AT (1) ATE339437T1 (enExample)
AU (1) AU2003285485A1 (enExample)
BR (1) BR0313523A (enExample)
CA (1) CA2495412A1 (enExample)
DE (1) DE60308388T2 (enExample)
ES (1) ES2271636T3 (enExample)
MX (1) MXPA05001857A (enExample)
TW (1) TW200406419A (enExample)
WO (1) WO2004016640A2 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ITMI20042338A1 (it) * 2004-12-06 2005-03-06 Ind Chimica Srl Processo per la preparazione di drospirenone
US8084446B2 (en) * 2005-04-26 2011-12-27 Eric Marchewitz Use of DHEA derivatives for enhancing physical performance
PL2527356T3 (pl) * 2005-07-21 2018-06-29 Bayer Intellectual Property Gmbh Sposób wytwarzania 3-okso-pregn-4-eno-21,17-karbolaktonów za pomocą wolnego od metali utleniania 17-(3-hydroksypropylo)-3,17- dihydroksyandrostanów
ATE403668T1 (de) 2005-07-21 2008-08-15 Bayer Schering Pharma Ag Verfahren zur herstellung von 3-oxo-pregn-4-en-21,17-carbolactonen durch die metallfreie oxidation von 17-(3-hydroxypropyl)-3,17- dihydroxyandrostanen
US7319154B2 (en) 2005-07-21 2008-01-15 Bayer Schering Pharma Ag Process for the production of 3-oxo-pregn-4-ene-21, 17-carbolactones by the metal free oxidation of 17-(3-hydroxypropyl)-3, 17-dihydroxyandrostanes
CN110331182A (zh) * 2019-08-06 2019-10-15 江苏远大仙乐药业有限公司 一种甾体中间体的生物转化制备方法
CN110885869A (zh) * 2019-12-24 2020-03-17 天津科技大学 一种利用微生物转化生产7α-羟基-脱氢表雄酮的方法
CN111057734A (zh) * 2019-12-24 2020-04-24 天津科技大学 一种甲基睾丸素高效转化生产11α-羟基-甲基睾丸素的方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3294646A (en) * 1963-10-23 1966-12-27 American Home Prod Microbiological hydroxylation of norsteroids using aspergillus ochraceus
DE2349022A1 (de) * 1973-09-26 1975-04-10 Schering Ag Neue d-homo-steroide
DK134348C (da) * 1973-11-30 1977-03-21 Schering Ag Analogifremgangsmade til fremstilling af d-homo-20-ketopregnaner
US4031074A (en) * 1974-09-02 1977-06-21 Akzona Incorporated Process for the preparation of 11β-hydroxy-18-alkyl-estrane compounds
IL48628A0 (en) * 1974-12-23 1976-02-29 Schering Ag D-homo-20-keto-pregnanes and process for their manufactur
US4054563A (en) * 1975-04-25 1977-10-18 Ciba-Geigy Corporation Process for the manufacture of spiro compounds of the steroid series
CH633562A5 (de) * 1976-12-10 1982-12-15 Schering Ag Verfahren zur herstellung neuer kortikoide.
US4336332A (en) * 1979-02-20 1982-06-22 Hoffmann-La Roche, Inc. Process for the manufacture of hydroxylated steroids
DE3042136A1 (de) * 1980-11-03 1982-06-09 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur herstellung von 3 (beta), 7 (beta) -dihydroxy- (delta) (pfeil hoch)5(pfeil hoch) -steroiden
US4559332A (en) * 1983-04-13 1985-12-17 Ciba Geigy Corporation 20-Spiroxanes and analogues having an open ring E, processes for their manufacture, and pharmaceutical preparations thereof
AU7978794A (en) * 1993-10-13 1995-05-04 Neurocrine Biosciences, Inc. 3,17-dihydroxy-3,7,16 and/or 17-methyl-androst-5-ene compounds, derivatives thereof, and their use
PT973791E (pt) * 1995-12-11 2007-09-26 Searle Llc Processo para a preparação de um composto epoxi
DE69620474T2 (de) * 1995-12-12 2002-11-14 Akzo Nobel N.V., Arnhem Mikrobielle 11alpha-hydroxylierung von steroiden
FR2771105A1 (fr) 1997-11-20 1999-05-21 Vitasterol Utilisation du fusarium monoliforme pour la preparation des derives 7alpha-hydroxyles de la dehydroepiandrosterone et de la pregnenolone

Also Published As

Publication number Publication date
JP2006507369A (ja) 2006-03-02
MXPA05001857A (es) 2005-06-03
WO2004016640A3 (en) 2004-07-08
CA2495412A1 (en) 2004-02-26
DE60308388T2 (de) 2007-09-20
US20040034215A1 (en) 2004-02-19
EP1534732A2 (en) 2005-06-01
US7002028B2 (en) 2006-02-21
ES2271636T3 (es) 2007-04-16
WO2004016640A2 (en) 2004-02-26
AU2003285485A1 (en) 2004-03-03
US20040220158A1 (en) 2004-11-04
ATE339437T1 (de) 2006-10-15
DE60308388D1 (de) 2006-10-26
TW200406419A (en) 2004-05-01
EP1534732B1 (en) 2006-09-13

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2069 DE 31/08/2010.